ZA200709951B - Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes - Google Patents
Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processesInfo
- Publication number
- ZA200709951B ZA200709951B ZA200709951A ZA200709951A ZA200709951B ZA 200709951 B ZA200709951 B ZA 200709951B ZA 200709951 A ZA200709951 A ZA 200709951A ZA 200709951 A ZA200709951 A ZA 200709951A ZA 200709951 B ZA200709951 B ZA 200709951B
- Authority
- ZA
- South Africa
- Prior art keywords
- processes
- novel intermediates
- glycoside derivatives
- preparing pyrazole
- pyrazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05015935 | 2005-07-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200709951B true ZA200709951B (en) | 2008-11-26 |
Family
ID=37102155
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200709951A ZA200709951B (en) | 2005-07-22 | 2007-11-19 | Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP1910391A1 (ja) |
| JP (2) | JP4888840B2 (ja) |
| KR (1) | KR20080036112A (ja) |
| CN (1) | CN101218244A (ja) |
| AR (1) | AR054852A1 (ja) |
| AU (1) | AU2006271653A1 (ja) |
| BR (1) | BRPI0613690A2 (ja) |
| CA (1) | CA2621269A1 (ja) |
| IL (1) | IL188898A0 (ja) |
| MX (1) | MX2008000011A (ja) |
| RU (1) | RU2008106461A (ja) |
| TW (1) | TW200728286A (ja) |
| WO (1) | WO2007010015A1 (ja) |
| ZA (1) | ZA200709951B (ja) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4530855B2 (ja) * | 2002-10-04 | 2010-08-25 | キッセイ薬品工業株式会社 | ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体 |
| US7375090B2 (en) | 2003-08-26 | 2008-05-20 | Boehringer Ingelheim International Gmbh | Glucopyranosyloxy-pyrazoles, pharmaceutical compositions containing these compounds, the use thereof and processed for the preparation thereof |
| UY29694A1 (es) * | 2005-07-28 | 2007-02-28 | Boehringer Ingelheim Int | Metodos para prevenir y tratar trastornos metabolicos y nuevos derivados de pirazol-o-glucosido |
| UY30082A1 (es) | 2006-01-11 | 2007-08-31 | Boehringer Ingelheim Int | Forma cristalina de 1-(1-metiletil)-4`-((2-fluoro-4-metoxifenil)metil)-5`- metil-1h-pirazol-3`-o-b-d-glucopiranosido, un metodo para su preparacion y el uso de la misma para preparar medicamentos |
| JP5902671B2 (ja) * | 2011-03-31 | 2016-04-13 | キッセイ薬品工業株式会社 | ベンジルピラゾール誘導体の製造方法およびその製造中間体 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS55157504A (en) * | 1979-05-24 | 1980-12-08 | Sankyo Co Ltd | Herbicide |
| ATE455785T1 (de) * | 2000-11-02 | 2010-02-15 | Ajinomoto Kk | Neue pyrazolderivate und diese enthaltende mittel gegen diabetes |
| SK287786B6 (sk) * | 2000-12-28 | 2011-09-05 | Kissei Pharmaceutical Co., Ltd. | Glukopyranosyloxypyrazolový derivát, farmaceutická kompozícia alebo kombinácia s jeho obsahom a ich použitie |
| CA2438593C (en) * | 2001-02-26 | 2010-09-21 | Kissei Pharmaceutical Co., Ltd. | Glucopyranosyloxypyrazole derivatives and medicinal use thereof |
| WO2002068440A1 (fr) * | 2001-02-27 | 2002-09-06 | Kissei Pharmaceutical Co., Ltd. | Derives de glycopyranosyloxypyrazole et utilisation medicinale de ceux-ci |
| EP1389621A4 (en) * | 2001-04-27 | 2005-05-11 | Ajinomoto Kk | N-SUBSTITUTED PYRAZOLYL-O-GLYCOSIDE DERIVATIVES AND DIABETES CONTAINING THEREOF |
