IL142502A0 - Intermediates for the preparation of biologically active benzothiazolone ethanamines - Google Patents
Intermediates for the preparation of biologically active benzothiazolone ethanaminesInfo
- Publication number
- IL142502A0 IL142502A0 IL14250296A IL14250296A IL142502A0 IL 142502 A0 IL142502 A0 IL 142502A0 IL 14250296 A IL14250296 A IL 14250296A IL 14250296 A IL14250296 A IL 14250296A IL 142502 A0 IL142502 A0 IL 142502A0
- Authority
- IL
- Israel
- Prior art keywords
- ethanamines
- intermediates
- preparation
- biologically active
- benzothiazolone
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pulmonology (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9526511.2A GB9526511D0 (en) | 1995-12-23 | 1995-12-23 | Pharmaceutically active compounds |
| PCT/SE1996/001650 WO1997023470A1 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
| IL12499896A IL124998A0 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL142502A0 true IL142502A0 (en) | 2002-03-10 |
Family
ID=10786064
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL12499896A IL124998A0 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
| IL14250296A IL142502A0 (en) | 1995-12-23 | 1996-12-13 | Intermediates for the preparation of biologically active benzothiazolone ethanamines |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL12499896A IL124998A0 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US5929100A (ru) |
| EP (1) | EP0918760B1 (ru) |
| JP (1) | JP2000502681A (ru) |
| KR (1) | KR19990076688A (ru) |
| CN (1) | CN1072214C (ru) |
| AR (1) | AR005008A1 (ru) |
| AT (1) | ATE209638T1 (ru) |
| AU (1) | AU704506B2 (ru) |
| BR (1) | BR9612234A (ru) |
| CA (1) | CA2238877A1 (ru) |
| CZ (1) | CZ288704B6 (ru) |
| DE (1) | DE69617472D1 (ru) |
| EE (1) | EE03440B1 (ru) |
| GB (1) | GB9526511D0 (ru) |
| HU (1) | HUP9900100A3 (ru) |
| IL (2) | IL124998A0 (ru) |
| IS (1) | IS4759A (ru) |
| MX (1) | MX9804828A (ru) |
| NO (1) | NO982927D0 (ru) |
| NZ (1) | NZ325500A (ru) |
| PL (1) | PL327475A1 (ru) |
| RU (1) | RU2177476C2 (ru) |
| SK (1) | SK82098A3 (ru) |
| TR (1) | TR199801196T2 (ru) |
| TW (1) | TW401411B (ru) |
| WO (1) | WO1997023470A1 (ru) |
| ZA (1) | ZA9610354B (ru) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999009018A1 (fr) * | 1997-08-14 | 1999-02-25 | Kirin Beer Kabushiki Kaisha | DERIVES DE BENZOTHIAZOLONE PRESENTANT UNE ACTIVITE SELECTIVE D'AGONISTE DU RECEPTEUR β2 |
| GB0218629D0 (en) * | 2002-08-09 | 2002-09-18 | Novartis Ag | Organic compounds |
| AR040962A1 (es) * | 2002-08-09 | 2005-04-27 | Novartis Ag | Compuestos derivados de tiazol 1,3-2-ona, composicion farmaceutica y proceso de preparacion del compuesto |
| ES2329586T3 (es) | 2003-11-21 | 2009-11-27 | Theravance, Inc. | Compuestos que tienen actividad agonista del receptor beta2 adrenergico y antagonista del receptor muscarino. |
| TW200738658A (en) | 2005-08-09 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
| TW200738659A (en) * | 2005-08-29 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
| TW200745067A (en) | 2006-03-14 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
| TW200833670A (en) | 2006-12-20 | 2008-08-16 | Astrazeneca Ab | Novel compounds 569 |
| GB0702458D0 (en) | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | Salts 668 |
| CN102124003A (zh) | 2008-06-18 | 2011-07-13 | 阿斯利康(瑞典)有限公司 | 作为治疗呼吸系统疾病的β2肾上腺素受体拮抗剂的苯并噁嗪酮衍生物 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4314944A (en) * | 1980-08-22 | 1982-02-09 | Smithkline Corporation | 4-Aminoalkyl-7-hydroxy-2(3H)-indolones |
| US4452808A (en) * | 1982-12-07 | 1984-06-05 | Smithkline Beckman Corporation | 4-Aminoalkyl-2(3H)-indolones |
| GB8426200D0 (en) * | 1984-10-17 | 1984-11-21 | Glaxo Holdings Ltd | Chemical compounds |
| US4554284A (en) * | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones |
