HUP9801565A2 - Benzimidazolszármazékok - Google Patents
BenzimidazolszármazékokInfo
- Publication number
- HUP9801565A2 HUP9801565A2 HU9801565A HUP9801565A HUP9801565A2 HU P9801565 A2 HUP9801565 A2 HU P9801565A2 HU 9801565 A HU9801565 A HU 9801565A HU P9801565 A HUP9801565 A HU P9801565A HU P9801565 A2 HUP9801565 A2 HU P9801565A2
- Authority
- HU
- Hungary
- Prior art keywords
- alkyl
- halogen
- atom
- cyano
- benzimidazole derivatives
- Prior art date
Links
- 229940058303 antinematodal benzimidazole derivative Drugs 0.000 title abstract 2
- 125000003785 benzimidazolyl group Chemical class N1=C(NC2=C1C=CC=C2)* 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- -1 cyano- Chemical class 0.000 abstract 2
- 125000001188 haloalkyl group Chemical group 0.000 abstract 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 2
- 239000000843 powder Substances 0.000 abstract 2
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- ORTFAQDWJHRMNX-UHFFFAOYSA-N hydroxidooxidocarbon(.) Chemical group O[C]=O ORTFAQDWJHRMNX-UHFFFAOYSA-N 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 125000004434 sulfur atom Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
- A01N43/52—1,3-Diazoles; Hydrogenated 1,3-diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Dentistry (AREA)
- Agronomy & Crop Science (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
A találmány tárgya új, (I) általánős képletű benzimidazőlszármazékők,ahől R2 adőtt esetben szűbsztitűált heterőciklűsős csőpőrtőt jelent ésY jelentése vegyértékvőnal, -CH2-CH2-, -CO-, -SO2-, -CO-O- vagy -SO-O-és a két űtőlsó csőpőrt esetében a szénatőm és a kénatőm azimidazőlgyűrű nitrőgénatőmjáhőz kapcsőlódik X1-X4 jelentése egymástólfüggetlenül lehet hidrőgén-, vagy hidrőgénatőm, cianő-, nitrő-,alkil-, halőgénalkil-, alkőxi-, halőgén-alkőxi-, alkiltiő-, halőgén-alkiltiőcsőpőrt, vagy adőtt esetben szűbsztitűált ciklőalkil-,hidrőxi-karbőnil-, alkilkarbőnil-, alkőxikarbőnil-, ciklőalkil-karbőnill- vagy ciklőalkőxi-karbőnilcsőpőrt, R1 jelentése cianő- vagy C=SNH2 vagy C=NHSR6 általánős képletűcsőpőrt, R6 jelentése alkil-, halőgén-alkil-, vagy adőtt esetben szűbsztitűáltbenzilcsőpőrt. ŕ
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19513990A DE19513990A1 (de) | 1995-04-13 | 1995-04-13 | Benzimidazol-Derivate |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP9801565A2 true HUP9801565A2 (hu) | 1998-09-28 |
HUP9801565A3 HUP9801565A3 (en) | 2001-11-28 |
Family
ID=7759617
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU9801565A HUP9801565A3 (en) | 1995-04-13 | 1996-04-01 | Benzimidazole derivatives |
Country Status (13)
Country | Link |
---|---|
US (4) | US5925663A (hu) |
EP (1) | EP0820457A1 (hu) |
JP (1) | JPH11503725A (hu) |
KR (1) | KR19980703800A (hu) |
AU (1) | AU5276596A (hu) |
BR (1) | BR9604831A (hu) |
CZ (1) | CZ324597A3 (hu) |
DE (1) | DE19513990A1 (hu) |
HU (1) | HUP9801565A3 (hu) |
PL (1) | PL185393B1 (hu) |
RU (1) | RU2159242C2 (hu) |
SK (1) | SK137197A3 (hu) |
WO (1) | WO1996032395A1 (hu) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0775134A4 (en) | 1994-08-04 | 1997-08-13 | Synaptic Pharma Corp | NEW BENZIMIDAZOLE DERIVATIVES |
DE19517840A1 (de) * | 1995-05-16 | 1996-11-21 | Bayer Ag | Wirkstoffkombinationen |
