IL67381A - N-substituted-4-aminomethyl-imidazole derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

N-substituted-4-aminomethyl-imidazole derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL67381A
IL67381A IL67381A IL6738182A IL67381A IL 67381 A IL67381 A IL 67381A IL 67381 A IL67381 A IL 67381A IL 6738182 A IL6738182 A IL 6738182A IL 67381 A IL67381 A IL 67381A
Authority
IL
Israel
Prior art keywords
sub
hydrogen
compounds
carbon atoms
substituted
Prior art date
Application number
IL67381A
Other languages
English (en)
Other versions
IL67381A0 (en
Original Assignee
Farmos Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmos Group Ltd filed Critical Farmos Group Ltd
Publication of IL67381A0 publication Critical patent/IL67381A0/xx
Publication of IL67381A publication Critical patent/IL67381A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Catalysts (AREA)
IL67381A 1981-12-04 1982-12-01 N-substituted-4-aminomethyl-imidazole derivatives,their preparation and pharmaceutical compositions containing them IL67381A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB08136646A GB2110663B (en) 1981-12-04 1981-12-04 Imidazole derivatives

Publications (2)

Publication Number Publication Date
IL67381A0 IL67381A0 (en) 1983-05-15
IL67381A true IL67381A (en) 1986-08-31

Family

ID=10526383

Family Applications (1)

Application Number Title Priority Date Filing Date
IL67381A IL67381A (en) 1981-12-04 1982-12-01 N-substituted-4-aminomethyl-imidazole derivatives,their preparation and pharmaceutical compositions containing them

Country Status (15)

Country Link
US (1) US4517198A (fr)
EP (1) EP0081324B1 (fr)
JP (1) JPS58105970A (fr)
AT (1) ATE21246T1 (fr)
AU (1) AU552908B2 (fr)
CA (1) CA1184183A (fr)
DE (1) DE3272478D1 (fr)
DK (1) DK157926C (fr)
FI (1) FI76569C (fr)
GB (1) GB2110663B (fr)
IE (1) IE54243B1 (fr)
IL (1) IL67381A (fr)
NO (1) NO158017C (fr)
NZ (1) NZ202649A (fr)
ZA (1) ZA828803B (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2548183B1 (fr) * 1983-07-01 1985-10-31 Synthelabo Diphenylazomethines portant un radical imidazolyle, leur preparation et leur application en therapeutique
FR2575470B1 (fr) * 1984-12-27 1987-02-13 Synthelabo Derives amines de n-imidazolylmethyl-diphenylazomethines, leur preparation et leur application en therapeutique
FR2575469B1 (fr) * 1984-12-27 1987-01-23 Synthelabo N-imidazolylmethyl-diphenylazomethines, leur preparation et leur application en therapeutique
US4996221A (en) * 1987-01-13 1991-02-26 The Board Of Trustees Of The Leland Stanford Junior University Histamine derivatives as immune modulators
JPH032168A (ja) * 1989-03-30 1991-01-08 Farmos Yhtymae Oy アロマターゼ阻害活性を有する新規な4(5)―イミダゾール
NZ238688A (en) * 1990-06-28 1992-05-26 Smithkline Beecham Corp Substituted histidines: pharmaceutical compositions, preparation and uses thereof
US5159083A (en) * 1990-12-28 1992-10-27 Neurogen Corporation Certain aminomethyl phenylimidazole derivatives; a class of dopamine receptor subtype specific ligands
GB9127304D0 (en) * 1991-12-23 1992-02-19 Boots Co Plc Therapeutic agents
USRE37303E1 (en) * 1992-01-10 2001-07-31 Institut National Del La Sante Et De La Recherche Medicale Imidazole compounds and their therapeutic applications
FR2686084B1 (fr) * 1992-01-10 1995-12-22 Bioprojet Soc Civ Nouveaux derives de l'imidazole, leur preparation et leurs applications therapeutiques.
FR2689508B1 (fr) * 1992-04-01 1994-06-17 Fournier Ind & Sante Derives de l'imidazole, leur procede de preparation et leur application en therapeutique.
GB9312893D0 (en) * 1993-06-22 1993-08-04 Boots Co Plc Therapeutic agents
AU7275894A (en) * 1993-08-04 1995-02-28 Yamanouchi Pharmaceutical Co., Ltd. Imidazolylalkylamine derivative and pharmaceutical composition thereof
CA2222099A1 (fr) * 1995-05-30 1996-12-05 Gliatech, Inc. Derives imidazole 1h-4(5)-substitues
US6448282B1 (en) 1995-05-30 2002-09-10 Gliatech, Inc. 1H-4(5)-substituted imidazole derivatives
US20060167269A1 (en) * 2001-07-11 2006-07-27 Hamilton Andrew D Compounds and methods for the inhibition of compounds cruzi
US20030152747A1 (en) * 2002-01-11 2003-08-14 The Garland Company, Inc., An Ohio Corporation Roofing materials
EP2076497B1 (fr) 2006-10-19 2012-02-22 F. Hoffmann-La Roche AG Aminométhyl-4-imidazoles

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE276541C (fr) *
GB1341375A (en) * 1969-11-19 1973-12-19 Smith Kline French Lab Aminoalkylimidazoles and process for their production
DE2842280A1 (de) * 1978-09-28 1980-04-10 Bayer Ag N-(1,3-azolyl)-alkyl-halogenacetanilide, verfahren zu ihrer herstellung sowie ihre verwendung als herbizide
AU518569B2 (en) * 1979-08-07 1981-10-08 Farmos-Yhtyma Oy 4-benzyl- and 4-benzoyl imidazole derivatives

Also Published As

Publication number Publication date
IE54243B1 (en) 1989-08-02
FI823871L (fi) 1983-06-05
NZ202649A (en) 1985-04-30
AU9095782A (en) 1983-06-09
DK157926C (da) 1990-08-06
ATE21246T1 (de) 1986-08-15
DK531282A (da) 1983-06-05
CA1184183A (fr) 1985-03-19
IE822877L (en) 1983-06-04
FI76569B (fi) 1988-07-29
JPS58105970A (ja) 1983-06-24
DK157926B (da) 1990-03-05
NO824062L (no) 1983-06-06
EP0081324A2 (fr) 1983-06-15
EP0081324A3 (en) 1983-12-07
AU552908B2 (en) 1986-06-26
ZA828803B (en) 1983-09-28
IL67381A0 (en) 1983-05-15
FI823871A0 (fi) 1982-11-11
EP0081324B1 (fr) 1986-08-06
US4517198A (en) 1985-05-14
NO158017C (no) 1988-06-29
NO158017B (no) 1988-03-21
FI76569C (fi) 1988-11-10
DE3272478D1 (en) 1986-09-11
GB2110663A (en) 1983-06-22
JPH0344072B2 (fr) 1991-07-04
GB2110663B (en) 1985-08-07

Similar Documents

Publication Publication Date Title
AU528275B2 (en) Imidazole derivatives
IL67381A (en) N-substituted-4-aminomethyl-imidazole derivatives,their preparation and pharmaceutical compositions containing them
DE3261153D1 (en) Substituted imidazole derivatives and their preparation and use

Legal Events

Date Code Title Description
RH Patent void