IN2012DN05125A - - Google Patents

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Publication number
IN2012DN05125A
IN2012DN05125A IN5125DEN2012A IN2012DN05125A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A IN 5125DEN2012 A IN5125DEN2012 A IN 5125DEN2012A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A
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India
Prior art keywords
sphingosine
modulators
pharmaceuticals
preparing
processes
Prior art date
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English (en)
Inventor
M Heidelbaugh Todd
X Nguyen Phong
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Allergan Inc
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Publication of IN2012DN05125A publication Critical patent/IN2012DN05125A/en

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    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
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US20140171393A1 (en) * 2012-12-13 2014-06-19 Allergan, Inc. Novel aromatic thio compounds as receptor modulators
PL2958913T3 (pl) * 2013-02-20 2019-03-29 Lg Chem, Ltd. Agoniści receptora sfingozyno-1-fosforanowego, sposoby ich przygotowania i zawierające je jako środek aktywny farmaceutyczne kompozycje
WO2014138075A1 (en) * 2013-03-07 2014-09-12 Allergan, Inc. Phosphonic acid compounds as sphingosine-1-phosphate receptor modulators
US20150045328A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl oxy derivatives as sphingosine-1 phosphate receptors modulators
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WO2015073547A1 (en) * 2013-11-13 2015-05-21 Allergan, Inc. Disubstituted phenoxy azetidine derivatives as sphingosine-1-phosphate (s1p) receptor modulators
SG11202006255UA (en) 2018-02-02 2020-07-29 Univ Kyoto Medicine for preventing or treating ophthalmic disease associated with enhanced intraocular neovascularization and/or intraocular vascular permeability
KR20220142388A (ko) * 2021-04-14 2022-10-21 주식회사 엘지화학 스핑고신-1-인산 수용체 효능제의 신규한 제조방법
CN117242057A (zh) * 2021-04-14 2023-12-15 株式会社Lg化学 制备用于合成鞘氨醇-1-磷酸酯受体激动剂的中间体的方法
TWI823341B (zh) * 2021-04-14 2023-11-21 南韓商Ｌｇ化學股份有限公司 製備鞘胺醇－１－磷酸酯受體促效劑的新穎方法

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US20140107075A1 (en) 2014-04-17
KR20120098796A (ko) 2012-09-05
EP2504323B1 (de) 2017-03-15
AU2010324983A1 (en) 2012-06-07
NZ599966A (en) 2014-09-26
JP2013512243A (ja) 2013-04-11
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CN102712618B (zh) 2014-11-26
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IL219758A0 (en) 2012-07-31
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IL219759A0 (en) 2012-07-31
AU2010324988A1 (en) 2012-06-07
BR112012012259A2 (pt) 2019-09-24
WO2011066179A1 (en) 2011-06-03
US8440644B2 (en) 2013-05-14
EP2504323A1 (de) 2012-10-03
US20110212925A1 (en) 2011-09-01
WO2011066184A1 (en) 2011-06-03
KR20120101686A (ko) 2012-09-14
CL2012001352A1 (es) 2012-08-31
RU2012122615A (ru) 2013-12-27
EP2504328A1 (de) 2012-10-03
ZA201203523B (en) 2013-01-31
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CA2780908A1 (en) 2011-06-03
BR112012012261A2 (pt) 2016-04-26
CA2780987C (en) 2018-03-06
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JP2013512244A (ja) 2013-04-11
JP5939158B2 (ja) 2016-06-22
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US20110152241A1 (en) 2011-06-23
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