HUP0400725A2 - Szubsztituált 1,2,4-tiazol-3(2H,4H)-tion-származékok, eljárás előállításukra és az ezeket tartalmazó gyógyászati készítmények - Google Patents

Szubsztituált 1,2,4-tiazol-3(2H,4H)-tion-származékok, eljárás előállításukra és az ezeket tartalmazó gyógyászati készítmények

Info

Publication number
HUP0400725A2
HUP0400725A2 HU0400725A HUP0400725A HUP0400725A2 HU P0400725 A2 HUP0400725 A2 HU P0400725A2 HU 0400725 A HU0400725 A HU 0400725A HU P0400725 A HUP0400725 A HU P0400725A HU P0400725 A2 HUP0400725 A2 HU P0400725A2
Authority
HU
Hungary
Prior art keywords
substituted
triazole
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
HU0400725A
Other languages
English (en)
Inventor
Rita Katoch
Ashok Rattan
Mohammed Salman
Jitendra Sattigeri
Ashwani Kumar Verma
Original Assignee
Ranbaxy Laboratories Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ranbaxy Laboratories Limited filed Critical Ranbaxy Laboratories Limited
Publication of HUP0400725A2 publication Critical patent/HUP0400725A2/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/12—Oxygen or sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Jelen találmány szubszutituált (I) általános képletűtriazolvegyületekre vonatkozik, amelyek gombaellenes hatásúak. Aképletben X jelentése -CH2-, -CO-, -C5-, vagy SO2-csoport; Arjelentése szubsztituált fenilcsoport, R1, R2 és R3 jelentésehidrogénatom vagy alkil-, alkoxi-, amino-, hidroxi-, nitro-, ciano-,karbonil-, védett karboxil vagy -SO2R1- csoport, Y jelentése adottesetben szubsztituált fenilcsoport, X1, X2, Y1, Y2 és Z jelentésehidrogén vagy halogénatom, nitro-, ciano-, amino-, aril-, karboxil-,védett karbonil- vagy adott esetben halogénezett alkil- vagyalkoxicsoport; n = 0 vagy 1. Ó
HU0400725A 2000-12-26 2001-12-21 Szubsztituált 1,2,4-tiazol-3(2H,4H)-tion-származékok, eljárás előállításukra és az ezeket tartalmazó gyógyászati készítmények HUP0400725A2 (hu)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1197DE2000 2000-12-26
PCT/IB2001/002620 WO2002051408A1 (en) 2000-12-26 2001-12-21 Azole compounds as anti-fungals agents

Publications (1)

Publication Number Publication Date
HUP0400725A2 true HUP0400725A2 (hu) 2004-07-28

Family

ID=11097140

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0400725A HUP0400725A2 (hu) 2000-12-26 2001-12-21 Szubsztituált 1,2,4-tiazol-3(2H,4H)-tion-származékok, eljárás előállításukra és az ezeket tartalmazó gyógyászati készítmények

Country Status (18)

Country Link
US (1) US6710049B2 (hu)
EP (1) EP1347758A1 (hu)
JP (1) JP2004518667A (hu)
CN (1) CN1489465A (hu)
AR (1) AR035525A1 (hu)
BG (1) BG108032A (hu)
BR (1) BR0116570A (hu)
CA (1) CA2433259A1 (hu)
CZ (1) CZ20032028A3 (hu)
EA (1) EA200300725A1 (hu)
EC (1) ECSP034673A (hu)
HU (1) HUP0400725A2 (hu)
MA (1) MA26066A1 (hu)
MX (1) MXPA03005899A (hu)
PL (1) PL362051A1 (hu)
SK (1) SK9522003A3 (hu)
WO (1) WO2002051408A1 (hu)
ZA (1) ZA200304980B (hu)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN191819B (hu) * 2001-07-19 2004-01-03 Ranbaxy Lab Ltd
WO2004018485A1 (en) * 2002-08-26 2004-03-04 Ranbaxy Laboratories Limited Azole derivatives as antifungal agents
WO2007047394A2 (en) * 2005-10-13 2007-04-26 Epix Delaware, Inc. Thiotriazolyl derivatives
TWI518075B (zh) * 2010-10-01 2016-01-21 大正製藥股份有限公司 1,2,4-triazolone derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB567981A (en) 1943-03-30 1945-03-13 Malcolm Edward Johnson Improvements in or relating to control valves for vehicle servo brakes
TW218017B (hu) * 1992-04-28 1993-12-21 Takeda Pharm Industry Co Ltd
CA2134417A1 (en) * 1993-12-22 1995-06-23 Katsumi Itoh Optically active azole derivatives, their production and use
CA2150533A1 (en) 1994-05-31 1995-12-01 Katsumi Itoh Production of optically active triazole compounds and their intermediates
TW318841B (hu) 1995-02-17 1997-11-01 Takeda Pharm Industry Co Ltd
DE19620407A1 (de) * 1996-05-21 1997-11-27 Bayer Ag Thiocyano-triazolyl-Derivate
AU3402301A (en) 2000-03-07 2001-09-17 Ranbaxy Laboratories Limited Azole compounds as therapeutic agents for fungal infections

Also Published As

Publication number Publication date
JP2004518667A (ja) 2004-06-24
PL362051A1 (en) 2004-10-18
CZ20032028A3 (cs) 2003-11-12
CN1489465A (zh) 2004-04-14
EA200300725A1 (ru) 2004-04-29
BR0116570A (pt) 2005-04-12
ZA200304980B (en) 2004-04-28
US6710049B2 (en) 2004-03-23
WO2002051408A1 (en) 2002-07-04
EP1347758A1 (en) 2003-10-01
US20020119984A1 (en) 2002-08-29
AR035525A1 (es) 2004-06-02
CA2433259A1 (en) 2002-07-04
MA26066A1 (fr) 2004-04-01
SK9522003A3 (en) 2003-12-02
BG108032A (bg) 2004-12-30
ECSP034673A (es) 2003-08-29
MXPA03005899A (es) 2004-01-26

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