HUP9600624A2 - Fused imidazole derivatives, process for producing them and pharmaceutical compositions containing them - Google Patents
Fused imidazole derivatives, process for producing them and pharmaceutical compositions containing themInfo
- Publication number
- HUP9600624A2 HUP9600624A2 HU9600624A HUP9600624A HUP9600624A2 HU P9600624 A2 HUP9600624 A2 HU P9600624A2 HU 9600624 A HU9600624 A HU 9600624A HU P9600624 A HUP9600624 A HU P9600624A HU P9600624 A2 HUP9600624 A2 HU P9600624A2
- Authority
- HU
- Hungary
- Prior art keywords
- producing
- pharmaceutical compositions
- compositions containing
- imidazole derivatives
- fused imidazole
- Prior art date
Links
- 150000002460 imidazoles Chemical class 0.000 title 1
- 229940079865 intestinal antiinfectives imidazole derivative Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9502863A FR2731708B1 (fr) | 1995-03-13 | 1995-03-13 | Derives de piperidine, leur procede de preparation et leur application en therapeutique |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HU9600624D0 HU9600624D0 (en) | 1996-05-28 |
| HUP9600624A2 true HUP9600624A2 (en) | 1997-01-28 |
Family
ID=9476960
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU9600624A HUP9600624A2 (en) | 1995-03-13 | 1996-03-12 | Fused imidazole derivatives, process for producing them and pharmaceutical compositions containing them |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP0732334A1 (hu) |
| JP (1) | JPH08269058A (hu) |
| KR (1) | KR960034205A (hu) |
| CN (1) | CN1140174A (hu) |
| AU (1) | AU4800896A (hu) |
| CA (1) | CA2171579A1 (hu) |
| CZ (1) | CZ75496A3 (hu) |
| FR (1) | FR2731708B1 (hu) |
| HU (1) | HUP9600624A2 (hu) |
| IL (1) | IL117455A0 (hu) |
| NO (1) | NO961000L (hu) |
| NZ (1) | NZ286164A (hu) |
| PL (1) | PL313204A1 (hu) |
| SK (1) | SK34196A3 (hu) |
| ZA (1) | ZA961994B (hu) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP9900606A2 (hu) * | 1995-09-18 | 2000-03-28 | Glaxo Group Limited | 5-HT3 Receptor antagonisták mozgászavar kezelésére |
| TW527186B (en) | 1996-03-19 | 2003-04-11 | Janssen Pharmaceutica Nv | Fused imidazole derivatives as multidrug resistance modulators |
| FR2801589A1 (fr) * | 1999-11-25 | 2001-06-01 | Sanofi Synthelabo | Derives de 2-arylquinoleine, leur preparation et leur application en therapeutique |
| FR2816619B1 (fr) * | 2000-11-15 | 2003-01-31 | Sanofi Synthelabo | Derives de benzimidazole, leur preparation et leur application en therapeutique |
| AR030121A1 (es) | 2000-08-08 | 2003-08-13 | Sanofi Aventis | Derivados de benzimidazol, su preparacion y su aplicacion en terapeutica |
| FR2816942B1 (fr) | 2000-11-23 | 2003-05-09 | Sanofi Synthelabo | Derives de benzimidazole, leur preparation et leur application en therapeutique |
| FR2816941B1 (fr) * | 2000-11-23 | 2003-01-31 | Sanofi Synthelabo | Derives de benzimidazole, leur preparation et leur application en therapeutique |
| EP2970282B1 (en) * | 2013-03-15 | 2019-08-21 | Incyte Holdings Corporation | Tricyclic heterocycles as bet protein inhibitors |
| ES2635560T3 (es) | 2013-07-08 | 2017-10-04 | Incyte Holdings Corporation | Heterociclos tricíclicos como inhibidores de la proteína NET |
