IN2014DN07762A - - Google Patents
Info
- Publication number
- IN2014DN07762A IN2014DN07762A IN7762DEN2014A IN2014DN07762A IN 2014DN07762 A IN2014DN07762 A IN 2014DN07762A IN 7762DEN2014 A IN7762DEN2014 A IN 7762DEN2014A IN 2014DN07762 A IN2014DN07762 A IN 2014DN07762A
- Authority
- IN
- India
- Prior art keywords
- solifenacin
- reacting
- salt
- prepare
- organic solvent
- Prior art date
Links
- FBOUYBDGKBSUES-VXKWHMMOSA-N solifenacin Chemical compound C1([C@H]2C3=CC=CC=C3CCN2C(O[C@@H]2C3CCN(CC3)C2)=O)=CC=CC=C1 FBOUYBDGKBSUES-VXKWHMMOSA-N 0.000 abstract 5
- 229960003855 solifenacin Drugs 0.000 abstract 5
- IOVVFSGCNWQFQT-UHFFFAOYSA-N bis(2,3,4,5,6-pentafluorophenyl) carbonate Chemical compound FC1=C(F)C(F)=C(F)C(F)=C1OC(=O)OC1=C(F)C(F)=C(F)C(F)=C1F IOVVFSGCNWQFQT-UHFFFAOYSA-N 0.000 abstract 2
- 239000003960 organic solvent Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- FSNYTEYOTCTPSO-SSDOTTSWSA-N (2r)-1-azabicyclo[2.2.2]octan-2-ol Chemical compound C1CN2[C@H](O)CC1CC2 FSNYTEYOTCTPSO-SSDOTTSWSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/49—Cinchonan derivatives, e.g. quinine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/41—Preparation of salts of carboxylic acids
- C07C51/412—Preparation of salts of carboxylic acids by conversion of the acids, their salts, esters or anhydrides with the same carboxylic acid part
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Urology & Nephrology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20120031492A KR101365849B1 (ko) | 2012-03-28 | 2012-03-28 | 솔리페나신 또는 그의 염의 제조방법 및 이에 사용되는 신규 중간체 |
| PCT/KR2013/002358 WO2013147458A1 (en) | 2012-03-28 | 2013-03-21 | Process of preparing solifenacin or salt thereof, and novel intermediate used in the process |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2014DN07762A true IN2014DN07762A (https=) | 2015-05-15 |
Family
ID=49260649
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN7762DEN2014 IN2014DN07762A (https=) | 2012-03-28 | 2013-03-21 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US9018379B1 (https=) |
| EP (1) | EP2831070A4 (https=) |
| JP (1) | JP5891334B2 (https=) |
| KR (1) | KR101365849B1 (https=) |
| CN (1) | CN104169280A (https=) |
| AU (1) | AU2013240842B2 (https=) |
| BR (1) | BR112014021223A2 (https=) |
| IN (1) | IN2014DN07762A (https=) |
| WO (1) | WO2013147458A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN116986986A (zh) * | 2023-07-19 | 2023-11-03 | 杭州国瑞生物科技有限公司 | 一种3-氧代-1-环丁烷羧酸中间体的合成方法 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO2005012I1 (no) | 1994-12-28 | 2005-06-06 | Debio Rech Pharma Sa | Triptorelin og farmasoytisk akseptable salter derav |
| US6664372B1 (en) * | 1996-03-20 | 2003-12-16 | The Scripps Research Institute | Azatide peptidomimetics |
| KR100669823B1 (ko) | 2001-02-20 | 2007-01-17 | 경동제약 주식회사 | 2-(4-클로로벤조일아미노)-3-[2(1ｈ)-퀴놀리논-4-일]프로피온산의 제조방법 및 그 중간체 |
| WO2004035577A2 (en) * | 2002-10-16 | 2004-04-29 | Gilead Sciences, Inc. | Pre-organized tricyclic integrase inhibitor compounds |
