ZA961994B - Piperidine derivatives process for the preparation thereof and application thereof in therapeutics - Google Patents
Piperidine derivatives process for the preparation thereof and application thereof in therapeuticsInfo
- Publication number
- ZA961994B ZA961994B ZA961994A ZA961994A ZA961994B ZA 961994 B ZA961994 B ZA 961994B ZA 961994 A ZA961994 A ZA 961994A ZA 961994 A ZA961994 A ZA 961994A ZA 961994 B ZA961994 B ZA 961994B
- Authority
- ZA
- South Africa
- Prior art keywords
- therapeutics
- preparation
- application
- piperidine derivatives
- derivatives process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9502863A FR2731708B1 (en) | 1995-03-13 | 1995-03-13 | PIPERIDINE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA961994B true ZA961994B (en) | 1996-09-03 |
Family
ID=9476960
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA961994A ZA961994B (en) | 1995-03-13 | 1996-03-12 | Piperidine derivatives process for the preparation thereof and application thereof in therapeutics |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP0732334A1 (en) |
| JP (1) | JPH08269058A (en) |
| KR (1) | KR960034205A (en) |
| CN (1) | CN1140174A (en) |
| AU (1) | AU4800896A (en) |
| CA (1) | CA2171579A1 (en) |
| CZ (1) | CZ75496A3 (en) |
| FR (1) | FR2731708B1 (en) |
| HU (1) | HUP9600624A2 (en) |
| IL (1) | IL117455A0 (en) |
| NO (1) | NO961000L (en) |
| NZ (1) | NZ286164A (en) |
| PL (1) | PL313204A1 (en) |
| SK (1) | SK34196A3 (en) |
| ZA (1) | ZA961994B (en) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1997010823A1 (en) * | 1995-09-18 | 1997-03-27 | Glaxo Group Limited | 5-ht3 receptor antagonists for dyskinesia |
| TW527186B (en) | 1996-03-19 | 2003-04-11 | Janssen Pharmaceutica Nv | Fused imidazole derivatives as multidrug resistance modulators |
| FR2801589A1 (en) * | 1999-11-25 | 2001-06-01 | Sanofi Synthelabo | 2-Aryl quinoline derivatives useful for the treatment of urinary incontinence. venous ulcers, migraine or gastro-intestinal disorders |
| FR2816619B1 (en) * | 2000-11-15 | 2003-01-31 | Sanofi Synthelabo | BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| AU2001282267A1 (en) * | 2000-08-08 | 2002-02-18 | Sanofi-Aventis | Benzimidazole derivatives, preparation and therapeutic use thereof |
| FR2816941B1 (en) * | 2000-11-23 | 2003-01-31 | Sanofi Synthelabo | BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| FR2816942B1 (en) | 2000-11-23 | 2003-05-09 | Sanofi Synthelabo | BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| SG10201707487VA (en) * | 2013-03-15 | 2017-10-30 | Incyte Corp | Tricyclic heterocycles as bet protein inhibitors |
| WO2015006193A1 (en) | 2013-07-08 | 2015-01-15 | Incyte Corporation | Tricyclic heterocycles as bet protein inhibitors |
| WO2015081203A1 (en) | 2013-11-26 | 2015-06-04 | Incyte Corporation | Bicyclic heterocycles as bet protein inhibitors |
| US9315501B2 (en) | 2013-11-26 | 2016-04-19 | Incyte Corporation | Bicyclic heterocycles as BET protein inhibitors |
| WO2015095492A1 (en) | 2013-12-19 | 2015-06-25 | Incyte Corporation | Tricyclic heterocycles as bet protein inhibitors |
| SG11201608843TA (en) | 2014-04-23 | 2016-11-29 | Incyte Corp | 1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS |
| WO2016044130A1 (en) * | 2014-09-15 | 2016-03-24 | Incyte Corporation | Tricyclic heterocycles for use as bet protein inhibitors |
| US20170121347A1 (en) | 2015-10-29 | 2017-05-04 | Incyte Corporation | Amorphous solid form of a bet protein inhibitor |
| IL263824B2 (en) | 2016-06-20 | 2023-10-01 | Incyte Corp | Crystalline solid forms of a bet inhibitor |
| KR20210025016A (en) * | 2018-06-28 | 2021-03-08 | 지앙수 헨그루이 메디슨 컴퍼니 리미티드 | Conjugated tricyclic heterocycle compound and its therapeutic use |
| US11833155B2 (en) | 2020-06-03 | 2023-12-05 | Incyte Corporation | Combination therapy for treatment of myeloproliferative neoplasms |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2674855B1 (en) * | 1991-04-03 | 1994-01-14 | Synthelabo | PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION. |
| FR2696176B1 (en) * | 1992-09-28 | 1994-11-10 | Synthelabo | Piperidine derivatives, their preparation and their therapeutic application. |
| FR2710915B1 (en) * | 1993-10-04 | 1995-11-24 | Synthelabo | Piperidine derivatives, their preparation and their therapeutic use. |
-
1995
- 1995-03-13 FR FR9502863A patent/FR2731708B1/en not_active Expired - Fee Related
-
1996
- 1996-03-04 EP EP96400452A patent/EP0732334A1/en not_active Withdrawn
- 1996-03-12 KR KR1019960006462A patent/KR960034205A/en not_active Application Discontinuation
- 1996-03-12 HU HU9600624A patent/HUP9600624A2/en unknown
- 1996-03-12 ZA ZA961994A patent/ZA961994B/en unknown
- 1996-03-12 PL PL96313204A patent/PL313204A1/en unknown
- 1996-03-12 JP JP8054560A patent/JPH08269058A/en active Pending
- 1996-03-12 AU AU48008/96A patent/AU4800896A/en not_active Abandoned
- 1996-03-12 CA CA002171579A patent/CA2171579A1/en not_active Abandoned
- 1996-03-12 SK SK341-96A patent/SK34196A3/en unknown
- 1996-03-12 NZ NZ286164A patent/NZ286164A/en unknown
- 1996-03-12 IL IL11745596A patent/IL117455A0/en unknown
- 1996-03-12 CZ CZ96754A patent/CZ75496A3/en unknown
- 1996-03-12 NO NO961000A patent/NO961000L/en unknown
- 1996-03-12 CN CN96107315A patent/CN1140174A/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| NO961000D0 (en) | 1996-03-12 |
| AU4800896A (en) | 1996-09-26 |
| HUP9600624A2 (en) | 1997-01-28 |
| NZ286164A (en) | 1996-11-26 |
| EP0732334A1 (en) | 1996-09-18 |
| NO961000L (en) | 1996-09-16 |
| JPH08269058A (en) | 1996-10-15 |
| IL117455A0 (en) | 1996-07-23 |
| CA2171579A1 (en) | 1996-09-14 |
| HU9600624D0 (en) | 1996-05-28 |
| CZ75496A3 (en) | 1996-10-16 |
| SK34196A3 (en) | 1996-10-02 |
| PL313204A1 (en) | 1996-09-16 |
| CN1140174A (en) | 1997-01-15 |
| FR2731708A1 (en) | 1996-09-20 |
| FR2731708B1 (en) | 1997-04-30 |
| KR960034205A (en) | 1996-10-22 |
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