IL142460A0 - A vitreous form of 8-[3-[n-[(e)-3-(6-acetamidopyridin-3-yl) acryloyl-glycyl] -n-methylamino] -2,6-dichlorobenzyloxy]-2-methylquinoline - Google Patents
A vitreous form of 8-[3-[n-[(e)-3-(6-acetamidopyridin-3-yl) acryloyl-glycyl] -n-methylamino] -2,6-dichlorobenzyloxy]-2-methylquinolineInfo
- Publication number
- IL142460A0 IL142460A0 IL14246099A IL14246099A IL142460A0 IL 142460 A0 IL142460 A0 IL 142460A0 IL 14246099 A IL14246099 A IL 14246099A IL 14246099 A IL14246099 A IL 14246099A IL 142460 A0 IL142460 A0 IL 142460A0
- Authority
- IL
- Israel
- Prior art keywords
- acetamidopyridin
- dichlorobenzyloxy
- methylquinoline
- glycyl
- acryloyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP29925298 | 1998-10-21 | ||
| PCT/JP1999/005519 WO2000023439A1 (en) | 1998-10-21 | 1999-10-07 | Vitreous form of known bradykinin antagonist |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL142460A0 true IL142460A0 (en) | 2002-03-10 |
Family
ID=17870134
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL14246099A IL142460A0 (en) | 1998-10-21 | 1999-10-07 | A vitreous form of 8-[3-[n-[(e)-3-(6-acetamidopyridin-3-yl) acryloyl-glycyl] -n-methylamino] -2,6-dichlorobenzyloxy]-2-methylquinoline |
Country Status (18)
| Country | Link |
|---|---|
| US (2) | US6509468B1 (xx) |
| EP (1) | EP1123288A1 (xx) |
| JP (1) | JP3353784B2 (xx) |
| KR (1) | KR100419404B1 (xx) |
| CN (1) | CN1144801C (xx) |
| AR (1) | AR024220A1 (xx) |
| AU (1) | AU756479B2 (xx) |
| BR (1) | BR9914785A (xx) |
| CA (1) | CA2347001A1 (xx) |
| CZ (1) | CZ20011417A3 (xx) |
| HK (1) | HK1040245B (xx) |
| HU (1) | HUP0104110A3 (xx) |
| IL (1) | IL142460A0 (xx) |
| RU (1) | RU2202550C2 (xx) |
| TR (1) | TR200101101T2 (xx) |
| TW (1) | TWI230158B (xx) |
| WO (1) | WO2000023439A1 (xx) |
| ZA (1) | ZA200102607B (xx) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001092254A1 (fr) * | 2000-05-30 | 2001-12-06 | Fujisawa Pharmaceutical Co., Ltd. | Procede permettant de remplacer des solvants contenus dans des cristaux de type clathrates |
| EP1495017A2 (en) * | 2002-04-10 | 2005-01-12 | Ortho-McNeil Pharmaceutical, Inc. | Novel heteroaryl alkylamide derivatives useful as bradykinin receptor modulators |
| TWI407960B (zh) | 2007-03-23 | 2013-09-11 | Jerini Ag | 小分子緩激肽ｂ２受體調節劑 |
| AR113839A1 (es) | 2017-11-24 | 2020-06-17 | Pharvaris B V | Antagonistas del receptor b2 de bradiquinina |
| UY38706A (es) | 2019-05-23 | 2020-12-31 | Pharvaris Gmbh | Antagonistas cíclicos del receptor b2 de bradiquinina |
| AR118983A1 (es) | 2019-05-23 | 2021-11-17 | Pharvaris Gmbh | Antagonistas cíclicos del receptor b2 de bradiquinina |
| WO2023180575A1 (en) | 2022-03-25 | 2023-09-28 | Pharvaris Gmbh | Solid composition comprising solubilised bradykinin b2-receptor antagonists |
| TW202345810A (zh) | 2022-03-25 | 2023-12-01 | 瑞士商帕法瑞斯有限責任公司 | 包含緩激肽ｂ２受體拮抗劑之固態延長釋放組成物 |