| GB0312426D0 (en) * | 2003-05-30 | 2003-07-09 | Albachem Ltd | Purification means |
| US20080287680A1 (en) | 2004-02-09 | 2008-11-20 | Astellas Pharma Inc. | Solifenacin Succinate-Containing Composition |
| JPWO2005087231A1 (ja) | 2004-03-16 | 2008-01-24 | アステラス製薬株式会社 | ソリフェナシン含有組成物 |
| WO2005117904A2 (en) * | 2004-04-14 | 2005-12-15 | Gilead Sciences, Inc. | Phosphonate analogs of hiv integrase inhibitor compounds |
| JP4803352B2 (ja) * | 2005-07-13 | 2011-10-26 | Ｊｓｒ株式会社 | アミノ酸−ｎ−カルボキシ無水物の製造方法 |
| EP1879867A2 (en) * | 2005-12-21 | 2008-01-23 | Teva Pharmaceutical Industries Ltd | Intermediates for preparing solifenacin |
| CA2670365A1 (en) * | 2006-11-22 | 2008-05-29 | Medichem S.A. | An improved process for the synthesis of solifenacin |
| JP2010523539A (ja) * | 2007-03-30 | 2010-07-15 | メディチェム ソシエダ アノニマ | ソリフェナシンの改良された合成法 |
| JP2009538362A (ja) * | 2007-07-13 | 2009-11-05 | テバ ファーマシューティカル インダストリーズ リミティド | ソリフェナシンの調製方法 |
| MX344559B (es) * | 2008-04-29 | 2016-12-20 | Ascendis Pharma As | Compuestos de hormona de crecimiento humana recombinante unidos al peg. |
| US8283470B2 (en) * | 2009-03-09 | 2012-10-09 | Megafine Pharma(P) Ltd. | Method for the preparation of solifenacin and intermediate thereof |
| US8178700B2 (en) * | 2009-05-04 | 2012-05-15 | International Business Machines Corporation | Method of preparing cyclic carbonates, cyclic carbamates, cyclic ureas, cyclic thiocarbonates, cyclic thiocarbamates, and cyclic dithiocarbonates |
| WO2011030139A1 (en) * | 2009-09-11 | 2011-03-17 | Astrazeneca Ab | 4- (pyrimidin-2-yl) -piperazine and 4- (pyrimidin-2-yl) -piperidine derivatives as gpr119 modulators |
-
2012
- 2012-03-28 KR KR20120031492A patent/KR101365849B1/ko active Active
-
2013
- 2013-03-21 CN CN201380016063.XA patent/CN104169280A/zh active Pending
- 2013-03-21 AU AU2013240842A patent/AU2013240842B2/en not_active Ceased
- 2013-03-21 US US14/382,529 patent/US9018379B1/en not_active Expired - Fee Related
- 2013-03-21 WO PCT/KR2013/002358 patent/WO2013147458A1/en not_active Ceased
- 2013-03-21 IN IN7762DEN2014 patent/IN2014DN07762A/en unknown
- 2013-03-21 EP EP13768214.2A patent/EP2831070A4/en not_active Withdrawn
- 2013-03-21 BR BR112014021223-6A patent/BR112014021223A2/pt not_active IP Right Cessation
- 2013-03-21 JP JP2015501582A patent/JP5891334B2/ja active Active
Also Published As
| Publication number | Publication date |
|---|---|
| JP5891334B2 (ja) | 2016-03-22 |
| KR101365849B1 (ko) | 2014-02-24 |
| AU2013240842A1 (en) | 2014-08-28 |
| US9018379B1 (en) | 2015-04-28 |
| BR112014021223A2 (pt) | 2020-10-27 |
| US20150112072A1 (en) | 2015-04-23 |
| AU2013240842B2 (en) | 2015-09-03 |
| EP2831070A1 (en) | 2015-02-04 |
| EP2831070A4 (en) | 2015-08-19 |
| JP2015510927A (ja) | 2015-04-13 |
| WO2013147458A1 (en) | 2013-10-03 |
| CN104169280A (zh) | 2014-11-26 |
| KR20130109609A (ko) | 2013-10-08 |
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