IL165826A0 - Substituted aryl boronic acids their preparation and their precursors - Google Patents
Substituted aryl boronic acids their preparation and their precursorsInfo
- Publication number
- IL165826A0 IL165826A0 IL16582603A IL16582603A IL165826A0 IL 165826 A0 IL165826 A0 IL 165826A0 IL 16582603 A IL16582603 A IL 16582603A IL 16582603 A IL16582603 A IL 16582603A IL 165826 A0 IL165826 A0 IL 165826A0
- Authority
- IL
- Israel
- Prior art keywords
- precursors
- preparation
- substituted aryl
- boronic acids
- aryl boronic
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 239000002243 precursor Substances 0.000 title 1
- 125000003107 substituted aryl group Chemical group 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C217/06—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
- C07C217/14—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring
- C07C217/18—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted
- C07C217/20—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted by halogen atoms, by trihalomethyl, nitro or nitroso groups, or by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39350102P | 2002-07-03 | 2002-07-03 | |
| PCT/IB2003/002947 WO2004005301A1 (en) | 2002-07-03 | 2003-06-23 | Substituted aryl boronic acids, their preparation and their precursors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL165826A0 true IL165826A0 (en) | 2006-01-15 |
Family
ID=30115592
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL16582603A IL165826A0 (en) | 2002-07-03 | 2003-06-23 | Substituted aryl boronic acids their preparation and their precursors |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US7045652B2 (zh) |
| EP (1) | EP1519940A1 (zh) |
| JP (1) | JP2005531642A (zh) |
| CN (1) | CN1665824A (zh) |
| AU (1) | AU2003244968A1 (zh) |
| BR (1) | BR0312335A (zh) |
| CA (1) | CA2491029A1 (zh) |
| IL (1) | IL165826A0 (zh) |
| MX (1) | MXPA05000258A (zh) |
| RU (1) | RU2004139087A (zh) |
| WO (1) | WO2004005301A1 (zh) |
| ZA (1) | ZA200410195B (zh) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7041280B2 (en) * | 2001-06-29 | 2006-05-09 | Genzyme Corporation | Aryl boronate functionalized polymers for treating obesity |
| US6858592B2 (en) * | 2001-06-29 | 2005-02-22 | Genzyme Corporation | Aryl boronic acids for treating obesity |
| US7145040B2 (en) * | 2004-07-02 | 2006-12-05 | Bristol-Myers Squibb Co. | Process for the preparation of amino acids useful in the preparation of peptide receptor modulators |
| JO3598B1 (ar) * | 2006-10-10 | 2020-07-05 | Infinity Discovery Inc | الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني |
| JP2013518886A (ja) * | 2010-02-03 | 2013-05-23 | インフイニトイ プハルマセウトイカルス インコーポレイテッド | 脂肪酸アミドヒドロラーゼ阻害剤 |
| ITMI20121390A1 (it) * | 2012-08-06 | 2014-02-07 | F I S Fabbrica Italiana Sint P A | Procedimento per la preparazione di acido 2-cianofenilboronico e suoi esteri, intermedi del perampanel o di e2040 |
| CN108409767B (zh) * | 2018-04-13 | 2020-07-10 | 上海泰坦科技股份有限公司 | 一种杂环联苯硼酸的制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1064252A (en) | 1963-09-19 | 1967-04-05 | Ici Ltd | Amides and pharmaceutical compositions containing them |
| GB1177548A (en) | 1967-11-28 | 1970-01-14 | Ici Ltd | Phenoxy-and Anilino-Alkanoic Acid Amides |
| CA2091864C (en) * | 1992-03-26 | 1999-09-07 | Tomokazu Hino | Process for producing halogenophenoxyfatty acid derivatives by selective halogenation and halogenophenoxyfatty acid derivatives |
| US5550134A (en) | 1995-05-10 | 1996-08-27 | Eli Lilly And Company | Methods for inhibiting bone loss |
| UA64740C2 (uk) | 1997-02-10 | 2004-03-15 | Пфайзер Продактс Інк. | Похідні 2-амінопіридинів, фармацевтична композиція на їх основі (варіанти), спосіб лікування (варіанти), спосіб інгібування nos у ссавця та проміжні сполуки (варіанти) |
| US6235771B1 (en) | 1998-12-21 | 2001-05-22 | Takeda Chemical Industries, Ltd. | Anilide derivative, production and use thereof |
| UA72611C2 (uk) * | 2000-05-17 | 2005-03-15 | Орто-Макнейл Фармацевтикал, Інк. | Похідні заміщеного піролопіридинону, корисні як інгібітори фосфодіестерази |
-
2003
- 2003-06-03 US US10/453,433 patent/US7045652B2/en not_active Expired - Fee Related
- 2003-06-23 CN CN038156237A patent/CN1665824A/zh active Pending
- 2003-06-23 MX MXPA05000258A patent/MXPA05000258A/es unknown
- 2003-06-23 IL IL16582603A patent/IL165826A0/xx unknown
- 2003-06-23 JP JP2004519102A patent/JP2005531642A/ja not_active Withdrawn
- 2003-06-23 BR BR0312335-9A patent/BR0312335A/pt not_active IP Right Cessation
- 2003-06-23 RU RU2004139087/04A patent/RU2004139087A/ru not_active Application Discontinuation
- 2003-06-23 EP EP03738442A patent/EP1519940A1/en not_active Withdrawn
- 2003-06-23 CA CA002491029A patent/CA2491029A1/en not_active Abandoned
- 2003-06-23 AU AU2003244968A patent/AU2003244968A1/en not_active Abandoned
- 2003-06-23 WO PCT/IB2003/002947 patent/WO2004005301A1/en not_active Application Discontinuation
-
2004
- 2004-12-17 ZA ZA200410195A patent/ZA200410195B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1665824A (zh) | 2005-09-07 |
| US7045652B2 (en) | 2006-05-16 |
| US20040038940A1 (en) | 2004-02-26 |
| JP2005531642A (ja) | 2005-10-20 |
| CA2491029A1 (en) | 2004-01-15 |
| EP1519940A1 (en) | 2005-04-06 |
| WO2004005301A1 (en) | 2004-01-15 |
| AU2003244968A1 (en) | 2004-01-23 |
| BR0312335A (pt) | 2005-04-12 |
| ZA200410195B (en) | 2006-07-26 |
| RU2004139087A (ru) | 2005-07-10 |
| MXPA05000258A (es) | 2005-04-11 |
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