DE69228017D1 - Verwendung von 4-Amino-1-(2-Pyridyl)Piperidinen als 5-HT3-Agonisten zur Behandlung und Verhütung von serotoninergen Dysfunktionen - Google Patents
Verwendung von 4-Amino-1-(2-Pyridyl)Piperidinen als 5-HT3-Agonisten zur Behandlung und Verhütung von serotoninergen DysfunktionenInfo
- Publication number
- DE69228017D1 DE69228017D1 DE69228017T DE69228017T DE69228017D1 DE 69228017 D1 DE69228017 D1 DE 69228017D1 DE 69228017 T DE69228017 T DE 69228017T DE 69228017 T DE69228017 T DE 69228017T DE 69228017 D1 DE69228017 D1 DE 69228017D1
- Authority
- DE
- Germany
- Prior art keywords
- serotoninergic
- piperidines
- pyridyl
- amino
- treatment
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9103735A FR2674435B1 (fr) | 1991-03-27 | 1991-03-27 | Utilisation de 4-amino-1-(2-pyridyl) piperidines pour la preparation d'agents psychotropes. |
FR9110890A FR2674752B1 (fr) | 1991-09-03 | 1991-09-03 | Utilisation de 4-amino-1-(2-pyridyl)piperidines pour la preparation de medicaments pour le traitement et la prophylaxie des etats decoulant d'un dysfonctionnement du systeme serotoninergique. |
EP91402753 | 1991-10-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
DE69228017D1 true DE69228017D1 (de) | 1999-02-11 |
Family
ID=27234263
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69228017T Expired - Lifetime DE69228017D1 (de) | 1991-03-27 | 1992-03-24 | Verwendung von 4-Amino-1-(2-Pyridyl)Piperidinen als 5-HT3-Agonisten zur Behandlung und Verhütung von serotoninergen Dysfunktionen |
Country Status (9)
Country | Link |
---|---|
US (1) | US5604245A (de) |
EP (1) | EP0506545B1 (de) |
JP (1) | JP2603023B2 (de) |
AT (1) | ATE175113T1 (de) |
AU (1) | AU656563B2 (de) |
CA (1) | CA2063941A1 (de) |
DE (1) | DE69228017D1 (de) |
HU (1) | HUT61465A (de) |
SG (1) | SG47477A1 (de) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2106840A1 (en) * | 1992-09-25 | 1994-03-26 | Marco Baroni | Heteroarylazetidines and -pyrrolidines, process for their preparation and pharmaceutical compositions containing them |
EP0591030A3 (de) * | 1992-09-25 | 1994-04-27 | Sanofi | 1-Heteroaryl-azetidine und -pyrrolidine als 5-HT3-Agoniste |
EP0647639A1 (de) * | 1993-10-11 | 1995-04-12 | Sanofi | Heteroarylpiperidinen, Verfahren zu deren Herstellung und diese enthaltende pharmazeutischen Zusammenstellungen |
NZ264634A (en) * | 1993-10-11 | 1995-12-21 | Sanofi Sa | 1-heteroaryl-4-alkyl-4-amino-piperidines and pharmaceutical compositions thereof and piperidine precursors |
US6833370B1 (en) | 1999-05-21 | 2004-12-21 | Abbott Laboratories | Heterocycle substituted aminoazacycles useful as central nervous system agents |
EP1235565B1 (de) * | 1999-11-23 | 2005-12-28 | Janssen Pharmaceutica N.V. | Verwendung von 5ht3 antagonisten zur fundusentspannung |
CA2398388A1 (en) * | 2000-01-20 | 2001-07-26 | Koji Kato | Novel piperidine compound and pharmaceutical thereof |
US20040191312A1 (en) * | 2002-12-31 | 2004-09-30 | Donna Oksenberg | 5-HT3 receptor agonists as neuroprotectors |
JP7090344B2 (ja) | 2017-06-28 | 2022-06-24 | 国立大学法人大阪大学 | セロトニン3受容体アゴニストによる疼痛の治療 |
WO2022118783A1 (ja) * | 2020-12-04 | 2022-06-09 | 国立大学法人大阪大学 | 治療抵抗性うつ病または緊急性を有するうつ病の症状を治療するための組成物 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2459240A1 (fr) * | 1979-06-21 | 1981-01-09 | Cm Ind | Aminopiperidines anorexigenes, procede pour leur preparation, intermediaires dans ledit procede et medicaments qui les contiennent |
-
1992
- 1992-03-24 EP EP92400792A patent/EP0506545B1/de not_active Expired - Lifetime
- 1992-03-24 AT AT92400792T patent/ATE175113T1/de not_active IP Right Cessation
- 1992-03-24 DE DE69228017T patent/DE69228017D1/de not_active Expired - Lifetime
- 1992-03-24 SG SG1996002112A patent/SG47477A1/en unknown
- 1992-03-25 AU AU13168/92A patent/AU656563B2/en not_active Ceased
- 1992-03-25 CA CA002063941A patent/CA2063941A1/en not_active Abandoned
- 1992-03-26 HU HU929200940A patent/HUT61465A/hu unknown
- 1992-03-26 JP JP4068374A patent/JP2603023B2/ja not_active Expired - Lifetime
- 1992-03-27 US US07/858,483 patent/US5604245A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
JPH07145166A (ja) | 1995-06-06 |
CA2063941A1 (en) | 1992-09-28 |
US5604245A (en) | 1997-02-18 |
EP0506545A3 (en) | 1993-01-27 |
SG47477A1 (en) | 1998-04-17 |
ATE175113T1 (de) | 1999-01-15 |
HUT61465A (en) | 1993-01-28 |
EP0506545A2 (de) | 1992-09-30 |
HU9200940D0 (en) | 1992-05-28 |
JP2603023B2 (ja) | 1997-04-23 |
EP0506545B1 (de) | 1998-12-30 |
AU656563B2 (en) | 1995-02-09 |
AU1316892A (en) | 1992-10-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8332 | No legal effect for de |