| WO2015081189A1 (en) | 2013-11-26 | 2015-06-04 | Incyte Corporation | Bicyclic heterocycles as bet protein inhibitors |
| US9399640B2 (en) | 2013-11-26 | 2016-07-26 | Incyte Corporation | Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors |
| WO2015095492A1 (en) | 2013-12-19 | 2015-06-25 | Incyte Corporation | Tricyclic heterocycles as bet protein inhibitors |
| CN106414442B (zh) | 2014-04-23 | 2019-03-15 | 因赛特公司 | 作为BET蛋白抑制剂的1H-吡咯并[2,3-c]吡啶-7(6H)-酮和吡唑并[3,4-c]吡啶-7(6H)-酮 |
| TWI712603B (zh) | 2014-09-15 | 2020-12-11 | 美商英塞特公司 | 作為ｂｅｔ蛋白抑制劑之三環雜環 |
| AR106520A1 (es) | 2015-10-29 | 2018-01-24 | Incyte Corp | Forma sólida amorfa de un inhibidor de proteína bet |
| PE20190623A1 (es) | 2016-06-20 | 2019-04-26 | Incyte Corp | Formas solidas cristalinas de un inhibidor de bet |
| KR20210025016A (ko) * | 2018-06-28 | 2021-03-08 | 지앙수 헨그루이 메디슨 컴퍼니 리미티드 | 접합 삼중고리형 헤테로사이클 화합물과 그 치료 용도 |
| US11833155B2 (en) | 2020-06-03 | 2023-12-05 | Incyte Corporation | Combination therapy for treatment of myeloproliferative neoplasms |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2674855B1 (fr) * | 1991-04-03 | 1994-01-14 | Synthelabo | Derives de piperidine, leur preparation et leur application en therapeutique. |
| FR2696176B1 (fr) * | 1992-09-28 | 1994-11-10 | Synthelabo | Dérivés de pipéridine, leur préparation et leur application en thérapeutique. |
| FR2710915B1 (fr) * | 1993-10-04 | 1995-11-24 | Synthelabo | Dérivés de pipéridine, leur préparation et leur utilisation en thérapeutique. |
-
1995
- 1995-03-13 FR FR9502863A patent/FR2731708B1/fr not_active Expired - Fee Related
-
1996
- 1996-03-04 EP EP96400452A patent/EP0732334A1/fr not_active Withdrawn
- 1996-03-12 CN CN96107315A patent/CN1140174A/zh active Pending
- 1996-03-12 AU AU48008/96A patent/AU4800896A/en not_active Abandoned
- 1996-03-12 PL PL96313204A patent/PL313204A1/xx unknown
- 1996-03-12 JP JP8054560A patent/JPH08269058A/ja active Pending
- 1996-03-12 NZ NZ286164A patent/NZ286164A/en unknown
- 1996-03-12 CA CA002171579A patent/CA2171579A1/en not_active Abandoned
- 1996-03-12 IL IL11745596A patent/IL117455A0/xx unknown
- 1996-03-12 NO NO961000A patent/NO961000L/no unknown
- 1996-03-12 CZ CZ96754A patent/CZ75496A3/cs unknown
- 1996-03-12 ZA ZA961994A patent/ZA961994B/xx unknown
- 1996-03-12 KR KR1019960006462A patent/KR960034205A/ko not_active Application Discontinuation
- 1996-03-12 SK SK341-96A patent/SK34196A3/sk unknown
- 1996-03-12 HU HU9600624A patent/HUP9600624A2/hu unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FR2731708B1 (fr) | 1997-04-30 |
| CN1140174A (zh) | 1997-01-15 |
| JPH08269058A (ja) | 1996-10-15 |
| PL313204A1 (en) | 1996-09-16 |
| AU4800896A (en) | 1996-09-26 |
| SK34196A3 (en) | 1996-10-02 |
| IL117455A0 (en) | 1996-07-23 |
| NO961000D0 (no) | 1996-03-12 |
| NO961000L (no) | 1996-09-16 |
| CZ75496A3 (en) | 1996-10-16 |
| CA2171579A1 (en) | 1996-09-14 |
| NZ286164A (en) | 1996-11-26 |
| KR960034205A (ko) | 1996-10-22 |
| HU9600624D0 (en) | 1996-05-28 |
| EP0732334A1 (fr) | 1996-09-18 |
| FR2731708A1 (fr) | 1996-09-20 |
| ZA961994B (en) | 1996-09-03 |
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