IN2012DN01661A - - Google Patents

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Publication number
IN2012DN01661A
IN2012DN01661A IN1661DEN2012A IN2012DN01661A IN 2012DN01661 A IN2012DN01661 A IN 2012DN01661A IN 1661DEN2012 A IN1661DEN2012 A IN 1661DEN2012A IN 2012DN01661 A IN2012DN01661 A IN 2012DN01661A
Authority
IN
India
Prior art keywords
disclosed
compounds
intended
kits
abstract
Prior art date
Application number
Other languages
English (en)
Inventor
H Alex Brown
Craig W Lindsley
Alex G Waterson
Sarah A Scott
Original Assignee
Univ Vanderbilt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Vanderbilt filed Critical Univ Vanderbilt
Publication of IN2012DN01661A publication Critical patent/IN2012DN01661A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/438The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
IN1661DEN2012 2009-07-24 2010-07-23 IN2012DN01661A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22849209P 2009-07-24 2009-07-24
PCT/US2010/043045 WO2011011680A1 (fr) 2009-07-24 2010-07-23 Inhibiteurs de phospholipase d sélectifs d'une isoforme

Publications (1)

Publication Number Publication Date
IN2012DN01661A true IN2012DN01661A (fr) 2015-06-05

Family

ID=43499428

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1661DEN2012 IN2012DN01661A (fr) 2009-07-24 2010-07-23

Country Status (14)

Country Link
US (1) US9127005B2 (fr)
EP (1) EP2456307B1 (fr)
JP (1) JP2013500260A (fr)
KR (1) KR20120090034A (fr)
CN (1) CN102573474A (fr)
AU (1) AU2010275526A1 (fr)
BR (1) BR112012001586A2 (fr)
CA (1) CA2768940C (fr)
IL (1) IL217720A0 (fr)
IN (1) IN2012DN01661A (fr)
MX (1) MX2012001064A (fr)
RU (1) RU2012106657A (fr)
SG (1) SG178102A1 (fr)
WO (1) WO2011011680A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9453017B2 (en) 2011-09-30 2016-09-27 Vanderbilt University Antiviral therapies with phospholipase D inhibitors

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG178102A1 (en) 2009-07-24 2012-03-29 Univ Vanderbilt Isoform selective phospholipase d inhibitors
CA2894843A1 (fr) * 2012-12-11 2014-06-19 Vanderbilt University Methodes et compositions pour le traitement d'une infection par le vih
CA2894847A1 (fr) * 2012-12-11 2014-06-19 Vanderbilt University Procedes et compositions comportant des inhibiteurs d'atk et/ou des inhibiteurs de phospholipase d
WO2023243686A1 (fr) * 2022-06-16 2023-12-21 日本たばこ産業株式会社 Composé dihydrooxadiazinone et son utilisation pharmaceutique

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1281502B1 (it) 1995-06-13 1998-02-18 Sardinian Antiviral Research C Impiego di un inibitore non nucleosidico della trascrittasi inversa in associazione con inibitori nucleosidici per il trattamento della
US6187559B1 (en) 1997-08-28 2001-02-13 Novartis Ag Phospholipase D gene
EP1313498A4 (fr) 2000-05-25 2004-04-21 Ben-Tsion Williger Effecteurs de la phospholipase d pour des applications therapeutiques et de dosage
US6482829B2 (en) * 2000-06-08 2002-11-19 Hoffmann-La Roche Inc. Substituted heterocyclic siprodecane compound active as an antagonist of neurokinin 1 receptor
US20060172363A1 (en) 2002-09-18 2006-08-03 Postech Foundation Peptide complexes containing phospholipase d
BRPI0517423A (pt) * 2004-12-27 2008-10-07 Astrazeneca Ab composto, composição farmacêutica, método para o tratamento ou prevenção de distúrbios neurológicos e psiquiátricos associados com disfunção do glutamato em um animal, e, uso em um composto
US20080300298A1 (en) 2005-02-23 2008-12-04 Arbiser Jack L Honokiol Derivates For the Treatment of Proliferative Disorders
CA2651769C (fr) * 2006-05-18 2013-12-17 F. Hoffmann-La Roche Ag Derives de thiazolo-pyramidine /d'uree pyridine comme antagonistes de recepteur d'adenosine a2b.
US20100009970A1 (en) 2008-03-19 2010-01-14 Combinatorx (Singapore) Pte. Ltd. Compositions and methods for treatment of viral diseases
WO2010037081A1 (fr) 2008-09-29 2010-04-01 Palatin Technologies, Inc. Composés de spiropipéridine spécifiques du récepteur de la mélanocortine
EP2413993B1 (fr) 2009-03-31 2020-07-15 Sanofi-Aventis Deutschland GmbH Corps de dispositif d'administration de médicaments
CN102459584A (zh) 2009-05-29 2012-05-16 纽约市哥伦比亚大学理事会 用于治疗神经退行性病症的磷脂酶d的调节
SG178102A1 (en) 2009-07-24 2012-03-29 Univ Vanderbilt Isoform selective phospholipase d inhibitors
US9149445B2 (en) 2009-07-27 2015-10-06 The Trustees Of Princeton University Inhibition of glycerol-3-phosphate acyltransferase (GPAT) and associated enzymes for treatment of viral infections
CA2850597A1 (fr) 2011-09-30 2013-04-04 Vanderbilt University Therapies antivirales avec des inhibiteurs de phospholipase d
CA2894847A1 (fr) 2012-12-11 2014-06-19 Vanderbilt University Procedes et compositions comportant des inhibiteurs d'atk et/ou des inhibiteurs de phospholipase d
CA2894843A1 (fr) 2012-12-11 2014-06-19 Vanderbilt University Methodes et compositions pour le traitement d'une infection par le vih

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9453017B2 (en) 2011-09-30 2016-09-27 Vanderbilt University Antiviral therapies with phospholipase D inhibitors

Also Published As

Publication number Publication date
IL217720A0 (en) 2012-03-29
CA2768940C (fr) 2018-03-13
EP2456307B1 (fr) 2016-11-02
EP2456307A4 (fr) 2013-01-16
MX2012001064A (es) 2012-07-17
SG178102A1 (en) 2012-03-29
RU2012106657A (ru) 2013-08-27
WO2011011680A1 (fr) 2011-01-27
US9127005B2 (en) 2015-09-08
US20120214832A1 (en) 2012-08-23
BR112012001586A2 (pt) 2015-09-01
CN102573474A (zh) 2012-07-11
JP2013500260A (ja) 2013-01-07
CA2768940A1 (fr) 2011-01-27
AU2010275526A1 (en) 2012-03-15
KR20120090034A (ko) 2012-08-16
EP2456307A1 (fr) 2012-05-30

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