IL109376A - Pharmaceutical composition containing (R)-5-(methyl-aminosulfonylmethyl)-3-(N-methylpyrrolidin-2-yl-methyl)-1H-indole and (R)-5-(methylamino-sulfonylmethyl)-3-(pyrrolidin-2-ylmethyl)-1H-indole - Google Patents

Pharmaceutical composition containing (R)-5-(methyl-aminosulfonylmethyl)-3-(N-methylpyrrolidin-2-yl-methyl)-1H-indole and (R)-5-(methylamino-sulfonylmethyl)-3-(pyrrolidin-2-ylmethyl)-1H-indole

Info

Publication number
IL109376A
IL109376A IL10937694A IL10937694A IL109376A IL 109376 A IL109376 A IL 109376A IL 10937694 A IL10937694 A IL 10937694A IL 10937694 A IL10937694 A IL 10937694A IL 109376 A IL109376 A IL 109376A
Authority
IL
Israel
Prior art keywords
indole
methyl
aminosulfonylmethyl
sulfonylmethyl
methylpyrrolidin
Prior art date
Application number
IL10937694A
Other languages
English (en)
Other versions
IL109376A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL109376A0 publication Critical patent/IL109376A0/xx
Publication of IL109376A publication Critical patent/IL109376A/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL10937694A 1993-04-27 1994-04-21 Pharmaceutical composition containing (R)-5-(methyl-aminosulfonylmethyl)-3-(N-methylpyrrolidin-2-yl-methyl)-1H-indole and (R)-5-(methylamino-sulfonylmethyl)-3-(pyrrolidin-2-ylmethyl)-1H-indole IL109376A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5393093A 1993-04-27 1993-04-27

Publications (2)

Publication Number Publication Date
IL109376A0 IL109376A0 (en) 1994-07-31
IL109376A true IL109376A (en) 2000-10-31

Family

ID=21987528

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10937694A IL109376A (en) 1993-04-27 1994-04-21 Pharmaceutical composition containing (R)-5-(methyl-aminosulfonylmethyl)-3-(N-methylpyrrolidin-2-yl-methyl)-1H-indole and (R)-5-(methylamino-sulfonylmethyl)-3-(pyrrolidin-2-ylmethyl)-1H-indole

Country Status (29)

Country Link
EP (1) EP0696194B1 (fr)
JP (1) JP2922307B2 (fr)
KR (1) KR960701636A (fr)
CN (3) CN1509713A (fr)
AP (1) AP486A (fr)
AT (1) ATE222492T1 (fr)
AU (1) AU689469B2 (fr)
BG (1) BG61898B1 (fr)
BR (1) BR9406435A (fr)
CA (1) CA2161533C (fr)
CO (1) CO4230093A1 (fr)
CZ (1) CZ290416B6 (fr)
DE (1) DE69431201T2 (fr)
DK (1) DK0696194T3 (fr)
ES (1) ES2180573T3 (fr)
HU (1) HU222488B1 (fr)
IL (1) IL109376A (fr)
MX (1) MX9403088A (fr)
NO (1) NO308236B1 (fr)
NZ (1) NZ263614A (fr)
OA (1) OA10189A (fr)
PL (1) PL175156B1 (fr)
PT (1) PT696194E (fr)
RO (1) RO117760B1 (fr)
RU (1) RU2132683C1 (fr)
SG (1) SG43951A1 (fr)
SK (1) SK283353B6 (fr)
WO (1) WO1994025023A1 (fr)
ZA (1) ZA942805B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5545644A (en) * 1990-10-15 1996-08-13 Pfizer Inc. Indole derivatives
US5607951A (en) * 1990-10-15 1997-03-04 Pfizer Inc Indole derivatives
US5578612A (en) * 1990-10-15 1996-11-26 Pfizer Inc. Indole derivatives
US5559246A (en) * 1990-10-15 1996-09-24 Pfizer Inc. Indole derivatives
US5559129A (en) * 1990-10-15 1996-09-24 Pfizer Inc Indole derivatives
JP2860603B2 (ja) * 1993-08-31 1999-02-24 ファイザー・インク. 5−アリールインドール誘導体
GB9417310D0 (en) * 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
PT804433E (pt) * 1994-10-12 2002-12-31 Pfizer Res & Dev Derivado de indole para o tratamento da enxaqueca
GB9424471D0 (en) * 1994-12-03 1995-01-18 Pfizer Ltd Treatment of emesis
GB9510223D0 (en) * 1995-05-20 1995-07-19 Pfizer Ltd Therapeutic agent
US5945118A (en) * 1995-09-29 1999-08-31 Pfizer Inc Indole derivative for the treatment of migraine
US5773015A (en) * 1996-11-27 1998-06-30 Elizabeth Arden Co., Division Of Conopco, Inc. Method for controlling skin oils and grease
GB9706089D0 (en) * 1997-03-24 1997-05-14 Scherer Ltd R P Pharmaceutical composition
US5994352A (en) * 1998-11-13 1999-11-30 Pfizer Inc. 5-arylindole derivatives
ES2199086B1 (es) * 2002-07-31 2005-06-01 Cepa Schwarz Pharma Sl Nuevos derivados de cicloalcanodionas, procedimiento para su preparacion y sus aplicaciones farmacologicas.
KR20220137085A (ko) * 2020-02-04 2022-10-11 마인드셋 파마 인크. Cns 장애의 치료를 위한 세로토닌성 사이키델릭 작용제로서의 3-피롤리딘-인돌 유도체

