IL65378A - Process for preparing 3-(4-aminoethoxybenzoyl)benzo-(b)thiophenes - Google Patents

Process for preparing 3-(4-aminoethoxybenzoyl)benzo-(b)thiophenes

Info

Publication number
IL65378A
IL65378A IL65378A IL6537882A IL65378A IL 65378 A IL65378 A IL 65378A IL 65378 A IL65378 A IL 65378A IL 6537882 A IL6537882 A IL 6537882A IL 65378 A IL65378 A IL 65378A
Authority
IL
Israel
Prior art keywords
aminoethoxybenzoyl
thiophenes
benzo
preparing
Prior art date
Application number
IL65378A
Other languages
English (en)
Other versions
IL65378A0 (en
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/246,334 external-priority patent/US4358593A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of IL65378A0 publication Critical patent/IL65378A0/xx
Publication of IL65378A publication Critical patent/IL65378A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Extrusion Moulding Of Plastics Or The Like (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
IL65378A 1981-04-03 1982-03-30 Process for preparing 3-(4-aminoethoxybenzoyl)benzo-(b)thiophenes IL65378A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24633581A 1981-04-03 1981-04-03
US06/246,334 US4358593A (en) 1981-04-03 1981-04-03 Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes
US33104581A 1981-12-16 1981-12-16

Publications (2)

Publication Number Publication Date
IL65378A0 IL65378A0 (en) 1982-05-31
IL65378A true IL65378A (en) 1986-02-28

Family

ID=27399920

Family Applications (1)

Application Number Title Priority Date Filing Date
IL65378A IL65378A (en) 1981-04-03 1982-03-30 Process for preparing 3-(4-aminoethoxybenzoyl)benzo-(b)thiophenes

Country Status (17)

Country Link
EP (1) EP0062504B1 (cs)
KR (1) KR850001882B1 (cs)
CS (1) CS227348B2 (cs)
DD (1) DD201793A5 (cs)
DE (1) DE3268227D1 (cs)
DK (1) DK151282A (cs)
EG (1) EG15610A (cs)
ES (1) ES8307240A1 (cs)
FI (1) FI821160L (cs)
GB (1) GB2097392B (cs)
GR (1) GR76468B (cs)
HU (1) HU191353B (cs)
IE (1) IE53187B1 (cs)
IL (1) IL65378A (cs)
PL (1) PL130867B1 (cs)
PT (1) PT74692B (cs)
SU (1) SU1155157A3 (cs)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4117512A1 (de) * 1991-05-25 1992-11-26 Schering Ag 2-phenylbenzo(b)furane und -thiophene, verfahren zu deren herstellung und diese enthaltende pharmazeutische praeparate
CA2145614A1 (en) * 1994-03-31 1995-10-01 Jeffrey A. Dodge Intermediates and processes for preparing benzothiophene compounds
US5523416A (en) * 1994-07-22 1996-06-04 Eli Lilly And Company Process for preparing 3-(4-aminoethoxy-benzoyl) benzo (B)-thiophenes
US5629425A (en) * 1994-09-19 1997-05-13 Eli Lilly And Company Haloalkyl hemisolvates of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-piperidinoethoxy)-benzoyl]benzo[b]thiophene
CO4410190A1 (es) * 1994-09-19 1997-01-09 Lilly Co Eli 3-[4-(2-AMINOETOXI)-BENZOIL]-2-ARIL-6-HIDROXIBENZO [b] TIOFENO CRISTALINO
US5589482A (en) * 1994-12-14 1996-12-31 Pfizer Inc. Benzo-thiophene estrogen agonists to treat prostatic hyperplasia
US6391892B1 (en) * 1995-03-10 2002-05-21 Eli Lilly And Company Naphthyl pharmaceutical compounds
US5728724A (en) * 1995-08-17 1998-03-17 Eli Lilly And Company Benzothiophene compounds
AU5258696A (en) * 1996-03-19 1997-10-10 Eli Lilly And Company Synthesis of 3-{4-(2-aminoethoxy)-benzoyl}-2-aryl-6-hydroxy-benzo{b}thiop henes
AR013321A1 (es) * 1996-09-25 2000-12-27 Lilly Co Eli Procedimiento para preparar 2-(4-alcoxifenil)-6-alcoxi-benzo[b]tiofenos.
US5916916A (en) * 1996-10-10 1999-06-29 Eli Lilly And Company 1-aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods
ZA9710262B (en) * 1996-11-19 1999-05-13 Lilly Co Eli Process for the synthesis of benzothiophenes
CN1254280A (zh) * 1997-04-30 2000-05-24 伊莱利利公司 用于制备取代的苯并[b]噻吩的区域选择性烷基化方法
CN1252717A (zh) * 1997-04-30 2000-05-10 伊莱利利公司 制备苯并[b]噻吩的中间体和方法
JP2001522372A (ja) * 1997-04-30 2001-11-13 イーライ・リリー・アンド・カンパニー ベンゾチオフェンの製造方法
AU7261498A (en) * 1997-04-30 1998-11-24 Eli Lilly And Company Intermediates and processes for preparing benzo{b}thiophenes
CA2236254A1 (en) * 1997-04-30 1998-10-30 David Warren Hoard Process for preparing benzo¬b|thiophenes
CA2231013A1 (en) * 1997-04-30 1998-10-30 Eli Lilly And Company Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
EP1832582A1 (en) 2002-09-30 2007-09-12 A/S GEA Farmaceutisk Fabrik Novel raloxifene malonic acid addition salts and/or solvates thereof, and pharmaceutical compositions comprising these
EP2322519A1 (en) * 2009-10-23 2011-05-18 Hexal AG A process for preparing benzo[b]thiophene derivatives
WO2011099942A1 (en) 2010-02-09 2011-08-18 Silverstone Pharma New addition salts of raloxifene, process for the preparation thereof and use thereof in therapy

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3947470A (en) * 1974-06-20 1976-03-30 Smithkline Corporation Substituted benzofurans and benzothiophenes
US4001426A (en) * 1974-10-17 1977-01-04 Smithkline Corporation Substituted benzofurans and benzothiophenes
FR2279395A1 (fr) * 1975-06-02 1976-02-20 Labaz Nouveaux derives de benzthiophene, leurs precedes de preparation ainsi que les compositions pharmaceutiques les contenant
US4133814A (en) 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents

Also Published As

Publication number Publication date
IE820786L (en) 1982-10-03
PL235752A1 (cs) 1982-11-22
KR850001882B1 (ko) 1985-12-28
IL65378A0 (en) 1982-05-31
PT74692A (en) 1982-05-01
ES511124A0 (es) 1983-06-16
CS227348B2 (en) 1984-04-16
GB2097392B (en) 1985-04-24
PT74692B (en) 1985-01-08
FI821160A0 (fi) 1982-04-02
EG15610A (en) 1986-06-30
HU191353B (en) 1987-02-27
IE53187B1 (en) 1988-08-17
FI821160A7 (fi) 1982-10-04
FI821160L (fi) 1982-10-04
EP0062504A1 (en) 1982-10-13
SU1155157A3 (ru) 1985-05-07
ES8307240A1 (es) 1983-06-16
GR76468B (cs) 1984-08-10
DE3268227D1 (en) 1986-02-13
GB2097392A (en) 1982-11-03
KR830010100A (ko) 1983-12-26
EP0062504B1 (en) 1986-01-02
DK151282A (da) 1982-10-04
DD201793A5 (de) 1983-08-10
PL130867B1 (en) 1984-09-29

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