HUT61465A - Process for producing pharmaceutical compositions having 5-ht3 agonist activity and comprising 4-amino-1-(2-pyridyl)-piperidine derivatives - Google Patents

Process for producing pharmaceutical compositions having 5-ht3 agonist activity and comprising 4-amino-1-(2-pyridyl)-piperidine derivatives

Info

Publication number
HUT61465A
HUT61465A HU929200940A HU9200940A HUT61465A HU T61465 A HUT61465 A HU T61465A HU 929200940 A HU929200940 A HU 929200940A HU 9200940 A HU9200940 A HU 9200940A HU T61465 A HUT61465 A HU T61465A
Authority
HU
Hungary
Prior art keywords
pyridyl
amino
pharmaceutical compositions
agonist activity
piperidine derivatives
Prior art date
Application number
HU929200940A
Other languages
English (en)
Other versions
HU9200940D0 (en
Inventor
Fur Gerard Le
Alberto Bianchetti
Antonina Guidice
Tiziano Croci
Philippe Soubrie
Original Assignee
Sanofi Elf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9103735A external-priority patent/FR2674435B1/fr
Priority claimed from FR9110890A external-priority patent/FR2674752B1/fr
Application filed by Sanofi Elf filed Critical Sanofi Elf
Publication of HU9200940D0 publication Critical patent/HU9200940D0/hu
Publication of HUT61465A publication Critical patent/HUT61465A/hu

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10—Laxatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
HU929200940A 1991-03-27 1992-03-26 Process for producing pharmaceutical compositions having 5-ht3 agonist activity and comprising 4-amino-1-(2-pyridyl)-piperidine derivatives HUT61465A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9103735A FR2674435B1 (fr) 1991-03-27 1991-03-27 Utilisation de 4-amino-1-(2-pyridyl) piperidines pour la preparation d'agents psychotropes.
FR9110890A FR2674752B1 (fr) 1991-09-03 1991-09-03 Utilisation de 4-amino-1-(2-pyridyl)piperidines pour la preparation de medicaments pour le traitement et la prophylaxie des etats decoulant d'un dysfonctionnement du systeme serotoninergique.
EP91402753 1991-10-15

Publications (2)

Publication Number Publication Date
HU9200940D0 HU9200940D0 (en) 1992-05-28
HUT61465A true HUT61465A (en) 1993-01-28

Family

ID=27234263

Family Applications (1)

Application Number Title Priority Date Filing Date
HU929200940A HUT61465A (en) 1991-03-27 1992-03-26 Process for producing pharmaceutical compositions having 5-ht3 agonist activity and comprising 4-amino-1-(2-pyridyl)-piperidine derivatives

Country Status (9)

Country Link
US (1) US5604245A (hu)
EP (1) EP0506545B1 (hu)
JP (1) JP2603023B2 (hu)
AT (1) ATE175113T1 (hu)
AU (1) AU656563B2 (hu)
CA (1) CA2063941A1 (hu)
DE (1) DE69228017D1 (hu)
HU (1) HUT61465A (hu)
SG (1) SG47477A1 (hu)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0591030A3 (fr) * 1992-09-25 1994-04-27 Sanofi 1-Hétéroaryl-azétidines et -pyrrolidines comme 5-HT3 agonistes
CA2106840A1 (en) * 1992-09-25 1994-03-26 Marco Baroni Heteroarylazetidines and -pyrrolidines, process for their preparation and pharmaceutical compositions containing them
EP0647639A1 (fr) * 1993-10-11 1995-04-12 Sanofi Hétéroarylpipéridines, procédé pour leur préparation et compositions pharmaceutiques les contenant
CA2133855A1 (en) * 1993-10-11 1995-04-12 Marco Baroni Heteroarylpiperidines, process for their preparation and pharmaceutical compositions in which they are present
US6833370B1 (en) * 1999-05-21 2004-12-21 Abbott Laboratories Heterocycle substituted aminoazacycles useful as central nervous system agents
KR100715344B1 (ko) * 1999-11-23 2007-05-08 얀센 파마슈티카 엔.브이. 기저부 이완을 위한 5ｈｔ3 효능제의 용도
CN1395575A (zh) 2000-01-20 2003-02-05 卫材株式会社 新的哌啶化合物及其药物
US20040191312A1 (en) * 2002-12-31 2004-09-30 Donna Oksenberg 5-HT3 receptor agonists as neuroprotectors
PL3646886T3 (pl) 2017-06-28 2024-03-04 Osaka University Leczenie bólu agonistą receptora serotoninowego 3
WO2022118783A1 (ja) * 2020-12-04 2022-06-09 国立大学法人大阪大学 治療抵抗性うつ病または緊急性を有するうつ病の症状を治療するための組成物

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2459240A1 (fr) * 1979-06-21 1981-01-09 Cm Ind Aminopiperidines anorexigenes, procede pour leur preparation, intermediaires dans ledit procede et medicaments qui les contiennent

Also Published As

Publication number Publication date
ATE175113T1 (de) 1999-01-15
AU656563B2 (en) 1995-02-09
EP0506545A2 (fr) 1992-09-30
JP2603023B2 (ja) 1997-04-23
SG47477A1 (en) 1998-04-17
AU1316892A (en) 1992-10-01
JPH07145166A (ja) 1995-06-06
EP0506545A3 (en) 1993-01-27
US5604245A (en) 1997-02-18
HU9200940D0 (en) 1992-05-28
CA2063941A1 (en) 1992-09-28
DE69228017D1 (de) 1999-02-11
EP0506545B1 (fr) 1998-12-30

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Legal Events

Date Code Title Description
DFC4 Cancellation of temporary protection due to refusal