IN2012DN03819A - - Google Patents

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Publication number
IN2012DN03819A
IN2012DN03819A IN3819DEN2012A IN2012DN03819A IN 2012DN03819 A IN2012DN03819 A IN 2012DN03819A IN 3819DEN2012 A IN3819DEN2012 A IN 3819DEN2012A IN 2012DN03819 A IN2012DN03819 A IN 2012DN03819A
Authority
IN
India
Prior art keywords
formula
tautomer
stereoisomer
stereoisomers
proportions
Prior art date
Application number
Other languages
English (en)
Inventor
Irene Erdelmeier
Sylvain Daunay
Original Assignee
Tetrahedron
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tetrahedron filed Critical Tetrahedron
Publication of IN2012DN03819A publication Critical patent/IN2012DN03819A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84Sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B55/00Racemisation; Complete or partial inversion
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
IN3819DEN2012 2009-10-06 2010-10-06 IN2012DN03819A (enrdf_load_stackoverflow)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0956968A FR2950890B1 (fr) 2009-10-06 2009-10-06 Procede de synthese de la 2-thiohistidine et analogues
PCT/EP2010/064947 WO2011042478A1 (fr) 2009-10-06 2010-10-06 Procede de synthese de la 2-thiohistidine et analogues

Publications (1)

Publication Number Publication Date
IN2012DN03819A true IN2012DN03819A (enrdf_load_stackoverflow) 2015-08-28

Family

ID=41664356

Family Applications (1)

Application Number Title Priority Date Filing Date
IN3819DEN2012 IN2012DN03819A (enrdf_load_stackoverflow) 2009-10-06 2010-10-06

Country Status (14)

Country Link
US (1) US8835477B2 (enrdf_load_stackoverflow)
EP (1) EP2486019B1 (enrdf_load_stackoverflow)
JP (1) JP5731515B2 (enrdf_load_stackoverflow)
KR (1) KR101773995B1 (enrdf_load_stackoverflow)
CN (1) CN102596915B (enrdf_load_stackoverflow)
AU (1) AU2010305397B2 (enrdf_load_stackoverflow)
BR (1) BR112012007944A2 (enrdf_load_stackoverflow)
CA (1) CA2776833C (enrdf_load_stackoverflow)
ES (1) ES2540279T3 (enrdf_load_stackoverflow)
FR (1) FR2950890B1 (enrdf_load_stackoverflow)
HU (1) HUE025487T2 (enrdf_load_stackoverflow)
IN (1) IN2012DN03819A (enrdf_load_stackoverflow)
RU (1) RU2548153C2 (enrdf_load_stackoverflow)
WO (1) WO2011042478A1 (enrdf_load_stackoverflow)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR3021655B1 (fr) 2014-05-30 2016-07-08 Tetrahedron Nouveaux composes de type 5-acylsulfanyl-histidine en tant que precurseurs des 5-sulfanylhistidines correspondantes et de leurs disulfures
JP6864131B1 (ja) * 2020-03-04 2021-04-28 長瀬産業株式会社 L−エルゴチオネイン含有組成物
US20240199687A1 (en) * 2021-04-22 2024-06-20 University Of Vermont And State Agricultural College Substitution of histidine with 2-thiohistidine in bioactive peptides

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2707087B1 (fr) * 1993-06-28 1995-10-13 Bioxytech Nouveau procédé de préparation de l'ergothionéine.
FR2714380B1 (fr) * 1993-12-24 1996-05-24 Bioxytech Utilisation de dérivés 2-mercapto-imidazole substitués en position 4 (ou 5) comme agents antioxydants, leur procédé de préparation et leurs applications en pharmacie, cosmétique ou alimentaire.
PT939628E (pt) * 1996-07-22 2003-07-31 Monsanto Co Inibidores tiolsulfona de metaloproteases
MXPA03003022A (es) * 2000-10-11 2003-07-14 Esperion Therapeutics Inc Compuestos de sulfuro y disulfuro y composiciones para el control del colesterol y usos relacionados.
US7767826B2 (en) * 2007-10-05 2010-08-03 Pharmatech International, Inc. Process for the synthesis of L-(+)-ergothioneine
FR2950889B1 (fr) 2009-10-06 2011-11-18 Tetrahedron Procede de synthese de l'ergothioneine et analogues

Also Published As

Publication number Publication date
WO2011042478A1 (fr) 2011-04-14
AU2010305397B2 (en) 2014-07-10
JP5731515B2 (ja) 2015-06-10
US8835477B2 (en) 2014-09-16
HUE025487T2 (en) 2016-04-28
EP2486019A1 (fr) 2012-08-15
EP2486019B1 (fr) 2015-03-25
FR2950890B1 (fr) 2011-12-30
CN102596915A (zh) 2012-07-18
AU2010305397A1 (en) 2012-05-24
ES2540279T3 (es) 2015-07-09
CN102596915B (zh) 2016-04-20
RU2548153C2 (ru) 2015-04-20
US20120330029A1 (en) 2012-12-27
FR2950890A1 (fr) 2011-04-08
RU2012117977A (ru) 2013-11-20
KR20120100977A (ko) 2012-09-12
JP2013506705A (ja) 2013-02-28
KR101773995B1 (ko) 2017-09-01
CA2776833C (fr) 2019-03-19
CA2776833A1 (fr) 2011-04-14
BR112012007944A2 (pt) 2015-09-22

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