| EP1400529A4 (en) * | 2001-05-30 | 2007-12-19 | Kissei Pharmaceutical | GLUCOPYRANOSYLOXYPYRAZOLE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL AND INTERMEDIARY USE THEREOF |
| EP1432720A1 (en) * | 2001-09-05 | 2004-06-30 | Bristol-Myers Squibb Company | O-pyrazole glucoside sglt2 inhibitors and method of use |
| AU2003231517A1 (en) * | 2002-04-26 | 2003-11-10 | Ajinomoto Co., Inc. | Preventive/remedy for diabetes |
| ATE469161T1 (de) * | 2002-08-08 | 2010-06-15 | Kissei Pharmaceutical | Pyrazolderivat, dieses enthaltende medizinische zusammensetzung, medizinische verwendung davon, und zwischenprodukt für dessen herstellung |
| JP2004137245A (ja) * | 2002-08-23 | 2004-05-13 | Kissei Pharmaceut Co Ltd | ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体 |
| AU2003262262A1 (en) * | 2002-08-27 | 2004-03-19 | Kissei Pharmaceutical Co., Ltd. | Pyrazole derivatives, medicinal composition containing the same, and medicinal use thereof |
| JP4530855B2 (ja) * | 2002-10-04 | 2010-08-25 | キッセイ薬品工業株式会社 | ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体 |
| JPWO2004089966A1 (ja) * | 2003-04-01 | 2006-07-06 | 大正製薬株式会社 | 選択的なヘテロアリール５−チオ−β−Ｄ−アルドヘキソピラノシドの製造法 |
| CA2529878C (en) * | 2003-06-20 | 2012-11-20 | Kissei Pharmaceutical Co., Ltd. | Pyrazole derivative, drug composition containing the same and production intermediate therefor |
| UY29694A1 (es) * | 2005-07-28 | 2007-02-28 | Boehringer Ingelheim Int | Metodos para prevenir y tratar trastornos metabolicos y nuevos derivados de pirazol-o-glucosido |
-
2006
- 2006-07-20 AU AU2006271653A patent/AU2006271653A1/en not_active Abandoned
- 2006-07-20 JP JP2008521974A patent/JP4888840B2/ja not_active Expired - Fee Related
- 2006-07-20 WO PCT/EP2006/064435 patent/WO2007010015A1/en active Application Filing
- 2006-07-20 MX MX2008000011A patent/MX2008000011A/es not_active Application Discontinuation
- 2006-07-20 AR ARP060103114A patent/AR054852A1/es unknown
- 2006-07-20 CA CA002621269A patent/CA2621269A1/en not_active Abandoned
- 2006-07-20 EP EP06777849A patent/EP1910391A1/en not_active Withdrawn
- 2006-07-20 CN CNA2006800246999A patent/CN101218244A/zh active Pending
- 2006-07-20 KR KR1020087004344A patent/KR20080036112A/ko not_active Application Discontinuation
- 2006-07-20 RU RU2008106461/04A patent/RU2008106461A/ru not_active Application Discontinuation
- 2006-07-20 BR BRPI0613690-7A patent/BRPI0613690A2/pt not_active IP Right Cessation
- 2006-07-21 TW TW095126625A patent/TW200728286A/zh unknown
-
2007
- 2007-11-19 ZA ZA200709951A patent/ZA200709951B/xx unknown
-
2008
- 2008-01-21 IL IL188898A patent/IL188898A0/en unknown
-
2011
- 2011-08-11 JP JP2011176119A patent/JP2012006956A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| IL188898A0 (en) | 2008-04-13 |
| CN101218244A (zh) | 2008-07-09 |
| EP1910391A1 (en) | 2008-04-16 |
| CA2621269A1 (en) | 2007-01-25 |
| RU2008106461A (ru) | 2009-08-27 |
| KR20080036112A (ko) | 2008-04-24 |
| AU2006271653A1 (en) | 2007-01-25 |
| JP2009502763A (ja) | 2009-01-29 |
| AR054852A1 (es) | 2007-07-18 |
| BRPI0613690A2 (pt) | 2011-01-25 |
| WO2007010015A1 (en) | 2007-01-25 |
| JP4888840B2 (ja) | 2012-02-29 |
| MX2008000011A (es) | 2008-03-26 |
| TW200728286A (en) | 2007-08-01 |
| JP2012006956A (ja) | 2012-01-12 |
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