IL85641A0 - Tendamistat derivatives - Google Patents
Tendamistat derivativesInfo
- Publication number
- IL85641A0 IL85641A0 IL85641A IL8564188A IL85641A0 IL 85641 A0 IL85641 A0 IL 85641A0 IL 85641 A IL85641 A IL 85641A IL 8564188 A IL8564188 A IL 8564188A IL 85641 A0 IL85641 A0 IL 85641A0
- Authority
- IL
- Israel
- Prior art keywords
- tendamistat
- derivatives
- imidazoles
- hydroxyethyl
- aryl
- Prior art date
Links
- 229950001790 tendamistat Drugs 0.000 title 1
- 108010037401 tendamistate Proteins 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 2
- 230000001430 anti-depressive effect Effects 0.000 abstract 1
- 230000001857 anti-mycotic effect Effects 0.000 abstract 1
- 239000002543 antimycotic Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C07D233/58—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Psychiatry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Paper (AREA)
- Photoreceptors In Electrophotography (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Lubricants (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19873707151 DE3707151A1 (de) | 1987-03-06 | 1987-03-06 | 1-(1-aryl-2-hydroxy-ethyl)-imidazole und deren salze, verfahren zu ihrer herstellung, diese verbindungen enthaltende arzneimittel und ihre verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL85641A0 true IL85641A0 (en) | 1988-08-31 |
Family
ID=6322380
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL85641A IL85641A0 (en) | 1987-03-06 | 1988-03-06 | Tendamistat derivatives |
| IL85640A IL85640A (en) | 1987-03-06 | 1988-03-06 | 1-(1-aryl-2-hydroxyethyl)-imidazoles and salts thereof,processes for the preparation thereof and pharmaceutical compositions containing them |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL85640A IL85640A (en) | 1987-03-06 | 1988-03-06 | 1-(1-aryl-2-hydroxyethyl)-imidazoles and salts thereof,processes for the preparation thereof and pharmaceutical compositions containing them |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4999352A (enExample) |
| EP (1) | EP0281121B1 (enExample) |
| JP (1) | JPS63230673A (enExample) |
| KR (1) | KR880011115A (enExample) |
| AT (1) | ATE75466T1 (enExample) |
| AU (1) | AU621815B2 (enExample) |
| DE (2) | DE3707151A1 (enExample) |
| DK (1) | DK118988A (enExample) |
| FI (1) | FI880987A7 (enExample) |
| GR (1) | GR3005194T3 (enExample) |
| HU (1) | HU201745B (enExample) |
| IL (2) | IL85641A0 (enExample) |
| NO (1) | NO170151C (enExample) |
| NZ (1) | NZ223749A (enExample) |
| PH (3) | PH24990A (enExample) |
| PT (1) | PT86890B (enExample) |
| ZA (1) | ZA881557B (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5229385A (en) * | 1986-01-30 | 1993-07-20 | Takeda Chemical Industries, Ltd. | Quinone derivatives, their production and use |
| DE3931554A1 (de) * | 1989-09-22 | 1991-04-04 | Hoechst Ag | (+)-(2-hydroxy-2-adamantyl)-1-imidazolyl-3- tolyl-methan und dessen salze, verfahren zu dessen herstellung, diese verbindung enthaltende arzneimittel und dessen verwendung |
| AT409084B (de) * | 2000-07-13 | 2002-05-27 | Ledochowski Maximilian Dr | Antimykotisch wirkendes arzneimittel |
| US7678749B2 (en) * | 2007-12-17 | 2010-03-16 | International Flavors & Fragrances Inc. | Organoleptic compounds |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3658813A (en) * | 1970-01-13 | 1972-04-25 | Janssen Pharmaceutica Nv | 1-(beta-aryl-beta-(r-oxy)-ethyl)-imidazoles |
| DE2009020C3 (de) * | 1970-02-26 | 1979-09-13 | Bayer Ag, 5090 Leverkusen | Verfahren zur Herstellung von N-(l,l,l-trisubstituierten)-Methylazolen |
| DE2041771C3 (de) * | 1970-08-22 | 1979-07-26 | Bayer Ag, 5090 Leverkusen | derivate |
| DE2430039C2 (de) * | 1974-06-22 | 1983-11-10 | Bayer Ag, 5090 Leverkusen | Climbazol in kosmetischen Mitteln |
| DE2431407C2 (de) * | 1974-06-29 | 1982-12-02 | Bayer Ag, 5090 Leverkusen | 1,2,4-Triazol-1-yl-alkanone und -alkanole, Verfahren zu ihrer Herstellung sowie ihre Verwendung als Fungizide |
| IE44186B1 (en) * | 1975-12-03 | 1981-09-09 | Ici Ltd | 1,2,4-triazolyl alkanols and their use as pesticides |
| IE45765B1 (en) * | 1976-08-19 | 1982-11-17 | Ici Ltd | Triazoles and imidazoles useful as plant fungicides and growth regulating agents |
| DE2720868A1 (de) * | 1977-05-10 | 1978-11-23 | Bayer Ag | Antimikrobielle mittel |
