IL117315A - Prokinetic piperidine substituted oxadiazole derivatives their preparation and pharmaceutical compositions containing them - Google Patents

Prokinetic piperidine substituted oxadiazole derivatives their preparation and pharmaceutical compositions containing them

Info

Publication number
IL117315A
IL117315A IL11731596A IL11731596A IL117315A IL 117315 A IL117315 A IL 117315A IL 11731596 A IL11731596 A IL 11731596A IL 11731596 A IL11731596 A IL 11731596A IL 117315 A IL117315 A IL 117315A
Authority
IL
Israel
Prior art keywords
prokinetic
preparation
pharmaceutical compositions
compositions containing
oxadiazole derivatives
Prior art date
Application number
IL11731596A
Other languages
English (en)
Other versions
IL117315A0 (en
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of IL117315A0 publication Critical patent/IL117315A0/xx
Publication of IL117315A publication Critical patent/IL117315A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10—Laxatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nutrition Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
IL11731596A 1995-03-01 1996-02-29 Prokinetic piperidine substituted oxadiazole derivatives their preparation and pharmaceutical compositions containing them IL117315A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP95200501 1995-03-01

Publications (2)

Publication Number Publication Date
IL117315A0 IL117315A0 (en) 1996-06-18
IL117315A true IL117315A (en) 2000-07-26

Family

ID=8220055

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11731596A IL117315A (en) 1995-03-01 1996-02-29 Prokinetic piperidine substituted oxadiazole derivatives their preparation and pharmaceutical compositions containing them

Country Status (25)

Country Link
US (1) US5854261A (ru)
EP (1) EP0812321B1 (ru)
JP (1) JP3980056B2 (ru)
KR (1) KR100443554B1 (ru)
CN (1) CN1092656C (ru)
AR (1) AR003932A1 (ru)
AT (1) ATE384716T1 (ru)
AU (1) AU702932B2 (ru)
BR (1) BR9607316A (ru)
CA (1) CA2212893C (ru)
CZ (1) CZ286992B6 (ru)
DE (1) DE69637412T2 (ru)
EA (1) EA001084B1 (ru)
ES (1) ES2301166T3 (ru)
FI (1) FI973562A (ru)
HU (1) HUP9702395A3 (ru)
IL (1) IL117315A (ru)
MY (1) MY113584A (ru)
NO (1) NO309425B1 (ru)
NZ (1) NZ301699A (ru)
PL (1) PL183712B1 (ru)
TR (1) TR199700876T1 (ru)
TW (1) TW360653B (ru)
WO (1) WO1996026937A1 (ru)
ZA (1) ZA961652B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9603755D0 (en) * 1996-02-22 1996-04-24 Pfizer Ltd Therapeutic agents
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
US7332508B2 (en) * 2002-12-18 2008-02-19 Novo Nordisk A/S Substituted homopiperidine, piperidine or pyrrolidine derivatives
GB0910667D0 (en) * 2009-06-19 2009-08-05 Glaxo Wellcome Mfg Pte Ltd Novel compounds
BR112014001083B8 (pt) * 2011-09-19 2022-06-14 Suven Life Sciences Ltd Composto, processo para a preparação de um composto, composição farmacêutica, uso da composiçâo farmacêutica e uso do composto
WO2018081167A1 (en) * 2016-10-24 2018-05-03 Yumanity Therapeutics Compounds and uses thereof
EP3700934A4 (en) 2017-10-24 2021-10-27 Yumanity Therapeutics, Inc. COMPOUNDS AND USES OF THESE COMPOUNDS

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1183847A (en) * 1981-10-01 1985-03-12 Georges Van Daele N-(3-hydroxy-4-piperidinyl)benzamide derivatives
US5374637A (en) * 1989-03-22 1994-12-20 Janssen Pharmaceutica N.V. N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
GB9005014D0 (en) * 1990-03-06 1990-05-02 Janssen Pharmaceutica Nv N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives
JPH06509574A (ja) * 1991-08-03 1994-10-27 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー ５−ｈｔ↓４レセプターアンタゴニスト
GB9202797D0 (en) * 1992-02-11 1992-03-25 Milsom Jonathan Glazed units
CA2146930A1 (en) * 1992-10-13 1994-04-28 Francis David King Heterocyclic -esters or -amides used as 5-ht4 receptor antagonists
MX9306311A (es) * 1992-10-13 1994-04-29 Smithkline Beecham Plc Compuestos antagonistas del receptor de 5-ht4, procedimiento para su preparacion y composiciones farmaceuticas que los contienen
KR950704328A (ko) * 1992-11-05 1995-11-17 데이비드 로버츠 5-HT₄ 수용체 길항제로서의 피페리딘 유도체(Piperidine Derivatives as 5-HT₄ Receptor Antagonists)
JPH06157518A (ja) * 1992-11-27 1994-06-03 Yamanouchi Pharmaceut Co Ltd 新規なオキサジアゾール誘導体又はその塩
WO1995032965A1 (fr) * 1994-06-01 1995-12-07 Yamanouchi Pharmaceutical Co. Ltd. Derive de l'oxadiazole et composition medicinale a base de ce dernier