| WO2023180577A1 (en) | 2022-03-25 | 2023-09-28 | Pharvaris Gmbh | Therapeutic uses of bradykinin b2-receptor antagonists |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US558455A (en) * | 1896-04-14 | Thomas lewty | ||
| AU680870B2 (en) * | 1993-04-28 | 1997-08-14 | Astellas Pharma Inc. | New heterocyclic compounds |
| JP3049648B2 (ja) | 1993-12-13 | 2000-06-05 | 日立金属株式会社 | 加圧成形方法および加圧成形機 |
| US5958455A (en) * | 1996-02-09 | 1999-09-28 | Quadrant Holdings Cambridge Ltd | Oral solid dosage forms, methods of making same and compositions thereof |
| JPH10316677A (ja) * | 1997-05-19 | 1998-12-02 | Fujisawa Pharmaceut Co Ltd | 結 晶 |
-
1999
- 1999-10-07 BR BR9914785-8A patent/BR9914785A/pt not_active IP Right Cessation
- 1999-10-07 TR TR2001/01101T patent/TR200101101T2/xx unknown
- 1999-10-07 CN CNB998124419A patent/CN1144801C/zh not_active Expired - Fee Related
- 1999-10-07 KR KR10-2001-7003995A patent/KR100419404B1/ko not_active IP Right Cessation
- 1999-10-07 IL IL14246099A patent/IL142460A0/xx unknown
- 1999-10-07 CA CA002347001A patent/CA2347001A1/en not_active Abandoned
- 1999-10-07 RU RU2001113511/04A patent/RU2202550C2/ru not_active IP Right Cessation
- 1999-10-07 HU HU0104110A patent/HUP0104110A3/hu unknown
- 1999-10-07 CZ CZ20011417A patent/CZ20011417A3/cs unknown
- 1999-10-07 AU AU60043/99A patent/AU756479B2/en not_active Ceased
- 1999-10-07 WO PCT/JP1999/005519 patent/WO2000023439A1/en not_active Application Discontinuation
- 1999-10-07 JP JP2000577166A patent/JP3353784B2/ja not_active Expired - Fee Related
- 1999-10-07 EP EP99970660A patent/EP1123288A1/en not_active Withdrawn
- 1999-10-07 US US09/807,421 patent/US6509468B1/en not_active Expired - Fee Related
- 1999-10-12 AR ARP990105154A patent/AR024220A1/es unknown
- 1999-10-18 TW TW088117980A patent/TWI230158B/zh not_active IP Right Cessation
-
2001
- 2001-03-29 ZA ZA200102607A patent/ZA200102607B/en unknown
-
2002
- 2002-03-01 HK HK02101581.1A patent/HK1040245B/zh not_active IP Right Cessation
- 2002-11-22 US US10/301,614 patent/US7094899B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| BR9914785A (pt) | 2001-07-03 |
| US7094899B2 (en) | 2006-08-22 |
| HK1040245B (zh) | 2004-10-08 |
| KR20010075445A (ko) | 2001-08-09 |
| EP1123288A1 (en) | 2001-08-16 |
| JP2002527514A (ja) | 2002-08-27 |
| TWI230158B (en) | 2005-04-01 |
| CZ20011417A3 (cs) | 2001-09-12 |
| CA2347001A1 (en) | 2000-04-27 |
| US6509468B1 (en) | 2003-01-21 |
| AR024220A1 (es) | 2002-09-25 |
| JP3353784B2 (ja) | 2002-12-03 |
| AU6004399A (en) | 2000-05-08 |
| CN1324354A (zh) | 2001-11-28 |
| TR200101101T2 (tr) | 2001-09-21 |
| KR100419404B1 (ko) | 2004-02-21 |
| AU756479B2 (en) | 2003-01-16 |
| RU2202550C2 (ru) | 2003-04-20 |
| HUP0104110A3 (en) | 2003-01-28 |
| ZA200102607B (en) | 2002-07-01 |
| US20030120076A1 (en) | 2003-06-26 |
| HK1040245A1 (en) | 2002-05-31 |
| CN1144801C (zh) | 2004-04-07 |
| HUP0104110A2 (hu) | 2002-03-28 |
| WO2000023439A1 (en) | 2000-04-27 |
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