DE19708688A1 (de) * | 1997-03-04 | 1998-09-10 | Bayer Ag | Annellierte Azolderivate |
US6495583B1 (en) | 1997-03-25 | 2002-12-17 | Synaptic Pharmaceutical Corporation | Benzimidazole derivatives |
KR101647856B1 (ko) * | 2008-07-18 | 2016-08-11 | 다우 글로벌 테크놀로지스 엘엘씨 | 살생물 조성물 |
EA202092643A1 (ru) | 2018-05-15 | 2021-03-22 | Байер Акциенгезельшафт | 2-бром-6-алкоксифенилзамещенные пирролин-2-оны и их применение в качестве гербицидов |
WO2019219584A1 (de) | 2018-05-15 | 2019-11-21 | Bayer Aktiengesellschaft | Neue spirocyclohexylpyrrolin-2-one und deren verwendung als herbizide |
WO2019219585A1 (de) | 2018-05-15 | 2019-11-21 | Bayer Aktiengesellschaft | Neue 3-(4-alkinyl-6-alkoxy-2-chlorphenyl)-3-pyrrolin-2-one und deren verwendung als herbizide |
WO2019228787A1 (de) | 2018-05-29 | 2019-12-05 | Bayer Aktiengesellschaft | Speziell substituierte 2-alkyl-6-alkoxyphenyl-3-pyrrolin-2-one und deren verwendung als herbizide |
WO2019228788A1 (de) | 2018-05-29 | 2019-12-05 | Bayer Aktiengesellschaft | 2-brom-6-alkoxyphenyl-substituierte pyrrolin-2-one und deren verwendung als herbizide |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU4948093A (en) * | 1992-08-25 | 1994-03-15 | Ciba-Geigy Ag | Benzimidazole derivatives as microbicides |
DE4237557A1 (de) * | 1992-11-06 | 1994-05-11 | Bayer Ag | Substituierte Benzimidazole |
DE4237567A1 (de) * | 1992-11-06 | 1994-05-11 | Bayer Ag | Schädlingsbekämpfungsmittel |
-
1995
- 1995-04-13 DE DE19513990A patent/DE19513990A1/de not_active Withdrawn
-
1996
- 1996-04-01 WO PCT/EP1996/001435 patent/WO1996032395A1/de active IP Right Grant
- 1996-04-01 CZ CZ973245A patent/CZ324597A3/cs unknown
- 1996-04-01 BR BR9604831A patent/BR9604831A/pt unknown
- 1996-04-01 AU AU52765/96A patent/AU5276596A/en not_active Abandoned
- 1996-04-01 PL PL96322721A patent/PL185393B1/pl unknown
- 1996-04-01 HU HU9801565A patent/HUP9801565A3/hu unknown
- 1996-04-01 JP JP8530687A patent/JPH11503725A/ja not_active Ceased
- 1996-04-01 EP EP96909163A patent/EP0820457A1/de not_active Withdrawn
- 1996-04-01 RU RU97118853/04A patent/RU2159242C2/ru active
- 1996-04-01 SK SK1371-97A patent/SK137197A3/sk unknown
- 1996-04-01 US US08/930,767 patent/US5925663A/en not_active Expired - Fee Related
- 1996-04-01 KR KR1019970707200A patent/KR19980703800A/ko active IP Right Grant
-
1999
- 1999-01-11 US US09/227,809 patent/US6080776A/en not_active Expired - Fee Related
-
2000
- 2000-01-24 US US09/490,482 patent/US6235765B1/en not_active Expired - Fee Related
-
2001
- 2001-01-22 US US09/767,194 patent/US20020026059A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
PL185393B1 (pl) | 2003-05-30 |
US5925663A (en) | 1999-07-20 |
CZ324597A3 (cs) | 1998-01-14 |
WO1996032395A1 (de) | 1996-10-17 |
US6080776A (en) | 2000-06-27 |
EP0820457A1 (de) | 1998-01-28 |
US20020026059A1 (en) | 2002-02-28 |
SK137197A3 (en) | 1998-05-06 |
HUP9801565A3 (en) | 2001-11-28 |
US6235765B1 (en) | 2001-05-22 |
BR9604831A (pt) | 1999-01-05 |
DE19513990A1 (de) | 1996-10-17 |
RU2159242C2 (ru) | 2000-11-20 |
JPH11503725A (ja) | 1999-03-30 |
AU5276596A (en) | 1996-10-30 |
PL322721A1 (en) | 1998-02-16 |
KR19980703800A (ko) | 1998-12-05 |
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