HUT72300A - New triazolopyrimidones, their production and their use - Google Patents

New triazolopyrimidones, their production and their use Download PDF

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Publication number
HUT72300A
HUT72300A HU9501692A HU9501692A HUT72300A HU T72300 A HUT72300 A HU T72300A HU 9501692 A HU9501692 A HU 9501692A HU 9501692 A HU9501692 A HU 9501692A HU T72300 A HUT72300 A HU T72300A
Authority
HU
Hungary
Prior art keywords
formula
alkyl
group
compounds
acid
Prior art date
Application number
HU9501692A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9501692D0 (en
Inventor
Berthold Behl
Hans Peter Hofmann
Rainer Schlecker
Hans-Joerg Treiber
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of HU9501692D0 publication Critical patent/HU9501692D0/hu
Publication of HUT72300A publication Critical patent/HUT72300A/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
HU9501692A 1992-12-10 1993-11-27 New triazolopyrimidones, their production and their use HUT72300A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4241562A DE4241562A1 (de) 1992-12-10 1992-12-10 Neue Triazolopyrimidone, ihre Herstellung und Verwendung

Publications (2)

Publication Number Publication Date
HU9501692D0 HU9501692D0 (en) 1995-08-28
HUT72300A true HUT72300A (en) 1996-04-29

Family

ID=6474848

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9501692A HUT72300A (en) 1992-12-10 1993-11-27 New triazolopyrimidones, their production and their use

Country Status (22)

Country Link
US (1) US5654310A (xx)
EP (1) EP0673378B1 (xx)
JP (1) JP3490445B2 (xx)
CN (1) CN1098414A (xx)
AT (1) ATE150023T1 (xx)
AU (1) AU674371B2 (xx)
CA (1) CA2151243A1 (xx)
CZ (1) CZ144995A3 (xx)
DE (2) DE4241562A1 (xx)
DK (1) DK0673378T3 (xx)
ES (1) ES2099577T3 (xx)
FI (1) FI952856A (xx)
GR (1) GR3022980T3 (xx)
HU (1) HUT72300A (xx)
IL (1) IL107916A (xx)
MX (1) MX9307735A (xx)
NO (1) NO952291L (xx)
NZ (1) NZ258558A (xx)
PL (1) PL309329A1 (xx)
RU (1) RU95121818A (xx)
WO (1) WO1994013673A1 (xx)
ZA (1) ZA939228B (xx)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4053600A (en) * 1973-03-08 1977-10-11 Sandoz, Inc. Tricyclic 1,2,4-triazolo-quinazolines
US4128644A (en) * 1977-07-29 1978-12-05 E. R. Squibb & Sons, Inc. Pyrazolo(1,5-c)quinazoline derivatives and related compounds
DE3146599A1 (de) * 1981-11-25 1983-07-07 Basf Ag, 6700 Ludwigshafen Neue triazolochinazoline, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen
EP0217748B1 (en) * 1985-09-30 1991-02-06 Ciba-Geigy Ag 2-Substituted-e-fused-[1,2,4,]triazolo-[1,5-c]pyrimidines pharmaceutical compositions and uses thereof
US5153196A (en) * 1991-06-05 1992-10-06 Eli Lilly And Company Excitatory amino acid receptor antagonists and methods for the use thereof

Also Published As

Publication number Publication date
IL107916A0 (en) 1994-04-12
CA2151243A1 (en) 1994-06-23
WO1994013673A1 (de) 1994-06-23
IL107916A (en) 1996-09-12
EP0673378B1 (de) 1997-03-12
DK0673378T3 (da) 1997-07-21
JPH08504412A (ja) 1996-05-14
ES2099577T3 (es) 1997-05-16
EP0673378A1 (de) 1995-09-27
PL309329A1 (en) 1995-10-02
FI952856A0 (fi) 1995-06-09
FI952856A (fi) 1995-06-09
AU5628594A (en) 1994-07-04
MX9307735A (es) 1994-06-30
JP3490445B2 (ja) 2004-01-26
GR3022980T3 (en) 1997-06-30
DE59305812D1 (de) 1997-04-17
DE4241562A1 (de) 1994-06-16
NO952291D0 (no) 1995-06-09
HU9501692D0 (en) 1995-08-28
CZ144995A3 (en) 1995-12-13
RU95121818A (ru) 1997-06-10
ZA939228B (en) 1995-06-09
CN1098414A (zh) 1995-02-08
AU674371B2 (en) 1996-12-19
US5654310A (en) 1997-08-05
ATE150023T1 (de) 1997-03-15
NZ258558A (en) 1997-06-24
NO952291L (no) 1995-06-09

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DFA9 Temporary protection cancelled due to abandonment