HUT59676A - Process for producing piperazinyl-alkyl-carbonyl derivatives of condensed heterocyclic compounds and pharmaceutical compositions containing them - Google Patents
Process for producing piperazinyl-alkyl-carbonyl derivatives of condensed heterocyclic compounds and pharmaceutical compositions containing themInfo
- Publication number
- HUT59676A HUT59676A HU913643A HU364391A HUT59676A HU T59676 A HUT59676 A HU T59676A HU 913643 A HU913643 A HU 913643A HU 364391 A HU364391 A HU 364391A HU T59676 A HUT59676 A HU T59676A
- Authority
- HU
- Hungary
- Prior art keywords
- producing
- condensed heterocyclic
- piperazinyl
- alkyl
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP31989790 | 1990-11-22 | ||
| JP7028691 | 1991-01-14 | ||
| JP20935891 | 1991-08-21 | ||
| JP24376891 | 1991-09-24 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| HU913643D0 HU913643D0 (en) | 1992-02-28 |
| HUT59676A true HUT59676A (en) | 1992-06-29 |
| HU214573B HU214573B (hu) | 2000-04-28 |
Family
ID=27465225
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU643/91A HU214573B (hu) | 1990-11-22 | 1991-11-21 | Kondenzált heterogyűrűs vegyületek piperidinil-alkil-karbonil-származékai, ezeket tartalmazó gyógyászati készítmények és eljárás előállításukra |
| HU95P/P00115P HU211130A9 (en) | 1990-11-22 | 1995-04-28 | Condensed heterocyclic compounds, their production and use |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU95P/P00115P HU211130A9 (en) | 1990-11-22 | 1995-04-28 | Condensed heterocyclic compounds, their production and use |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US5273974A (hu) |
| EP (1) | EP0487071B1 (hu) |
| JP (1) | JP2650537B2 (hu) |
| KR (1) | KR100211437B1 (hu) |
| CN (1) | CN1036458C (hu) |
| AT (1) | ATE124695T1 (hu) |
| AU (1) | AU643337B2 (hu) |
| CA (1) | CA2055947C (hu) |
| DE (1) | DE69111029T2 (hu) |
| DK (1) | DK0487071T3 (hu) |
| ES (1) | ES2074205T3 (hu) |
| FI (2) | FI102965B (hu) |
| GR (1) | GR3017366T3 (hu) |
| HU (2) | HU214573B (hu) |
| IE (1) | IE68346B1 (hu) |
| NO (1) | NO179868C (hu) |
| NZ (1) | NZ240676A (hu) |
| RU (1) | RU2095361C1 (hu) |
| TW (1) | TW197435B (hu) |
Families Citing this family (37)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5965574A (en) * | 1996-08-13 | 1999-10-12 | Chen; Yuhpyng Liang | Heteroaryl amines as novel acetylcholinesterase inhibitors |
| TW263504B (hu) * | 1991-10-03 | 1995-11-21 | Pfizer | |
| TW218875B (hu) * | 1992-03-09 | 1994-01-11 | Takeda Pharm Industry Co Ltd | |
| US5462934A (en) * | 1992-03-09 | 1995-10-31 | Takeda Chemical Industries | Condensed heterocyclic ketone derivatives and their use |
| ATE194982T1 (de) | 1992-04-24 | 2000-08-15 | Takeda Chemical Industries Ltd | Benzoxazepin-derivate als cholinesterase- inhibitoren |
| TW248556B (hu) * | 1993-01-18 | 1995-06-01 | Takeda Pharm Industry Co | |
| US5620973A (en) * | 1993-11-30 | 1997-04-15 | Takeda Chemical Industries, Ltd. | Tetracyclic condensed heterocyclic compounds and their use |
| US5674891A (en) * | 1994-07-27 | 1997-10-07 | The Procter & Gamble Company | Dihydrobenzothiophene compounds useful as anti-inflammatory agents |