Also Published As

Publication number Publication date
NO973808D0 (no) 1997-08-19
MX9706622A (es) 1997-11-29
NO973808L (no) 1997-08-19
AU4718896A (en) 1996-09-18
FI973562A0 (fi) 1997-08-29
KR100443554B1 (ko) 2004-10-06
CA2212893A1 (en) 1996-09-06
US5854261A (en) 1998-12-29
ATE384716T1 (de) 2008-02-15
NO309425B1 (no) 2001-01-29
HUP9702395A2 (hu) 1999-09-28
ES2301166T3 (es) 2008-06-16
CZ286992B6 (en) 2000-08-16
PL322019A1 (en) 1998-01-05
TW360653B (en) 1999-06-11
EA199700205A1 (ru) 1998-02-26
CZ272397A3 (cs) 1998-02-18
CN1177352A (zh) 1998-03-25
JP3980056B2 (ja) 2007-09-19
JPH11501021A (ja) 1999-01-26
EA001084B1 (ru) 2000-10-30
CA2212893C (en) 2007-01-16
PL183712B1 (pl) 2002-07-31
ZA961652B (en) 1997-09-11
TR199700876T1 (xx) 1998-02-21
MY113584A (en) 2002-04-30
IL117315A0 (en) 1996-06-18
WO1996026937A1 (en) 1996-09-06
BR9607316A (pt) 1997-12-30
NZ301699A (en) 1998-02-26
EP0812321B1 (en) 2008-01-23
CN1092656C (zh) 2002-10-16
AU702932B2 (en) 1999-03-11
DE69637412D1 (de) 2008-03-13
FI973562A (fi) 1997-08-29
DE69637412T2 (de) 2009-01-22
KR19980702304A (ko) 1998-07-15
HUP9702395A3 (en) 1999-10-28
EP0812321A1 (en) 1997-12-17
AR003932A1 (es) 1998-09-30

Similar Documents

Publication Publication Date Title
IL116917A (en) Piperidine derivatives and pharmaceutical compositions containing them
IL111002A0 (en) Piperidine derivatives, their preparation and pharmaceutical compositions containing them
IL104445A0 (en) Piperidine derivatives,their preparation and pharmaceutical compositions containing them
IL116851A (en) 3-arylidene-2-oxindole derivatives and pharmaceutical compositions containing them
HUP9701281A3 (en) Piperidine derivatives as neurokinin antagonists and pharmaceutical compositions containing them
IL117860A0 (en) Substituted 1-phenyl-3-pyrazolecarboxamides their preparation and pharmaceutical compositions containing them
IL119995A0 (en) Pyrido-fused thienyl - and furanyl-oxazolidinones their preparation and pharmaceutical compositions containing them
IL116486A0 (en) Novel piperidine derivatives processes for their preparation and pharmaceutical compositions containing them
IL116957A0 (en) Substituted heterocyclic compounds their preparation and pharmaceutical compositions containing them
HUP0003362A2 (en) Piperidine derivatives and pharmaceutical compositions containing them
IL122618A0 (en) Substituted imidazolylacetonitrile compounds their preparation and pharmaceutical compositions containing them
IL122293A0 (en) Substituted 4-phenylaminothiazoles their preparation and pharmaceutical compositions containing them
IL119559A0 (en) Purin -6- one derivatives their preparation and pharmaceutical compositions containing them
IL118768A0 (en) Diphenylmethylene piperidine derivatives and pharmaceutical compositions containing them
IL115905A0 (en) Sordarin derivatives their preparation and pharmaceutical compositions containing them
IL118410A0 (en) Substituted camptothecin derivatives their preparation and pharmaceutical compositions containing them
IL117554A0 (en) Imidazoquinazolines their preparation and pharmaceutical compositions containing them
IL122705A (en) 2-(4-Susbstituted)-benzylamino-2-methyl-propanamide derivatives their preparation and pharmaceutical compositions containing them
IL117817A0 (en) N-subsituted azaheterocyclic compounds their preparation and pharmaceutical compositions containing them
IL116930A (en) 4-(1H-indol-1-YL)-1-piperidinyl derivatives their preparation and pharmaceutical compositions containing them
NZ234124A (en) Piperidine derivatives and pharmaceutical compositions
IL109751A0 (en) Piperidine derivatives, their preparation and pharmaceutical compositions containing them
ZA948689B (en) New taxicin derivatives their preparation and pharmaceutical compositions containing them
IL119371A0 (en) Sulfonylaminopyrimidines their preparation and pharmaceutical compositions containing them
IL118672A (en) Benzisothiazolyl-substituted aminomethylchromans their preparation and pharmaceutical compositions containing them

Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees