HUT48818A - Process for production of analgetic medical preparatives containing as active substance derivatives of pirido-pirimidin or pirimido-pirimidin - Google Patents

Process for production of analgetic medical preparatives containing as active substance derivatives of pirido-pirimidin or pirimido-pirimidin

Info

Publication number
HUT48818A
HUT48818A HU885883A HU588388A HUT48818A HU T48818 A HUT48818 A HU T48818A HU 885883 A HU885883 A HU 885883A HU 588388 A HU588388 A HU 588388A HU T48818 A HUT48818 A HU T48818A
Authority
HU
Hungary
Prior art keywords
pirimidin
pirimido
pirido
analgetic
production
Prior art date
Application number
HU885883A
Other languages
English (en)
Other versions
HU203199B (en
Inventor
Peter Raddatz
Wolf-Dietrich Weber
Andrew Barber
Hans-Peter Wolf
Christoph Seyfried
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of HUT48818A publication Critical patent/HUT48818A/hu
Publication of HU203199B publication Critical patent/HU203199B/hu

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
HU885883A 1987-11-16 1988-11-15 Process for producing pharmaceutical compositions with analgetic effect and comprising pyridopyrimidine derivatives as active ingredient HU203199B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19873738844 DE3738844A1 (de) 1987-11-16 1987-11-16 Analgetikum

Publications (2)

Publication Number Publication Date
HUT48818A true HUT48818A (en) 1989-07-28
HU203199B HU203199B (en) 1991-06-28

Family

ID=6340578

Family Applications (1)

Application Number Title Priority Date Filing Date
HU885883A HU203199B (en) 1987-11-16 1988-11-15 Process for producing pharmaceutical compositions with analgetic effect and comprising pyridopyrimidine derivatives as active ingredient

Country Status (15)

Country Link
US (1) US4950648A (hu)
EP (1) EP0316668B1 (hu)
JP (1) JPH01160919A (hu)
KR (1) KR890007741A (hu)
AT (1) ATE89481T1 (hu)
AU (1) AU616695B2 (hu)
CA (1) CA1317549C (hu)
DE (2) DE3738844A1 (hu)
ES (1) ES2069541T3 (hu)
GR (1) GR3007918T3 (hu)
HU (1) HU203199B (hu)
IE (1) IE61301B1 (hu)
PH (1) PH25353A (hu)
PT (1) PT89000B (hu)
ZA (1) ZA888574B (hu)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2807577B2 (ja) * 1990-06-15 1998-10-08 エーザイ株式会社 環状アミド誘導体
US5095019A (en) * 1990-08-27 1992-03-10 Hoechst-Roussel Pharmaceuticals Inc. 4-substituted dihydropyrido(4,3-D)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders
US6166019A (en) * 1998-07-16 2000-12-26 Abbott Laboratories Piperazinyl pyrimidine dione compounds selective for adrenoceptors
WO2001089508A1 (en) * 2000-05-24 2001-11-29 University Of Kentucky Research Foundation Novel long acting, reversible veterinary sedative and analgesic and method of use
FR2832711B1 (fr) 2001-11-26 2004-01-30 Warner Lambert Co Derives de triazolo [4,3-a] pyrido [2,3-d] pyrimidin-5-ones, compositions les contenant, procede de preparation et utilisation
JP2007509865A (ja) * 2003-10-30 2007-04-19 ティオガ ファーマシュウティカルズ,インコーポレイテッド 神経障害の治療における選択的オピエート受容体調節物質の使用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB843073A (en) * 1958-05-09 1960-08-04 Toraude Lab 2-methyl-3-orthotolyl-4-quinazolone and acid addition salts thereof
FR1043M (fr) * 1960-12-28 1962-02-09 Soc Ind Fab Antibiotiques Sifa Dérivé de la quinazolone et ses sels, utilisés en thérapeutique.
US3919425A (en) * 1971-04-09 1975-11-11 Miles Lab Method of producing vasodilation using certain 3-substituted-quinazoline derivatives
DE2143117A1 (de) * 1971-08-28 1973-03-08 Troponwerke Dinklage & Co Neue 2-methyl-3-geschweifte klammer auf 3- eckige klammer auf 4-phenylpiperazinyl(1) eckige klammer zu -2-hydroxypropyl geschweifte klammer zu chinazolinon-(4)derivate, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln
US4335127A (en) * 1979-01-08 1982-06-15 Janssen Pharmaceutica, N.V. Piperidinylalkyl quinazoline compounds, composition and method of use
DE3012837A1 (de) * 1979-04-10 1980-10-30 Sandoz Ag Analgetische und myotonolytische praeparate
US4485107A (en) * 1982-11-01 1984-11-27 Janssen Pharmaceutica N.V. [[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones
DE3601731A1 (de) * 1986-01-22 1987-07-23 Merck Patent Gmbh Pyrimidinderivate

Also Published As

Publication number Publication date
PH25353A (en) 1991-05-13
HU203199B (en) 1991-06-28
AU2510788A (en) 1989-05-18
ES2069541T3 (es) 1995-05-16
GR3007918T3 (hu) 1993-08-31
ZA888574B (en) 1989-08-30
IE883417L (en) 1989-05-16
AU616695B2 (en) 1991-11-07
EP0316668A2 (de) 1989-05-24
EP0316668A3 (en) 1990-09-19
JPH01160919A (ja) 1989-06-23
CA1317549C (en) 1993-05-11
EP0316668B1 (de) 1993-05-19
IE61301B1 (en) 1994-10-19
PT89000A (pt) 1988-12-01
US4950648A (en) 1990-08-21
DE3881164D1 (de) 1993-06-24
ATE89481T1 (de) 1993-06-15
DE3738844A1 (de) 1989-05-24
PT89000B (pt) 1993-02-26
KR890007741A (ko) 1989-07-05

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Legal Events

Date Code Title Description
HMM4 Cancellation of final prot. due to non-payment of fee