IL154222A0 - Imidazolyl derivatives - Google Patents

Imidazolyl derivatives

Info

Publication number
IL154222A0
IL154222A0 IL15422201A IL15422201A IL154222A0 IL 154222 A0 IL154222 A0 IL 154222A0 IL 15422201 A IL15422201 A IL 15422201A IL 15422201 A IL15422201 A IL 15422201A IL 154222 A0 IL154222 A0 IL 154222A0
Authority
IL
Israel
Prior art keywords
imidazolyl derivatives
imidazolyl
derivatives
Prior art date
Application number
IL15422201A
Other languages
English (en)
Original Assignee
Sod Conseils Rech Applic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Publication of IL154222A0 publication Critical patent/IL154222A0/xx

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    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
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    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Hematology (AREA)
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IL15422201A 2000-08-01 2001-07-31 Imidazolyl derivatives IL154222A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22258400P 2000-08-01 2000-08-01
PCT/US2001/023959 WO2002010140A2 (en) 2000-08-01 2001-07-31 Imidazolyl derivatives

Publications (1)

Publication Number Publication Date
IL154222A0 true IL154222A0 (en) 2003-07-31

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Application Number Title Priority Date Filing Date
IL15422201A IL154222A0 (en) 2000-08-01 2001-07-31 Imidazolyl derivatives

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US (2) US7566734B2 (es)
EP (1) EP1305294B1 (es)
JP (1) JP2004518613A (es)
KR (1) KR20030020960A (es)
CN (1) CN1444566A (es)
AR (1) AR035040A1 (es)
AT (1) ATE360620T1 (es)
AU (2) AU2001279098B2 (es)
CA (1) CA2417204A1 (es)
DE (1) DE60128102T2 (es)
ES (1) ES2282275T3 (es)
IL (1) IL154222A0 (es)
NO (1) NO20030473L (es)
NZ (1) NZ523774A (es)
WO (1) WO2002010140A2 (es)

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CA2499586A1 (en) * 2002-10-07 2004-04-22 Merck & Co., Inc. Antidiabetic beta-amino heterocyclic dipeptidyl peptidase inhibitors
US20060052382A1 (en) * 2002-12-20 2006-03-09 Duffy Joseph L 3-Amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
US20040186151A1 (en) * 2003-02-12 2004-09-23 Mjalli Adnan M.M. Substituted azole derivatives as therapeutic agents
US7569578B2 (en) 2003-12-05 2009-08-04 Bristol-Meyers Squibb Company Heterocyclic anti-migraine agents
WO2005077373A2 (en) * 2004-02-03 2005-08-25 Astrazeneca Ab Treatment of gastro-esophageal reflux disease (gerd)
TW200533398A (en) 2004-03-29 2005-10-16 Bristol Myers Squibb Co Novel therapeutic agents for the treatment of migraine
US7453002B2 (en) 2004-06-15 2008-11-18 Bristol-Myers Squibb Company Five-membered heterocycles useful as serine protease inhibitors
JP4836280B2 (ja) 2004-06-18 2011-12-14 ノバルティス バクシンズ アンド ダイアグノスティックス,インコーポレーテッド 癌を治療するためのキネシンスピンドルタンパク質(ksp)阻害剤としてのn−(1−(1−ベンジル−4−フェニル−1h−イミダゾール−2−イル)−2,2−ジメチルプロピル)ベンズアミド誘導体および関連化合物
US7608723B2 (en) 2004-10-19 2009-10-27 Novartis Vaccines And Diagnostics, Inc. Indole and benzimidazole derivatives
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