| JPH10506615A (ja) * | 1994-07-27 | 1998-06-30 | ザ、プロクター、エンド、ギャンブル、カンパニー | 抗炎症剤として有用なジヒドロベンゾフラン及び関連化合物 |
| US5672620A (en) * | 1996-02-01 | 1997-09-30 | The Procter & Gamble Company | Dihydrobenzofuran and related compounds useful as anti-inflammatory agents |
| US5684031A (en) * | 1996-02-01 | 1997-11-04 | The Procter & Gamble Company | Dihydrobenzofuran and related compounds useful as anti-inflammatory agents |
| US6251938B1 (en) | 1996-12-18 | 2001-06-26 | Teva Pharmaceutical Industries, Ltd., | Phenylethylamine derivatives |
| DK0966435T3 (da) | 1996-12-18 | 2005-08-15 | Teva Pharma | Aminoindanderivater |
| US5962535A (en) * | 1997-01-17 | 1999-10-05 | Takeda Chemical Industries, Ltd. | Composition for alzheimer's disease |
| EP0952826B1 (en) * | 1997-01-17 | 2001-11-14 | Takeda Chemical Industries, Ltd. | Idebenone containing combination agent for treating alzheimer's disease |
| CA2282390A1 (en) | 1997-04-17 | 1998-10-22 | Yukio Fujisawa | Thermogenic composition and benzazepine thermogenics |
| EP1079816A2 (en) | 1998-04-23 | 2001-03-07 | Takeda Chemical Industries, Ltd. | Pharmaceutical composition for neurotrophic action |
| WO2000018391A1 (fr) | 1998-09-30 | 2000-04-06 | Takeda Chemical Industries, Ltd. | Medicaments qui ameliorent le pouvoir de vidange de la vessie |
| KR100694682B1 (ko) * | 1999-03-03 | 2007-03-13 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 4-치환 피페리딘 유도체 불화물 |
| WO2002002530A1 (fr) * | 2000-07-04 | 2002-01-10 | Takeda Chemical Industries, Ltd. | Antagoniste de gpr14 |
| US20040053826A1 (en) * | 2000-08-10 | 2004-03-18 | Yoshio Matsumoto | Uses of polypeptides |
| CN1317276C (zh) * | 2000-09-29 | 2007-05-23 | 中国科学院上海药物研究所 | 一类吲哚基哌啶类化合物及其制备方法和用途 |
| KR20060005009A (ko) | 2001-12-28 | 2006-01-16 | 다케다 야쿠힌 고교 가부시키가이샤 | 배뇨 장애 예방제/치료제 |
| US20040010038A1 (en) * | 2002-02-27 | 2004-01-15 | Eran Blaugrund | Propargylamino indan derivatives and propargylamino tetralin derivatives as brain-selective MAO inhibitors |
| ES2379948T3 (es) | 2002-06-14 | 2012-05-07 | Toyama Chemical Co., Ltd. | Composición medicinal que comprende Tacrine o Donepezil para mejorar la función cerebral |
| NZ540148A (en) | 2002-12-20 | 2007-11-30 | Glaxo Group Ltd | Benzazepine derivatives for the treatment of neurological disorders |
| US20080045500A1 (en) * | 2004-07-01 | 2008-02-21 | Eisai R&D Management Co., Ltd. | Nerve Regeneration Stimulator |
| US20080188510A1 (en) * | 2005-05-23 | 2008-08-07 | Eisai R & D Management Co., Ltd. | Novel methods using zonisamide |
| ES2632638T3 (es) * | 2005-12-09 | 2017-09-14 | Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. | Ladostigilo de baja dosis para el tratamiento de la deficiencia cognitiva |
| TW200744576A (en) * | 2006-02-24 | 2007-12-16 | Teva Pharma | Propargylated aminoindans, processes for preparation, and uses thereof |
| CN102099339A (zh) * | 2008-07-18 | 2011-06-15 | 武田药品工业株式会社 | 苯并氮杂衍生物及其作为组胺h3拮抗剂的用途 |
| CA2789014C (en) | 2010-02-09 | 2019-01-15 | Michela Gallagher | Methods and compositions for improving cognitive function |
| JP6440625B2 (ja) | 2012-11-14 | 2018-12-19 | ザ・ジョンズ・ホプキンス・ユニバーシティー | 精神分裂病を処置するための方法および組成物 |
| CA2904767C (en) | 2013-03-15 | 2022-06-21 | Agenebio, Inc. | Methods and compositions for improving cognitive function |