| US4554287A (en) * | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | Antihypertensive 7-[2-(dialkylamino)ethyl]-4-hydroxy-1,3-benzimidazol-2-ones |
| DK514585A (da) * | 1984-11-08 | 1986-05-09 | Syntex Inc | Aminoethylanilinderivater |
| DE3728695A1 (de) * | 1987-08-25 | 1989-03-09 | Schering Ag | Neue benzimidazol-derivate |
| US5648370A (en) * | 1990-11-20 | 1997-07-15 | Astra Pharmaceuticals Limited | 7-(2-aminoethyl) benzothiazolones |
| GB9211172D0 (en) * | 1992-05-27 | 1992-07-08 | Fisons Plc | Compounds |
| GB9210632D0 (en) * | 1992-05-19 | 1992-07-01 | Fisons Plc | Compounds |
| IE914003A1 (en) * | 1990-11-20 | 1992-05-20 | Astra Pharma Prod | Biologically Active Amines |
-
1995
- 1995-12-23 GB GBGB9526511.2A patent/GB9526511D0/en active Pending
-
1996
- 1996-12-09 ZA ZA9610354A patent/ZA9610354B/xx unknown
- 1996-12-09 AR ARP960105568A patent/AR005008A1/es unknown
- 1996-12-11 TW TW085115316A patent/TW401411B/zh not_active IP Right Cessation
- 1996-12-13 TR TR1998/01196T patent/TR199801196T2/xx unknown
- 1996-12-13 IL IL12499896A patent/IL124998A0/xx unknown
- 1996-12-13 EE EE9800193A patent/EE03440B1/xx not_active IP Right Cessation
- 1996-12-13 EP EP96944153A patent/EP0918760B1/en not_active Expired - Lifetime
- 1996-12-13 PL PL96327475A patent/PL327475A1/xx unknown
- 1996-12-13 SK SK820-98A patent/SK82098A3/sk unknown
- 1996-12-13 HU HU9900100A patent/HUP9900100A3/hu unknown
- 1996-12-13 US US08/793,706 patent/US5929100A/en not_active Expired - Fee Related
- 1996-12-13 WO PCT/SE1996/001650 patent/WO1997023470A1/en not_active Application Discontinuation
- 1996-12-13 CA CA002238877A patent/CA2238877A1/en not_active Abandoned
- 1996-12-13 DE DE69617472T patent/DE69617472D1/de not_active Expired - Lifetime
- 1996-12-13 KR KR1019980704800A patent/KR19990076688A/ko not_active Application Discontinuation
- 1996-12-13 NZ NZ325500A patent/NZ325500A/xx unknown
- 1996-12-13 CN CN96199237A patent/CN1072214C/zh not_active Expired - Fee Related
- 1996-12-13 AU AU14025/97A patent/AU704506B2/en not_active Ceased
- 1996-12-13 JP JP09523560A patent/JP2000502681A/ja active Pending
- 1996-12-13 BR BR9612234A patent/BR9612234A/pt not_active Application Discontinuation
- 1996-12-13 CZ CZ19981684A patent/CZ288704B6/cs not_active IP Right Cessation
- 1996-12-13 RU RU98114080/04A patent/RU2177476C2/ru active
- 1996-12-13 IL IL14250296A patent/IL142502A0/xx unknown
- 1996-12-13 AT AT96944153T patent/ATE209638T1/de not_active IP Right Cessation
-
1998
- 1998-05-27 IS IS4759A patent/IS4759A/is unknown
- 1998-06-16 MX MX9804828A patent/MX9804828A/es unknown
- 1998-06-23 NO NO982927A patent/NO982927D0/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AU704506B2 (en) | 1999-04-22 |
| CN1211242A (zh) | 1999-03-17 |
| TW401411B (en) | 2000-08-11 |
| HUP9900100A3 (en) | 2001-10-29 |
| IS4759A (is) | 1998-05-27 |
| NO982927L (no) | 1998-06-23 |
| MX9804828A (es) | 1998-09-30 |
| ATE209638T1 (de) | 2001-12-15 |
| HUP9900100A2 (hu) | 1999-05-28 |
| CZ168498A3 (cs) | 1998-09-16 |
| ZA9610354B (en) | 1997-06-23 |
| JP2000502681A (ja) | 2000-03-07 |
| NZ325500A (en) | 1999-01-28 |
| AR005008A1 (es) | 1999-04-07 |
| EP0918760B1 (en) | 2001-11-28 |
| NO982927D0 (no) | 1998-06-23 |
| CN1072214C (zh) | 2001-10-03 |
| EP0918760A1 (en) | 1999-06-02 |
| GB9526511D0 (en) | 1996-02-28 |
| PL327475A1 (en) | 1998-12-07 |
| BR9612234A (pt) | 1999-07-13 |
| EE03440B1 (et) | 2001-06-15 |
| CA2238877A1 (en) | 1997-07-03 |
| CZ288704B6 (cs) | 2001-08-15 |
| US5929100A (en) | 1999-07-27 |
| KR19990076688A (ko) | 1999-10-15 |
| AU1402597A (en) | 1997-07-17 |
| DE69617472D1 (de) | 2002-01-10 |
| TR199801196T2 (xx) | 1998-10-21 |
| RU2177476C2 (ru) | 2001-12-27 |
| SK82098A3 (en) | 1998-11-04 |
| EE9800193A (et) | 1998-12-15 |
| WO1997023470A1 (en) | 1997-07-03 |
| IL124998A0 (en) | 1999-01-26 |
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