EE03440B1 - Bioloogilise toimega bensotiasolooni etaanamiinid ja nende valmistamise protsess - Google Patents

Bioloogilise toimega bensotiasolooni etaanamiinid ja nende valmistamise protsess

Info

Publication number
EE03440B1
EE03440B1 EE9800193A EE9800193A EE03440B1 EE 03440 B1 EE03440 B1 EE 03440B1 EE 9800193 A EE9800193 A EE 9800193A EE 9800193 A EE9800193 A EE 9800193A EE 03440 B1 EE03440 B1 EE 03440B1
Authority
EE
Estonia
Prior art keywords
ethanamines
preparation
biologically active
benzothiazolone
active benzothiazolone
Prior art date
Application number
EE9800193A
Other languages
English (en)
Other versions
EE9800193A (et
Inventor
Victor Bonnert Roger
Charles Brown Roger
Alan Cage Peter
Cheshire David
Ince Francis
Original Assignee
Astra Pharmaceuticals Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Pharmaceuticals Limited filed Critical Astra Pharmaceuticals Limited
Publication of EE9800193A publication Critical patent/EE9800193A/et
Publication of EE03440B1 publication Critical patent/EE03440B1/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
EE9800193A 1995-12-23 1996-12-13 Bioloogilise toimega bensotiasolooni etaanamiinid ja nende valmistamise protsess EE03440B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9526511.2A GB9526511D0 (en) 1995-12-23 1995-12-23 Pharmaceutically active compounds
PCT/SE1996/001650 WO1997023470A1 (en) 1995-12-23 1996-12-13 Biologically active benzothiazolone ethanamines

Publications (2)

Publication Number Publication Date
EE9800193A EE9800193A (et) 1998-12-15
EE03440B1 true EE03440B1 (et) 2001-06-15

Family

ID=10786064

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9800193A EE03440B1 (et) 1995-12-23 1996-12-13 Bioloogilise toimega bensotiasolooni etaanamiinid ja nende valmistamise protsess

Country Status (27)

Country Link
US (1) US5929100A (et)
EP (1) EP0918760B1 (et)
JP (1) JP2000502681A (et)
KR (1) KR19990076688A (et)
CN (1) CN1072214C (et)
AR (1) AR005008A1 (et)
AT (1) ATE209638T1 (et)
AU (1) AU704506B2 (et)
BR (1) BR9612234A (et)
CA (1) CA2238877A1 (et)
CZ (1) CZ288704B6 (et)
DE (1) DE69617472D1 (et)
EE (1) EE03440B1 (et)
GB (1) GB9526511D0 (et)
HU (1) HUP9900100A3 (et)
IL (2) IL124998A0 (et)
IS (1) IS4759A (et)
MX (1) MX9804828A (et)
NO (1) NO982927D0 (et)
NZ (1) NZ325500A (et)
PL (1) PL327475A1 (et)
RU (1) RU2177476C2 (et)
SK (1) SK82098A3 (et)
TR (1) TR199801196T2 (et)
TW (1) TW401411B (et)
WO (1) WO1997023470A1 (et)
ZA (1) ZA9610354B (et)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999009018A1 (fr) * 1997-08-14 1999-02-25 Kirin Beer Kabushiki Kaisha DERIVES DE BENZOTHIAZOLONE PRESENTANT UNE ACTIVITE SELECTIVE D'AGONISTE DU RECEPTEUR β2
GB0218629D0 (en) * 2002-08-09 2002-09-18 Novartis Ag Organic compounds
PE20050130A1 (es) * 2002-08-09 2005-03-29 Novartis Ag Compuestos organicos
JP4851937B2 (ja) 2003-11-21 2012-01-11 セラヴァンス， インコーポレーテッド β２アドレナリン作動性受容体作動薬活性およびムスカリン受容体拮抗薬活性を有する化合物
TW200738658A (en) 2005-08-09 2007-10-16 Astrazeneca Ab Novel compounds
TW200738659A (en) * 2005-08-29 2007-10-16 Astrazeneca Ab Novel compounds
TW200745067A (en) 2006-03-14 2007-12-16 Astrazeneca Ab Novel compounds
TW200833670A (en) 2006-12-20 2008-08-16 Astrazeneca Ab Novel compounds 569
GB0702458D0 (en) 2007-02-08 2007-03-21 Astrazeneca Ab Salts 668
CN102124003A (zh) 2008-06-18 2011-07-13 阿斯利康(瑞典)有限公司 作为治疗呼吸系统疾病的β2肾上腺素受体拮抗剂的苯并噁嗪酮衍生物

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4314944A (en) * 1980-08-22 1982-02-09 Smithkline Corporation 4-Aminoalkyl-7-hydroxy-2(3H)-indolones
US4452808A (en) * 1982-12-07 1984-06-05 Smithkline Beckman Corporation 4-Aminoalkyl-2(3H)-indolones
GB8426200D0 (en) * 1984-10-17 1984-11-21 Glaxo Holdings Ltd Chemical compounds
US4554287A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation Antihypertensive 7-[2-(dialkylamino)ethyl]-4-hydroxy-1,3-benzimidazol-2-ones
US4554284A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
EP0180994A3 (en) * 1984-11-08 1987-09-23 Syntex (U.S.A.) Inc. Antihypertensive dialkyl aminoethylaniline derivatives
DE3728695A1 (de) * 1987-08-25 1989-03-09 Schering Ag Neue benzimidazol-derivate
GB9210632D0 (en) * 1992-05-19 1992-07-01 Fisons Plc Compounds
US5648370A (en) * 1990-11-20 1997-07-15 Astra Pharmaceuticals Limited 7-(2-aminoethyl) benzothiazolones
IE914003A1 (en) * 1990-11-20 1992-05-20 Astra Pharma Prod Biologically Active Amines
GB9211172D0 (en) * 1992-05-27 1992-07-08 Fisons Plc Compounds

Also Published As

Publication number Publication date
HUP9900100A3 (en) 2001-10-29
AU1402597A (en) 1997-07-17
CA2238877A1 (en) 1997-07-03
IS4759A (is) 1998-05-27
CN1211242A (zh) 1999-03-17
BR9612234A (pt) 1999-07-13
CN1072214C (zh) 2001-10-03
ZA9610354B (en) 1997-06-23
NO982927L (no) 1998-06-23
PL327475A1 (en) 1998-12-07
TR199801196T2 (xx) 1998-10-21
IL124998A0 (en) 1999-01-26
TW401411B (en) 2000-08-11
WO1997023470A1 (en) 1997-07-03
SK82098A3 (en) 1998-11-04
RU2177476C2 (ru) 2001-12-27
EP0918760A1 (en) 1999-06-02
AR005008A1 (es) 1999-04-07
AU704506B2 (en) 1999-04-22
GB9526511D0 (en) 1996-02-28
CZ288704B6 (cs) 2001-08-15
EP0918760B1 (en) 2001-11-28
MX9804828A (es) 1998-09-30
IL142502A0 (en) 2002-03-10
NO982927D0 (no) 1998-06-23
EE9800193A (et) 1998-12-15
KR19990076688A (ko) 1999-10-15
US5929100A (en) 1999-07-27
ATE209638T1 (de) 2001-12-15
DE69617472D1 (de) 2002-01-10
NZ325500A (en) 1999-01-28
HUP9900100A2 (hu) 1999-05-28
CZ168498A3 (cs) 1998-09-16
JP2000502681A (ja) 2000-03-07

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Legal Events

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Effective date: 20011213