| WO2014144663A1 (en) | 2013-03-15 | 2014-09-18 | The Johns Hopkins University | Methods and compositions for improving cognitive function |
| WO2016191288A1 (en) | 2015-05-22 | 2016-12-01 | Agenebio, Inc. | Extended release pharmaceutical compositions of levetiracetam |
| CN109880635B (zh) * | 2019-03-19 | 2021-02-02 | 石家庄晶奥量新材料有限公司 | 含有二苯并呋喃并含氧杂环类液晶化合物和组合物及应用 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2334358A1 (fr) * | 1975-12-12 | 1977-07-08 | Sogeras | Nouveaux medicaments derives de l'indole |
| US4208417A (en) * | 1978-06-29 | 1980-06-17 | Pharmindustrie | Indole derivatives and their use as anxiolytics |
| DK623586A (da) * | 1985-12-27 | 1987-06-28 | Eisai Co Ltd | Piperidinderivater eller salte deraf og farmaceutiske kompositioner indeholdende forbindelserne |
| KR910006138B1 (ko) * | 1986-09-30 | 1991-08-16 | 에자이 가부시끼가이샤 | 환상아민 유도체 |
| FI95572C (fi) * | 1987-06-22 | 1996-02-26 | Eisai Co Ltd | Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi |
| FR2640266B2 (fr) * | 1988-07-12 | 1992-07-10 | Synthelabo | Derives de (hydroxy-1 piperidinyl-2 alkyl) indolones-2, quinoleinones-2, benzo(b)azepinones-2 et benzimidazolones-2, leur preparation et leur application en therapeutique |
| JP2969359B2 (ja) * | 1989-01-13 | 1999-11-02 | 武田薬品工業株式会社 | 環状アミン化合物 |
| CA2023492A1 (en) * | 1989-08-31 | 1991-03-01 | Barry Clifford Lange | Herbicidal glutarimides |
| US5109002A (en) * | 1989-09-08 | 1992-04-28 | Du Pont Merck Pharmaceutical Company | Antipsychotic 1-cycloalkylpiperidines |
-
1991
- 1991-11-19 TW TW080109059A patent/TW197435B/zh active
- 1991-11-20 NZ NZ240676A patent/NZ240676A/xx unknown
- 1991-11-20 JP JP3305062A patent/JP2650537B2/ja not_active Expired - Fee Related
- 1991-11-21 AU AU88045/91A patent/AU643337B2/en not_active Ceased
- 1991-11-21 CA CA002055947A patent/CA2055947C/en not_active Expired - Fee Related
- 1991-11-21 HU HU643/91A patent/HU214573B/hu not_active IP Right Cessation
- 1991-11-21 DE DE69111029T patent/DE69111029T2/de not_active Expired - Fee Related
- 1991-11-21 DK DK91119818.2T patent/DK0487071T3/da active
- 1991-11-21 RU SU915010491A patent/RU2095361C1/ru active
- 1991-11-21 AT AT91119818T patent/ATE124695T1/de not_active IP Right Cessation
- 1991-11-21 IE IE405391A patent/IE68346B1/en not_active IP Right Cessation
- 1991-11-21 ES ES91119818T patent/ES2074205T3/es not_active Expired - Lifetime
- 1991-11-21 EP EP91119818A patent/EP0487071B1/en not_active Expired - Lifetime
- 1991-11-21 NO NO914558A patent/NO179868C/no not_active IP Right Cessation
- 1991-11-21 FI FI915488A patent/FI102965B/fi active
- 1991-11-22 CN CN 91110950 patent/CN1036458C/zh not_active Expired - Fee Related
- 1991-11-22 KR KR1019910020944A patent/KR100211437B1/ko not_active IP Right Cessation
- 1991-11-22 US US07/796,430 patent/US5273974A/en not_active Expired - Lifetime
-
1995
- 1995-04-28 HU HU95P/P00115P patent/HU211130A9/hu unknown
- 1995-09-13 GR GR950402483T patent/GR3017366T3/el unknown
-
1998
- 1998-11-10 FI FI982436A patent/FI982436A/fi unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| HMM4 | Cancellation of final prot. due to non-payment of fee |