HUP0103877A2 - Arilcsoporttal szubsztituált propanolaminszármazékok, eljárás előállításukra, ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk - Google Patents

Arilcsoporttal szubsztituált propanolaminszármazékok, eljárás előállításukra, ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk

Info

Publication number
HUP0103877A2
HUP0103877A2 HU0103877A HUP0103877A HUP0103877A2 HU P0103877 A2 HUP0103877 A2 HU P0103877A2 HU 0103877 A HU0103877 A HU 0103877A HU P0103877 A HUP0103877 A HU P0103877A HU P0103877 A2 HUP0103877 A2 HU P0103877A2
Authority
HU
Hungary
Prior art keywords
aryl
compounds
production
methods
medicaments containing
Prior art date
Application number
HU0103877A
Other languages
English (en)
Inventor
Wendelin Frick
Heiner Glombik
Reinhard Kirsch
Werner Kramer
Hans-Ludwig Schäfer
Original Assignee
Aventis Pharma Deutschland Gmbh.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Deutschland Gmbh. filed Critical Aventis Pharma Deutschland Gmbh.
Publication of HUP0103877A2 publication Critical patent/HUP0103877A2/hu
Publication of HUP0103877A3 publication Critical patent/HUP0103877A3/hu
Publication of HU228987B1 publication Critical patent/HU228987B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18—Acyclic radicals, substituted by carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Genetics & Genomics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Peptides Or Proteins (AREA)
  • Pyridine Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HU0103877A 1998-10-02 1999-09-18 Arilcsoporttal szubsztituált propanolamin-származékok, eljárás elõállításukra, ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk HU228987B1 (hu)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19845405A DE19845405C2 (de) 1998-10-02 1998-10-02 Arylsubstituierte Propanolaminderivate und deren Verwendung
PCT/EP1999/006931 WO2000020392A1 (de) 1998-10-02 1999-09-18 Arylsubstituierte propanolaminderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung

Publications (3)

Publication Number Publication Date
HUP0103877A2 true HUP0103877A2 (hu) 2002-02-28
HUP0103877A3 HUP0103877A3 (en) 2002-10-28
HU228987B1 HU228987B1 (hu) 2013-07-29

Family

ID=7883186

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0103877A HU228987B1 (hu) 1998-10-02 1999-09-18 Arilcsoporttal szubsztituált propanolamin-származékok, eljárás elõállításukra, ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk

Country Status (23)

Country Link
US (4) US6245744B1 (hu)
EP (1) EP1117645B1 (hu)
JP (1) JP3794618B2 (hu)
KR (1) KR100600425B1 (hu)
CN (1) CN1135223C (hu)
AR (1) AR021844A1 (hu)
AT (1) ATE266005T1 (hu)
AU (1) AU757871B2 (hu)
BR (1) BR9915967A (hu)
CA (1) CA2345369C (hu)
CZ (1) CZ299828B6 (hu)
DE (2) DE19845405C2 (hu)
DK (1) DK1117645T3 (hu)
ES (1) ES2219110T3 (hu)
HK (1) HK1040708B (hu)
HU (1) HU228987B1 (hu)
ID (1) ID27762A (hu)
PL (1) PL347107A1 (hu)
PT (1) PT1117645E (hu)
RU (1) RU2226532C2 (hu)
TR (1) TR200100894T2 (hu)
WO (1) WO2000020392A1 (hu)
ZA (1) ZA200102588B (hu)

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DE19845405C2 (de) 2000-07-13
AR021844A1 (es) 2002-08-07
US6245744B1 (en) 2001-06-12
ID27762A (id) 2001-04-26
HU228987B1 (hu) 2013-07-29
HUP0103877A3 (en) 2002-10-28
CN1321148A (zh) 2001-11-07
EP1117645B1 (de) 2004-05-06
DE59909418D1 (de) 2004-06-09
CA2345369C (en) 2009-12-29
JP2002526529A (ja) 2002-08-20
TR200100894T2 (tr) 2001-10-22
ES2219110T3 (es) 2004-11-16
US20030195145A1 (en) 2003-10-16
KR100600425B1 (ko) 2006-07-13
CZ299828B6 (cs) 2008-12-10
HK1040708A1 (en) 2002-06-21
US6566340B2 (en) 2003-05-20
PT1117645E (pt) 2004-09-30
RU2226532C2 (ru) 2004-04-10
WO2000020392A1 (de) 2000-04-13
ATE266005T1 (de) 2004-05-15
AU757871B2 (en) 2003-03-06
EP1117645A1 (de) 2001-07-25
BR9915967A (pt) 2001-08-28
JP3794618B2 (ja) 2006-07-05
US20020042381A1 (en) 2002-04-11
KR20010103592A (ko) 2001-11-23
ZA200102588B (en) 2002-01-30
HK1040708B (zh) 2004-06-18
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DE19845405A1 (de) 2000-04-20
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