IN2012DN05171A - - Google Patents

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Publication number
IN2012DN05171A
IN2012DN05171A IN5171DEN2012A IN2012DN05171A IN 2012DN05171 A IN2012DN05171 A IN 2012DN05171A IN 5171DEN2012 A IN5171DEN2012 A IN 5171DEN2012A IN 2012DN05171 A IN2012DN05171 A IN 2012DN05171A
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India
Prior art keywords
sphingosine
modulators
pharmaceuticals
preparing
processes
Prior art date
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English (en)
Inventor
M Heidelbaugh Todd
X Nguyen Phong
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Allergan Inc
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Publication of IN2012DN05171A publication Critical patent/IN2012DN05171A/en

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    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65586—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom
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US20140256945A1 (en) * 2013-03-07 2014-09-11 Allergan, Inc. Phosphonic acid compounds as sphingosine-1-phosphate receptor modulators
US20150045341A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl azetidine derivatives as sphingosine-1 phosphate receptors modulators
US20150045328A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl oxy derivatives as sphingosine-1 phosphate receptors modulators
WO2015073547A1 (en) * 2013-11-13 2015-05-21 Allergan, Inc. Disubstituted phenoxy azetidine derivatives as sphingosine-1-phosphate (s1p) receptor modulators
SG11202006255UA (en) 2018-02-02 2020-07-29 Univ Kyoto Medicine for preventing or treating ophthalmic disease associated with enhanced intraocular neovascularization and/or intraocular vascular permeability
CN117242057A (zh) * 2021-04-14 2023-12-15 株式会社Lg化学 制备用于合成鞘氨醇-1-磷酸酯受体激动剂的中间体的方法
CN117177964A (zh) * 2021-04-14 2023-12-05 株式会社Lg化学 制备鞘氨醇-1-磷酸酯受体激动剂的新方法
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WO2011066179A1 (en) 2011-06-03
MX2012006028A (es) 2012-06-19
AU2010324988A1 (en) 2012-06-07
IL219758A0 (en) 2012-07-31
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EP2504323B1 (en) 2017-03-15
US20110212925A1 (en) 2011-09-01
US20140107075A1 (en) 2014-04-17
RU2012125184A (ru) 2013-12-27
JP2013512244A (ja) 2013-04-11
CL2012001352A1 (es) 2012-08-31
US8653062B2 (en) 2014-02-18
BR112012012259A2 (pt) 2019-09-24
US8440644B2 (en) 2013-05-14
MX2012006022A (es) 2012-08-15
EP2504328A1 (en) 2012-10-03
CA2780908A1 (en) 2011-06-03
RU2012122615A (ru) 2013-12-27
KR20120101686A (ko) 2012-09-14
CA2780987A1 (en) 2011-06-03
IL219759A0 (en) 2012-07-31
WO2011066184A1 (en) 2011-06-03
AU2010324983A1 (en) 2012-06-07
KR20120098796A (ko) 2012-09-05
JP2013512243A (ja) 2013-04-11
AU2010324988B2 (en) 2016-05-26
CN102712618A (zh) 2012-10-03
CN102712607B (zh) 2016-06-22
IN2012DN05125A (es) 2015-10-23
BR112012012261A2 (pt) 2016-04-26
US20110152241A1 (en) 2011-06-23
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