IL235133A - History 5 - [[4 - [[morpholine-2-yl] methyl amino] -5- (trifluoromethyl) -2-pyridyl] amino] pyrazine-2-carbonitrile and therapeutic uses thereof - Google Patents
History 5 - [[4 - [[morpholine-2-yl] methyl amino] -5- (trifluoromethyl) -2-pyridyl] amino] pyrazine-2-carbonitrile and therapeutic uses thereofInfo
- Publication number
- IL235133A IL235133A IL235133A IL23513314A IL235133A IL 235133 A IL235133 A IL 235133A IL 235133 A IL235133 A IL 235133A IL 23513314 A IL23513314 A IL 23513314A IL 235133 A IL235133 A IL 235133A
- Authority
- IL
- Israel
- Prior art keywords
- cancer
- treatment
- compound according
- inhibitor
- compound
- Prior art date
Links
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261647200P | 2012-05-15 | 2012-05-15 | |
| PCT/GB2013/051233 WO2013171470A1 (en) | 2012-05-15 | 2013-05-14 | 5-[[4-[[morpholin-2-yl]methylamino]-5-(trifluoromethyl)-2-pyridyl]amino]pyrazine-2-carbonitrile and therapeutic uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL235133A true IL235133A (en) | 2017-03-30 |
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| HUE046727T2 (hu) | 2013-12-06 | 2020-03-30 | Vertex Pharma | Az ATR-kináz inhibitoraként használható vegyület, 2-amino-6-fluoro-N-[5-fluoro-piridin-3-IL]-pirazolo-[1,5-A]-pirimidin-3-karboxamid, ennek elõállítása, különbözõ szilárd formái és ezek radioaktív nyomjelzett származékai |
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