IL83304A - Process for the synthesis of penem allyl esters - Google Patents

Process for the synthesis of penem allyl esters

Info

Publication number
IL83304A
IL83304A IL83304A IL8330487A IL83304A IL 83304 A IL83304 A IL 83304A IL 83304 A IL83304 A IL 83304A IL 8330487 A IL8330487 A IL 8330487A IL 83304 A IL83304 A IL 83304A
Authority
IL
Israel
Prior art keywords
synthesis
penem
allyl esters
esters
allyl
Prior art date
Application number
IL83304A
Other languages
English (en)
Other versions
IL83304A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL83304A0 publication Critical patent/IL83304A0/xx
Publication of IL83304A publication Critical patent/IL83304A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Electric Double-Layer Capacitors Or The Like (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Paints Or Removers (AREA)
  • Control Of El Displays (AREA)
  • Pens And Brushes (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Steroid Compounds (AREA)
  • Mechanical Pencils And Projecting And Retracting Systems Therefor, And Multi-System Writing Instruments (AREA)
IL83304A 1986-07-29 1987-07-23 Process for the synthesis of penem allyl esters IL83304A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/891,493 US4695626A (en) 1986-07-29 1986-07-29 1-aza-4,5-dithiabicyclo [4.2.0] oct-2-en-8-one-2 carboxylate esters

Publications (2)

Publication Number Publication Date
IL83304A0 IL83304A0 (en) 1987-12-31
IL83304A true IL83304A (en) 1992-06-21

Family

ID=25398284

Family Applications (1)

Application Number Title Priority Date Filing Date
IL83304A IL83304A (en) 1986-07-29 1987-07-23 Process for the synthesis of penem allyl esters

Country Status (18)

Country Link
US (2) US4695626A (fr)
EP (1) EP0255307B1 (fr)
JP (1) JPH0737462B2 (fr)
KR (1) KR890004581B1 (fr)
AT (1) ATE70064T1 (fr)
AU (1) AU583465B2 (fr)
CA (1) CA1285275C (fr)
DE (1) DE3774954D1 (fr)
DK (1) DK170169B1 (fr)
ES (1) ES2038665T3 (fr)
FI (1) FI87651C (fr)
GR (1) GR3003660T3 (fr)
HU (1) HU198068B (fr)
IE (1) IE60029B1 (fr)
IL (1) IL83304A (fr)
NZ (1) NZ221201A (fr)
PT (1) PT85407B (fr)
ZA (1) ZA875541B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU563157B2 (en) * 1982-12-08 1987-07-02 Farmitalia Carlo Erba S.P.A. 2-thiacephems and (5r) penems derivatives
US4782145A (en) * 1986-06-02 1988-11-01 Pfizer Inc. Process for penem derivatives
US4751297A (en) * 1987-03-20 1988-06-14 Pfizer Inc. Method for preparation of azetidinone-1-oxoacetate by oxidation of the corresponding 2-hydroxyacetate
US5191077A (en) * 1987-05-11 1993-03-02 Pfizer Inc. Diastereomeric 5R,6S-6-(1R-hydroxyethyl)-2-(cis-1-oxo-3-thiolanylthio)-2-penem-3-carboxylic acids
WO1988008845A1 (fr) * 1987-05-11 1988-11-17 Pfizer Inc. Acides diastereomeres 5r,6s-6-(1r-hydroxyethyle)-2-(cis-1-oxo-3-thiolanylthio)-2-penem-3-carboxyliques
DE19512050A1 (de) * 1995-03-31 1996-10-02 Gimmy Lindomare Dr Vorrichtung zum Sichern von Schrauben vor unbefugtem Zugriff
MXPA06013412A (es) * 2004-05-19 2007-01-23 Maxygen Inc Polipeptidos de interferon-alfa y conjugados.
WO2009029554A2 (fr) * 2007-08-24 2009-03-05 Codexis, Inc. Polypeptides cétoréductases ayant des propriétés améliorées pour la production stéréosélective de (r)-3-hydroxythiolane
EP3523309B1 (fr) * 2016-10-10 2024-04-17 The Johns Hopkins University Agents antibactériens contre d, d- et l, d-transpeptidases

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH541577A (de) * 1970-11-03 1973-09-15 Ciba Geigy Ag Verfahren zur Herstellung thiaheterocyclischer Verbindungen
EP0051813B1 (fr) * 1980-11-06 1986-07-30 Hoechst Uk Limited Dérivés de 7-oxo-4-thia-1-aza(3.2.0)heptane et de 7-oxo-4-thia-1-aza(3.2.0)hept-2-ène
JPS57176988A (en) * 1981-04-09 1982-10-30 Sankyo Co Ltd Penam-3-carboxylic acid derivative and its preparation
AU563157B2 (en) * 1982-12-08 1987-07-02 Farmitalia Carlo Erba S.P.A. 2-thiacephems and (5r) penems derivatives
GB2131432B (en) * 1982-12-08 1986-10-15 Erba Farmitalia Preparation of (5r)-penem derivatives
EP0115308A3 (fr) * 1983-01-25 1984-10-10 Merck & Co. Inc. Acides pen-2-em-3-carboxyliques 2-alkylthio non-substitués et procédé pour préparer des 2-thioxopénames substitués et des thiopénèmes 2-substitués
EP0130025B1 (fr) * 1983-06-21 1987-07-08 Pfizer Inc. Dérivés de 2-alkylthiopénème
EP0132101A1 (fr) * 1983-07-14 1985-01-23 Pfizer Inc. Dérivés de 2-hétérocycloalkylthiopénème

Also Published As

Publication number Publication date
GR3003660T3 (fr) 1993-03-16
CA1285275C (fr) 1991-06-25
FI87651C (fi) 1993-02-10
PT85407A (en) 1987-08-01
NZ221201A (en) 1990-06-26
EP0255307B1 (fr) 1991-12-04
FI873290A0 (fi) 1987-07-28
IE60029B1 (en) 1994-05-18
AU7618787A (en) 1988-02-04
PT85407B (pt) 1990-04-30
EP0255307A1 (fr) 1988-02-03
KR890004581B1 (ko) 1989-11-16
KR880001668A (ko) 1988-04-26
HUT45067A (en) 1988-05-30
ES2038665T3 (es) 1993-08-01
FI87651B (fi) 1992-10-30
AU583465B2 (en) 1989-04-27
FI873290A (fi) 1988-01-30
ZA875541B (en) 1989-03-29
IE872046L (en) 1988-01-29
DE3774954D1 (de) 1992-01-16
DK392287A (da) 1988-01-30
US4695626A (en) 1987-09-22
HU198068B (en) 1989-07-28
DK392287D0 (da) 1987-07-28
IL83304A0 (en) 1987-12-31
DK170169B1 (da) 1995-06-06
JPS6341481A (ja) 1988-02-22
JPH0737462B2 (ja) 1995-04-26
ATE70064T1 (de) 1991-12-15
US4782146A (en) 1988-11-01

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Legal Events

Date Code Title Description
RH Patent void