| DE2758784A1 (de) * | 1977-12-29 | 1979-07-12 | Basf Ag | Triazolyl-glykolaether |
| DE2938575A1 (de) * | 1979-09-24 | 1981-04-23 | Bayer Ag, 5090 Leverkusen | Acylierte imidazolyl-(gamma)-fluorpinakolyl-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide |
| DE2948206A1 (de) * | 1979-11-30 | 1981-06-25 | Basf Ag, 6700 Ludwigshafen | Fungizide (gamma) -azolyl-verbindungen, ihre herstellung und verwendung |
| EP0061835B1 (en) * | 1981-03-18 | 1989-02-01 | Imperial Chemical Industries Plc | Triazole compounds, a process for preparing them, their use as plant fungicides and fungicidal compositions containing them |
| DE3124580A1 (de) * | 1981-06-23 | 1983-01-05 | Bayer Ag, 5090 Leverkusen | Fungizide mittel |
| EP0099165A1 (en) * | 1982-03-23 | 1984-01-25 | Imperial Chemical Industries Plc | Triazole and imidazole compounds, process for their preparation and their use as fungicides and plant growth regulators, and intermediates for their synthesis |
| DE3222191A1 (de) * | 1982-06-12 | 1983-12-15 | Bayer Ag, 5090 Leverkusen | Hydroxyalkinyl-azolyl-derivate, verfahren zu ihrer herstellung sowie ihre verwendung als fungizide |
| EP0097426B1 (en) * | 1982-06-14 | 1988-09-07 | Imperial Chemical Industries Plc | Triazole compounds |
| DE3322526A1 (de) * | 1983-06-23 | 1985-01-10 | Basf Ag, 6700 Ludwigshafen | Fungizide azolverbindungen, ihre herstellung und verwendung |
| DE3345813A1 (de) * | 1983-12-17 | 1985-06-27 | Boehringer Ingelheim KG, 6507 Ingelheim | Neue 2-(1-imidazolyl)-ethanol-derivate |
| EP0149976A3 (de) * | 1983-12-30 | 1986-12-10 | Ciba-Geigy Ag | Substituierte Imidazole |
| DE3628545A1 (de) * | 1985-09-23 | 1987-04-23 | Hoechst Ag | Arylmethylazole und deren salze, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung |
-
1987
- 1987-03-06 DE DE19873707151 patent/DE3707151A1/de not_active Withdrawn
-
1988
- 1988-03-03 EP EP88103225A patent/EP0281121B1/de not_active Expired - Lifetime
- 1988-03-03 AT AT88103225T patent/ATE75466T1/de not_active IP Right Cessation
- 1988-03-03 FI FI880987A patent/FI880987A7/fi not_active Application Discontinuation
- 1988-03-03 PT PT86890A patent/PT86890B/pt not_active IP Right Cessation
- 1988-03-03 DE DE8888103225T patent/DE3870486D1/de not_active Expired - Fee Related
- 1988-03-04 AU AU12641/88A patent/AU621815B2/en not_active Ceased
- 1988-03-04 HU HU881058A patent/HU201745B/hu not_active IP Right Cessation
- 1988-03-04 NZ NZ223749A patent/NZ223749A/en unknown
- 1988-03-04 NO NO880973A patent/NO170151C/no unknown
- 1988-03-04 JP JP63049939A patent/JPS63230673A/ja active Pending
- 1988-03-04 DK DK118988A patent/DK118988A/da not_active Application Discontinuation
- 1988-03-04 ZA ZA881557A patent/ZA881557B/xx unknown
- 1988-03-04 PH PH36596A patent/PH24990A/en unknown
- 1988-03-05 KR KR1019880002282A patent/KR880011115A/ko not_active Withdrawn
- 1988-03-06 IL IL85641A patent/IL85641A0/xx unknown
- 1988-03-06 IL IL85640A patent/IL85640A/xx unknown
- 1988-12-07 PH PH37893A patent/PH25682A/en unknown
- 1988-12-07 PH PH37895A patent/PH25797A/en unknown
-
1989
- 1989-11-28 US US07/441,200 patent/US4999352A/en not_active Expired - Fee Related
-
1992
- 1992-07-16 GR GR920401189T patent/GR3005194T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US4999352A (en) | 1991-03-12 |
| IL85640A (en) | 1992-11-15 |
| JPS63230673A (ja) | 1988-09-27 |
| EP0281121B1 (de) | 1992-04-29 |
| PT86890A (pt) | 1988-04-01 |
| IL85640A0 (en) | 1988-08-31 |
| NO170151B (no) | 1992-06-09 |
| GR3005194T3 (enExample) | 1993-05-24 |
| DK118988D0 (da) | 1988-03-04 |
| AU1264188A (en) | 1988-09-08 |
| FI880987A7 (fi) | 1988-09-07 |
| EP0281121A1 (de) | 1988-09-07 |
| ATE75466T1 (de) | 1992-05-15 |
| AU621815B2 (en) | 1992-03-26 |
| NZ223749A (en) | 1990-11-27 |
| PH24990A (en) | 1990-12-26 |
| ZA881557B (en) | 1988-08-25 |
| PH25682A (en) | 1991-09-04 |
| NO880973L (no) | 1988-09-07 |
| DK118988A (da) | 1988-09-07 |
| NO170151C (no) | 1992-09-16 |
| FI880987A0 (fi) | 1988-03-03 |
| DE3707151A1 (de) | 1988-09-15 |
| HU201745B (en) | 1990-12-28 |
| NO880973D0 (no) | 1988-03-04 |
| PT86890B (pt) | 1992-05-29 |
| KR880011115A (ko) | 1988-10-26 |
| PH25797A (en) | 1991-11-05 |
| DE3870486D1 (de) | 1992-06-04 |
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