ID30182A - PENGHAMBAT-PENGHAMBAT PIRIDOPIRIDAZINA LEBURAN DARI cGMP FOSFODIESTERASE - Google Patents
PENGHAMBAT-PENGHAMBAT PIRIDOPIRIDAZINA LEBURAN DARI cGMP FOSFODIESTERASEInfo
- Publication number
- ID30182A ID30182A IDW00200102056A ID20012056A ID30182A ID 30182 A ID30182 A ID 30182A ID W00200102056 A IDW00200102056 A ID W00200102056A ID 20012056 A ID20012056 A ID 20012056A ID 30182 A ID30182 A ID 30182A
- Authority
- ID
- Indonesia
- Prior art keywords
- pyropyroidazine
- phosphodiesterage
- cgmp
- lights
- displacement
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US12548899P | 1999-03-22 | 1999-03-22 | |
US14800999P | 1999-08-10 | 1999-08-10 |
Publications (1)
Publication Number | Publication Date |
---|---|
ID30182A true ID30182A (id) | 2001-11-08 |
Family
ID=26823624
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IDW00200102056A ID30182A (id) | 1999-03-22 | 2000-03-09 | PENGHAMBAT-PENGHAMBAT PIRIDOPIRIDAZINA LEBURAN DARI cGMP FOSFODIESTERASE |
Country Status (10)
Country | Link |
---|---|
US (1) | US6316438B1 (fr) |
EP (1) | EP1165521A4 (fr) |
JP (1) | JP2002540102A (fr) |
KR (1) | KR20020015030A (fr) |
CN (1) | CN1161341C (fr) |
AU (1) | AU765128B2 (fr) |
CA (1) | CA2368023A1 (fr) |
ID (1) | ID30182A (fr) |
UY (1) | UY26071A1 (fr) |
WO (1) | WO2000056719A1 (fr) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6548490B1 (en) * | 1997-10-28 | 2003-04-15 | Vivus, Inc. | Transmucosal administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction |
US6403597B1 (en) | 1997-10-28 | 2002-06-11 | Vivus, Inc. | Administration of phosphodiesterase inhibitors for the treatment of premature ejaculation |
US20040014761A1 (en) * | 1997-10-28 | 2004-01-22 | Place Virgil A. | Treatment of female sexual dysfunction with phosphodiesterase inhibitors |
US6613768B1 (en) * | 1999-04-30 | 2003-09-02 | Lilly Icos Llc | Treatment of female arousal disorder |
JP2004506009A (ja) * | 2000-08-11 | 2004-02-26 | ファイザー・インク | インスリン抵抗性症候群の治療 |
US6576644B2 (en) * | 2000-09-06 | 2003-06-10 | Bristol-Myers Squibb Co. | Quinoline inhibitors of cGMP phosphodiesterase |
EP2526958B1 (fr) * | 2003-06-13 | 2017-10-18 | Ironwood Pharmaceuticals, Inc. | Procédé et compositions de traitement des troubles gastro-intestinaux |
TW200534879A (en) * | 2004-03-25 | 2005-11-01 | Bristol Myers Squibb Co | Coated tablet formulation and method |
US20050256314A1 (en) * | 2004-05-04 | 2005-11-17 | Soojin Kim | Process employing controlled crystallization in forming crystals of a pharmaceutical |
US7829720B2 (en) * | 2004-05-04 | 2010-11-09 | Bristol-Myers Squibb Company | Process for preparing atazanavir bisulfate and novel forms |
US20050288343A1 (en) * | 2004-05-19 | 2005-12-29 | Andrew Rusowicz | Process of preparing substituted carbamates and intermediates thereof |
