IL188898A0 - Processes for preparing pyrazol-o-glycoside derivatives and novel intermediates of said processes - Google Patents

Processes for preparing pyrazol-o-glycoside derivatives and novel intermediates of said processes

Info

Publication number
IL188898A0
IL188898A0 IL188898A IL18889808A IL188898A0 IL 188898 A0 IL188898 A0 IL 188898A0 IL 188898 A IL188898 A IL 188898A IL 18889808 A IL18889808 A IL 18889808A IL 188898 A0 IL188898 A0 IL 188898A0
Authority
IL
Israel
Prior art keywords
processes
novel intermediates
glycoside derivatives
pyrazol
preparing
Prior art date
Application number
IL188898A
Other languages
English (en)
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of IL188898A0 publication Critical patent/IL188898A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
IL188898A 2005-07-22 2008-01-21 Processes for preparing pyrazol-o-glycoside derivatives and novel intermediates of said processes IL188898A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05015935 2005-07-22
PCT/EP2006/064435 WO2007010015A1 (en) 2005-07-22 2006-07-20 Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes

Publications (1)

Publication Number Publication Date
IL188898A0 true IL188898A0 (en) 2008-04-13

Family

ID=37102155

Family Applications (1)

Application Number Title Priority Date Filing Date
IL188898A IL188898A0 (en) 2005-07-22 2008-01-21 Processes for preparing pyrazol-o-glycoside derivatives and novel intermediates of said processes

Country Status (14)

Country Link
EP (1) EP1910391A1 (ja)
JP (2) JP4888840B2 (ja)
KR (1) KR20080036112A (ja)
CN (1) CN101218244A (ja)
AR (1) AR054852A1 (ja)
AU (1) AU2006271653A1 (ja)
BR (1) BRPI0613690A2 (ja)
CA (1) CA2621269A1 (ja)
IL (1) IL188898A0 (ja)
MX (1) MX2008000011A (ja)
RU (1) RU2008106461A (ja)
TW (1) TW200728286A (ja)
WO (1) WO2007010015A1 (ja)
ZA (1) ZA200709951B (ja)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1550668A4 (en) * 2002-10-04 2008-10-01 Kissei Pharmaceutical PYRAZOLE DERIVATIVE, MEDICINAL COMPOSITION COMPRISING THE DERIVATIVE, MEDICINAL USE THEREOF, AND INTERMEDIATE ENTERING THE PRODUCTION THEREOF
US7375090B2 (en) 2003-08-26 2008-05-20 Boehringer Ingelheim International Gmbh Glucopyranosyloxy-pyrazoles, pharmaceutical compositions containing these compounds, the use thereof and processed for the preparation thereof
UY29694A1 (es) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int Metodos para prevenir y tratar trastornos metabolicos y nuevos derivados de pirazol-o-glucosido
UY30082A1 (es) 2006-01-11 2007-08-31 Boehringer Ingelheim Int Forma cristalina de 1-(1-metiletil)-4`-((2-fluoro-4-metoxifenil)metil)-5`- metil-1h-pirazol-3`-o-b-d-glucopiranosido, un metodo para su preparacion y el uso de la misma para preparar medicamentos
JP5902671B2 (ja) * 2011-03-31 2016-04-13 キッセイ薬品工業株式会社 ベンジルピラゾール誘導体の製造方法およびその製造中間体

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55157504A (en) * 1979-05-24 1980-12-08 Sankyo Co Ltd Herbicide
ATE455785T1 (de) * 2000-11-02 2010-02-15 Ajinomoto Kk Neue pyrazolderivate und diese enthaltende mittel gegen diabetes
PT1354888E (pt) * 2000-12-28 2009-07-27 Kissei Pharmaceutical Derivados de glucopiranosiloxipirazole e sua utilização em medicamentos
EP1364957B1 (en) * 2001-02-26 2008-12-31 Kissei Pharmaceutical Co., Ltd. Glycopyranosyloxypyrazole derivatives and medicinal use thereof
JP4147111B2 (ja) * 2001-02-27 2008-09-10 キッセイ薬品工業株式会社 グルコピラノシルオキシピラゾール誘導体およびその医薬用途
WO2002088157A1 (fr) * 2001-04-27 2002-11-07 Ajinomoto Co., Inc. Derives pyrazolyl-o-glycoside n-substitues et medicament contre le diabete en contenant
JP4399251B2 (ja) * 2001-05-30 2010-01-13 キッセイ薬品工業株式会社 グルコピラノシルオキシピラゾール誘導体、それを含有する医薬組成物、その医薬用途およびその製造中間体
EP1432720A1 (en) * 2001-09-05 2004-06-30 Bristol-Myers Squibb Company O-pyrazole glucoside sglt2 inhibitors and method of use
JP4424203B2 (ja) * 2002-04-26 2010-03-03 味の素株式会社 糖尿病予防・治療剤
ES2345250T3 (es) * 2002-08-08 2010-09-20 Kissei Pharmaceutical Co., Ltd. Derivado de pirazol en la composicion medicinal que contiene el mismo, el uso medicinal del mismo, y un intermedio para la produccion del mismo.
JP2004137245A (ja) * 2002-08-23 2004-05-13 Kissei Pharmaceut Co Ltd ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体
WO2004019958A1 (ja) * 2002-08-27 2004-03-11 Kissei Pharmaceutical Co., Ltd. ピラゾール誘導体、それを含有する医薬組成物及びその医薬用途
EP1550668A4 (en) * 2002-10-04 2008-10-01 Kissei Pharmaceutical PYRAZOLE DERIVATIVE, MEDICINAL COMPOSITION COMPRISING THE DERIVATIVE, MEDICINAL USE THEREOF, AND INTERMEDIATE ENTERING THE PRODUCTION THEREOF
WO2004089967A1 (ja) * 2003-04-01 2004-10-21 Taisho Pharmaceutical Co., Ltd. ヘテロアリール ５－チオ－β－Ｄ－グルコピラノシド誘導体及びそれを含有する糖尿病治療薬
WO2004113359A1 (ja) * 2003-06-20 2004-12-29 Kissei Pharmaceutical Co., Ltd. ピラゾール誘導体、それを含有する医薬組成物及びその製造中間体
UY29694A1 (es) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int Metodos para prevenir y tratar trastornos metabolicos y nuevos derivados de pirazol-o-glucosido

Also Published As

Publication number Publication date
BRPI0613690A2 (pt) 2011-01-25
AR054852A1 (es) 2007-07-18
TW200728286A (en) 2007-08-01
JP4888840B2 (ja) 2012-02-29
KR20080036112A (ko) 2008-04-24
ZA200709951B (en) 2008-11-26
WO2007010015A1 (en) 2007-01-25
AU2006271653A1 (en) 2007-01-25
MX2008000011A (es) 2008-03-26
EP1910391A1 (en) 2008-04-16
RU2008106461A (ru) 2009-08-27
JP2009502763A (ja) 2009-01-29
JP2012006956A (ja) 2012-01-12
CN101218244A (zh) 2008-07-09
CA2621269A1 (en) 2007-01-25

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