ID19401A - N-sianoimina trisiklik baru yang berguna sebagai inhibitor farnesil-protein transferase - Google Patents
N-sianoimina trisiklik baru yang berguna sebagai inhibitor farnesil-protein transferaseInfo
- Publication number
- ID19401A ID19401A IDP972631A ID972631A ID19401A ID 19401 A ID19401 A ID 19401A ID P972631 A IDP972631 A ID P972631A ID 972631 A ID972631 A ID 972631A ID 19401 A ID19401 A ID 19401A
- Authority
- ID
- Indonesia
- Prior art keywords
- protein transferase
- trisiclic
- sianoimina
- farnesil
- new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69052296A | 1996-07-31 | 1996-07-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ID19401A true ID19401A (id) | 1998-07-09 |
Family
ID=24772812
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IDP972631A ID19401A (id) | 1996-07-31 | 1997-07-29 | N-sianoimina trisiklik baru yang berguna sebagai inhibitor farnesil-protein transferase |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0915869B1 (id) |
| JP (1) | JP3153555B2 (id) |
| CN (1) | CN1117745C (id) |
| AT (1) | ATE240313T1 (id) |
| AU (1) | AU3737097A (id) |
| CA (1) | CA2261724C (id) |
| CO (1) | CO4900031A1 (id) |
| DE (1) | DE69722002T2 (id) |
| ES (1) | ES2194207T3 (id) |
| ID (1) | ID19401A (id) |
| PE (1) | PE92098A1 (id) |
| WO (1) | WO1998004545A1 (id) |
| ZA (1) | ZA976754B (id) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR200101755T2 (tr) * | 1998-12-18 | 2001-09-21 | Schering Corporation | Trisiklik farnezil protein transferaz inhibitörleri. |
| AR033680A1 (es) * | 2000-08-30 | 2004-01-07 | Schering Corp | Compuestos triciclicos utiles como inhibidores de la farnesil proteino transferasa y su uso para la manufactura de medicamentos como agentes antitumorales |
| CN102731476A (zh) * | 2012-05-29 | 2012-10-17 | 安徽宏业药业有限公司 | 含氰胍结构的苯并环庚基吡啶衍生物、制备方法、药物组合物及其医药用途 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4826853A (en) * | 1986-10-31 | 1989-05-02 | Schering Corporation | 6,11-Dihydro-11-(N-substituted-4-piperidylidene)-5H-benzo(5,6)cyclohepta(1,2-B)pyridines and compositions and methods of use |
| ES2056214T3 (es) * | 1988-04-28 | 1994-10-01 | Schering Corp | Compuestos de benzopirido-piperidina, -piperidilideno y -piperazina, composiciones, metodos de preparacion y metodos de uso. |
| IL111235A (en) * | 1993-10-15 | 2001-03-19 | Schering Plough Corp | Medicinal preparations for inhibiting protein G activity and for the treatment of malignant diseases, containing tricyclic compounds, some such new compounds and a process for the preparation of some of them |
| ES2164716T3 (es) * | 1993-10-15 | 2002-03-01 | Schering Corp | Compuestos triciclicos de carbamato utiles para inhibir la funcion de la proteina-g y para el tratamiento de enfermedades proliferativas. |
-
1997
- 1997-07-22 PE PE1997000654A patent/PE92098A1/es not_active Application Discontinuation
- 1997-07-29 CO CO97043296A patent/CO4900031A1/es unknown
- 1997-07-29 CN CN97196817A patent/CN1117745C/zh not_active Expired - Fee Related
- 1997-07-29 JP JP50895298A patent/JP3153555B2/ja not_active Expired - Fee Related
- 1997-07-29 ID IDP972631A patent/ID19401A/id unknown
- 1997-07-29 WO PCT/US1997/012923 patent/WO1998004545A1/en active IP Right Grant
- 1997-07-29 DE DE69722002T patent/DE69722002T2/de not_active Expired - Fee Related
- 1997-07-29 AU AU37370/97A patent/AU3737097A/en not_active Abandoned
- 1997-07-29 ES ES97934269T patent/ES2194207T3/es not_active Expired - Lifetime
- 1997-07-29 ZA ZA9706754A patent/ZA976754B/xx unknown
- 1997-07-29 AT AT97934269T patent/ATE240313T1/de not_active IP Right Cessation
- 1997-07-29 CA CA002261724A patent/CA2261724C/en not_active Expired - Fee Related
- 1997-07-29 EP EP97934269A patent/EP0915869B1/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| ES2194207T3 (es) | 2003-11-16 |
| EP0915869A1 (en) | 1999-05-19 |
| WO1998004545A1 (en) | 1998-02-05 |
| JP2000500783A (ja) | 2000-01-25 |
| CA2261724A1 (en) | 1998-02-05 |
| EP0915869B1 (en) | 2003-05-14 |
| CN1226246A (zh) | 1999-08-18 |
| CA2261724C (en) | 2003-05-13 |
| PE92098A1 (es) | 1998-12-31 |
| DE69722002D1 (de) | 2003-06-18 |
| CO4900031A1 (es) | 2000-03-27 |
| CN1117745C (zh) | 2003-08-13 |
| ZA976754B (en) | 1998-02-02 |
| JP3153555B2 (ja) | 2001-04-09 |
| ATE240313T1 (de) | 2003-05-15 |
| DE69722002T2 (de) | 2004-04-01 |
| AU3737097A (en) | 1998-02-20 |
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