TWI354569B (en) * | 2004-05-28 | 2011-12-21 | Bristol Myers Squibb Co | Coated tablet formulation and method |
US8648100B2 (en) | 2005-04-19 | 2014-02-11 | Takeda Gmbh | Roflumilast for the treatment of pulmonary hypertension |
ES2360336T3 (es) * | 2007-06-22 | 2011-06-03 | Bristol-Myers Squibb Company | Composiciones en comprimidos que contienen atazanavir. |
PL2170292T3 (pl) * | 2007-06-22 | 2014-06-30 | Bristol Myers Squibb Holdings Ireland | Tabletkowane kompozycje zawierające atazanawir |
ES2359770T3 (es) * | 2007-06-22 | 2011-05-26 | Bristol-Myers Squibb Company | Composiciones en comprimidos que contienen atazanavir. |
EP2178513B1 (fr) * | 2007-06-22 | 2011-03-30 | Bristol-Myers Squibb Company | Compositions en comprimés contenant de l'atazanavir |
JP2011505366A (ja) | 2007-11-30 | 2011-02-24 | ワイス・エルエルシー | ホスホエステラーゼ10の阻害剤としてのアリールおよびヘテロアリール縮合イミダゾ[1,5−a]ピラジン |
US20090143361A1 (en) * | 2007-11-30 | 2009-06-04 | Elbion Gmbh | Pyrido[3,2-E]Pyrazines, Process For Preparing The Same, And Their Use As Inhibitors Of Phosphodiesterase 10 |
WO2010114904A1 (fr) | 2009-03-31 | 2010-10-07 | Arqule, Inc. | Dérivés pyrazolo-pyrrolopyridine-dione utiles dans le traitement du cancer |
EP2688890B1 (fr) * | 2011-03-22 | 2017-08-30 | Advinus Therapeutics Limited | Composés tricycliques substitués; compositions et applications médicinales correspondantes |
JP6389513B2 (ja) * | 2014-04-30 | 2018-09-12 | エア・ウォーター株式会社 | 3−クロロ−4−メトキシベンジルアミン塩酸塩含有組成物およびその製造方法 |
WO2017168174A1 (fr) | 2016-04-02 | 2017-10-05 | N4 Pharma Uk Limited | Nouvelles formes pharmaceutiques du sildénafil |
WO2018002673A1 (fr) | 2016-07-01 | 2018-01-04 | N4 Pharma Uk Limited | Nouvelles formulations d'antagonistes du récepteur de l'angiotensine ii |
CN108395377A (zh) * | 2018-01-16 | 2018-08-14 | 吴江信凯医药科技有限公司 | 一种3-氯-4-甲氧基苄胺盐酸盐的制备方法 |
US11618751B1 (en) | 2022-03-25 | 2023-04-04 | Ventus Therapeutics U.S., Inc. | Pyrido-[3,4-d]pyridazine amine derivatives useful as NLRP3 derivatives |
Family Cites Families (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3669950A (en) | 1970-12-01 | 1972-06-13 | Squibb & Sons Inc | DIPYRAZOLO{8 3,4-b:3,4d{9 -PYRIDIN-3-ONES |
US3787430A (en) | 1972-07-13 | 1974-01-22 | Squibb & Sons Inc | Derivatives of dipyrazolo(3,4-b;3',4'-d)pyridines |
US4072681A (en) | 1977-03-02 | 1978-02-07 | E. R. Squibb & Sons, Inc. | 3,7-Dihydro- and 1,7-dihydro-4H-pyrazolo[4',3':5,6]pyrido[4,3-d]pyrimidin-4-ones |
US5055465A (en) * | 1989-05-31 | 1991-10-08 | Berlex Laboratories, Inc. | Imidazoquinoxalinones, their aza analogs and process for their preparation |
US5250534A (en) | 1990-06-20 | 1993-10-05 | Pfizer Inc. | Pyrazolopyrimidinone antianginal agents |
CA2056142A1 (fr) | 1990-11-27 | 1992-05-28 | Hirotomo Masuya | Composes a base de pyridopyridazine et leur utilisation |
JP3477651B2 (ja) * | 1993-01-28 | 2003-12-10 | 武田薬品工業株式会社 | スーパーオキシドラジカルの検出・定量法 |
GB9311920D0 (en) | 1993-06-09 | 1993-07-28 | Pfizer Ltd | Therapeutic agents |
US5849741A (en) * | 1994-08-09 | 1998-12-15 | Eisai Co., Ltd. | Fused pyridazine compounds |
JP3919835B2 (ja) * | 1994-08-09 | 2007-05-30 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 縮合ピリダジン系化合物 |
JPH08143558A (ja) * | 1994-11-21 | 1996-06-04 | Fujisawa Pharmaceut Co Ltd | アミノピペラジン誘導体の新規医薬用途 |
GB9423910D0 (en) * | 1994-11-26 | 1995-01-11 | Pfizer Ltd | Therapeutic agents |
US5614530A (en) * | 1995-03-10 | 1997-03-25 | Sterling Winthrop Inc. | Substituted N-arylmethyl and heterocyclmethyl-1H-pyrazolo[3,4-b]quinolin-4-amines and compositions and methods of use thereof |
US5488055A (en) * | 1995-03-10 | 1996-01-30 | Sanofi Winthrop Inc. | Substituted N-cycloalkylmethyl-1H-pyrazolo(3,4-b)quinolin-4 amines and compositions and methods of use thereof |
JPH10114657A (ja) * | 1996-08-20 | 1998-05-06 | Eisai Co Ltd | 縮合ピリダジン系化合物の勃起機能不全症治療剤 |
CN1121220C (zh) * | 1996-08-20 | 2003-09-17 | 卫材株式会社 | 稠合哒嗪系化合物的勃起机能不全症治疗剂 |
US5874437A (en) | 1996-11-01 | 1999-02-23 | Nitromed, Inc. | Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses |
AU7553198A (en) * | 1997-06-12 | 1998-12-30 | Sumitomo Pharmaceuticals Company, Limited | Pyrazole derivatives |
US6087368A (en) | 1998-06-08 | 2000-07-11 | Bristol-Myers Squibb Company | Quinazolinone inhibitors of cGMP phosphodiesterase |
US6326379B1 (en) * | 1998-09-16 | 2001-12-04 | Bristol-Myers Squibb Co. | Fused pyridine inhibitors of cGMP phosphodiesterase |
-
2000
- 2000-03-09 AU AU37327/00A patent/AU765128B2/en not_active Ceased
- 2000-03-09 CA CA002368023A patent/CA2368023A1/fr not_active Abandoned
- 2000-03-09 KR KR1020017012014A patent/KR20020015030A/ko not_active Application Discontinuation
- 2000-03-09 WO PCT/US2000/006100 patent/WO2000056719A1/fr not_active Application Discontinuation
- 2000-03-09 ID IDW00200102056A patent/ID30182A/id unknown
- 2000-03-09 EP EP00916180A patent/EP1165521A4/fr not_active Withdrawn
- 2000-03-09 JP JP2000606580A patent/JP2002540102A/ja active Pending
- 2000-03-09 CN CNB008053766A patent/CN1161341C/zh not_active Expired - Fee Related
- 2000-03-15 US US09/526,162 patent/US6316438B1/en not_active Expired - Lifetime
- 2000-03-22 UY UY26071A patent/UY26071A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CN1161341C (zh) | 2004-08-11 |
AU765128B2 (en) | 2003-09-11 |
KR20020015030A (ko) | 2002-02-27 |
CA2368023A1 (fr) | 2000-09-28 |
EP1165521A4 (fr) | 2002-05-22 |
WO2000056719A1 (fr) | 2000-09-28 |
EP1165521A1 (fr) | 2002-01-02 |
JP2002540102A (ja) | 2002-11-26 |
CN1344257A (zh) | 2002-04-10 |
US6316438B1 (en) | 2001-11-13 |
AU3732700A (en) | 2000-10-09 |
UY26071A1 (es) | 2000-10-31 |
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