TW200728286A - Processes for preparing pyrazole-O-glycoside derivatives and novel intermediates of said processes - Google Patents

Processes for preparing pyrazole-O-glycoside derivatives and novel intermediates of said processes

Info

Publication number
TW200728286A
TW200728286A TW095126625A TW95126625A TW200728286A TW 200728286 A TW200728286 A TW 200728286A TW 095126625 A TW095126625 A TW 095126625A TW 95126625 A TW95126625 A TW 95126625A TW 200728286 A TW200728286 A TW 200728286A
Authority
TW
Taiwan
Prior art keywords
processes
novel intermediates
glycoside derivatives
preparing
preparing pyrazole
Prior art date
Application number
TW095126625A
Other languages
Chinese (zh)
Inventor
Waldemar Pfrengle
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of TW200728286A publication Critical patent/TW200728286A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5

Abstract

The present invention relates to processes for preparing the compounds of general formula I, wherein the groups R1 to R6 and R7a, R7b, R7c are defined according to claim 1. Furthermore the present invention relates to processes for preparing educts and intermediates in the above processes and to intermediates as such.
TW095126625A 2005-07-22 2006-07-21 Processes for preparing pyrazole-O-glycoside derivatives and novel intermediates of said processes TW200728286A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05015935 2005-07-22

Publications (1)

Publication Number Publication Date
TW200728286A true TW200728286A (en) 2007-08-01

Family

ID=37102155

Family Applications (1)

Application Number Title Priority Date Filing Date
TW095126625A TW200728286A (en) 2005-07-22 2006-07-21 Processes for preparing pyrazole-O-glycoside derivatives and novel intermediates of said processes

Country Status (14)

Country Link
EP (1) EP1910391A1 (en)
JP (2) JP4888840B2 (en)
KR (1) KR20080036112A (en)
CN (1) CN101218244A (en)
AR (1) AR054852A1 (en)
AU (1) AU2006271653A1 (en)
BR (1) BRPI0613690A2 (en)
CA (1) CA2621269A1 (en)
IL (1) IL188898A0 (en)
MX (1) MX2008000011A (en)
RU (1) RU2008106461A (en)
TW (1) TW200728286A (en)
WO (1) WO2007010015A1 (en)
ZA (1) ZA200709951B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4530855B2 (en) * 2002-10-04 2010-08-25 キッセイ薬品工業株式会社 Pyrazole derivative, pharmaceutical composition containing the same, pharmaceutical use thereof and production intermediate thereof
US7375090B2 (en) 2003-08-26 2008-05-20 Boehringer Ingelheim International Gmbh Glucopyranosyloxy-pyrazoles, pharmaceutical compositions containing these compounds, the use thereof and processed for the preparation thereof
UY29694A1 (en) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int METHODS TO PREVENT AND TREAT METABOLIC AND NEW DISORDERS DERIVED FROM PIRAZOL-O-GLUCOSIDO
UY30082A1 (en) 2006-01-11 2007-08-31 Boehringer Ingelheim Int CRYSTAL FORM OF 1- (1-METHYLETHYL) -4` - ((2-FLUORO-4-METOXIFENIL) METHYL) -5`- METHYL-1H-PIRAZOL-3`-OBD-GLUCOPYRANOSIDE, A METHOD FOR PREPARATION AND USE OF THE SAME TO PREPARE MEDICATIONS
WO2012133783A1 (en) * 2011-03-31 2012-10-04 キッセイ薬品工業株式会社 Method for producing benzylpyrazole derivative and production intermediate thereof

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55157504A (en) * 1979-05-24 1980-12-08 Sankyo Co Ltd Herbicide
EP1338603B1 (en) * 2000-11-02 2010-01-20 Ajinomoto Co., Inc. Novel pyrazole derivatives and diabetes remedies containing the same
CZ305971B6 (en) * 2000-12-28 2016-06-01 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivatives and use thereof in medicaments
US7087579B2 (en) * 2001-02-26 2006-08-08 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivatives and medicinal use thereof
JP4147111B2 (en) * 2001-02-27 2008-09-10 キッセイ薬品工業株式会社 Glucopyranosyloxypyrazole derivative and its pharmaceutical use
CA2445346C (en) * 2001-04-27 2010-04-06 Ajinomoto Co., Inc. N-substituted pyrazole-o-glycoside derivatives and therapeutic agent for diabetes containing the same
CA2448741C (en) * 2001-05-30 2010-06-22 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate therefor
WO2003020737A1 (en) * 2001-09-05 2003-03-13 Bristol-Myers Squibb Company O-pyrazole glucoside sglt2 inhibitors and method of use
AU2003231517A1 (en) * 2002-04-26 2003-11-10 Ajinomoto Co., Inc. Preventive/remedy for diabetes
RU2356906C2 (en) * 2002-08-08 2009-05-27 Киссеи Фармасьютикал Ко., Лтд. Pyrazole derivatieves, medical compositions, containing said derivatives, their application in medicine and intermediate compounds for their obtaining
JP2004137245A (en) * 2002-08-23 2004-05-13 Kissei Pharmaceut Co Ltd Pyrazole derivative, pharmaceutical composition containing the same, its pharmaceutical use and production intermediate
JP4606876B2 (en) * 2002-08-27 2011-01-05 キッセイ薬品工業株式会社 Pyrazole derivative, pharmaceutical composition containing the same, and pharmaceutical use thereof
JP4530855B2 (en) * 2002-10-04 2010-08-25 キッセイ薬品工業株式会社 Pyrazole derivative, pharmaceutical composition containing the same, pharmaceutical use thereof and production intermediate thereof
JPWO2004089966A1 (en) * 2003-04-01 2006-07-06 大正製薬株式会社 Process for selective production of heteroaryl 5-thio-β-D-aldohexopyranoside
EP1637539B1 (en) * 2003-06-20 2012-01-18 Kissei Pharmaceutical Co., Ltd. Pyrazole derivative, drug composition containing the same and production intermediate therefor
UY29694A1 (en) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int METHODS TO PREVENT AND TREAT METABOLIC AND NEW DISORDERS DERIVED FROM PIRAZOL-O-GLUCOSIDO

Also Published As

Publication number Publication date
IL188898A0 (en) 2008-04-13
WO2007010015A1 (en) 2007-01-25
MX2008000011A (en) 2008-03-26
BRPI0613690A2 (en) 2011-01-25
RU2008106461A (en) 2009-08-27
CA2621269A1 (en) 2007-01-25
JP4888840B2 (en) 2012-02-29
CN101218244A (en) 2008-07-09
AR054852A1 (en) 2007-07-18
EP1910391A1 (en) 2008-04-16
JP2009502763A (en) 2009-01-29
JP2012006956A (en) 2012-01-12
KR20080036112A (en) 2008-04-24
ZA200709951B (en) 2008-11-26
AU2006271653A1 (en) 2007-01-25

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