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0592438B1 (fr) * 1990-10-15 1997-08-27 Pfizer Inc. Derives d'indole
GB9102579D0 (en) * 1991-01-24 1991-03-27 Glaxo Group Ltd Compositions
GB9103770D0 (en) * 1991-02-22 1991-04-10 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
AU689469B2 (en) 1998-04-02
ZA942805B (en) 1995-10-23
WO1994025023A1 (fr) 1994-11-10
ATE222492T1 (de) 2002-09-15
OA10189A (en) 1996-12-18
KR960701636A (ko) 1996-03-28
HUT73670A (en) 1996-09-30
DE69431201D1 (de) 2002-09-26
AP9400633A0 (en) 1994-04-30
HU9503089D0 (en) 1995-12-28
EP0696194A1 (fr) 1996-02-14
BG100093A (bg) 1996-04-30
RU2132683C1 (ru) 1999-07-10
AU6436094A (en) 1994-11-21
IL109376A0 (en) 1994-07-31
CZ290416B6 (cs) 2002-07-17
ES2180573T3 (es) 2003-02-16
HU222488B1 (hu) 2003-07-28
CN1515252A (zh) 2004-07-28
CZ9502802A3 (en) 1996-04-17
CO4230093A1 (es) 1995-10-19
PT696194E (pt) 2002-11-29
SK133295A3 (en) 1997-01-08
MX9403088A (es) 1997-02-28
RO117760B1 (ro) 2002-07-30
CN1509713A (zh) 2004-07-07
NO954287L (no) 1995-10-26
NZ263614A (en) 1998-02-26
PL311266A1 (en) 1996-02-05
PL175156B1 (pl) 1998-11-30
NO954287D0 (no) 1995-10-26
DE69431201T2 (de) 2002-12-05
BR9406435A (pt) 1996-01-09
BG61898B1 (bg) 1998-09-30
SG43951A1 (en) 1997-11-14
CN1121689A (zh) 1996-05-01
CA2161533C (fr) 1998-08-04
SK283353B6 (sk) 2003-06-03
NO308236B1 (no) 2000-08-21
CA2161533A1 (fr) 1994-11-10
EP0696194B1 (fr) 2002-08-21
DK0696194T3 (da) 2002-10-07
JP2922307B2 (ja) 1999-07-19
AP486A (en) 1996-04-16
JPH08504829A (ja) 1996-05-28

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees