HUP0103749A2 - Triciklusos delta3-piperidinek mint gyógyszerkészítmények hatóanyagai és eljárás az előállításukra - Google Patents
Triciklusos delta3-piperidinek mint gyógyszerkészítmények hatóanyagai és eljárás az előállításukraInfo
- Publication number
- HUP0103749A2 HUP0103749A2 HU0103749A HUP0103749A HUP0103749A2 HU P0103749 A2 HUP0103749 A2 HU P0103749A2 HU 0103749 A HU0103749 A HU 0103749A HU P0103749 A HUP0103749 A HU P0103749A HU P0103749 A2 HUP0103749 A2 HU P0103749A2
- Authority
- HU
- Hungary
- Prior art keywords
- piperidines
- pharmaceuticals
- preparation
- delta3
- tricyclic
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Ophthalmology & Optometry (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Reproductive Health (AREA)
- Hospice & Palliative Care (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Psychology (AREA)
- Emergency Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP98203371 | 1998-10-06 | ||
PCT/EP1999/007420 WO2000020423A1 (en) | 1998-10-06 | 1999-10-01 | Tricyclic δ3-piperidines as pharmaceuticals |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP0103749A2 true HUP0103749A2 (hu) | 2002-02-28 |
HUP0103749A3 HUP0103749A3 (en) | 2003-03-28 |
Family
ID=8234192
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0103749A HUP0103749A3 (en) | 1998-10-06 | 1999-10-01 | Tricyclic delta3-piperidines as pharmaceuticals and process for their preparation |
Country Status (28)
Country | Link |
---|---|
US (1) | US6352999B1 (hu) |
EP (1) | EP1119570B1 (hu) |
JP (1) | JP4590102B2 (hu) |
KR (1) | KR20010071844A (hu) |
CN (1) | CN1131868C (hu) |
AR (1) | AR023679A1 (hu) |
AT (1) | ATE269337T1 (hu) |
AU (1) | AU759199B2 (hu) |
BG (1) | BG64871B1 (hu) |
BR (1) | BR9913108A (hu) |
CA (1) | CA2346082C (hu) |
CZ (1) | CZ20011105A3 (hu) |
DE (1) | DE69918148T2 (hu) |
EE (1) | EE04680B1 (hu) |
ES (1) | ES2222735T3 (hu) |
HK (1) | HK1038009A1 (hu) |
HU (1) | HUP0103749A3 (hu) |
ID (1) | ID28451A (hu) |
IL (2) | IL142444A0 (hu) |
NO (1) | NO20011402D0 (hu) |
NZ (1) | NZ510116A (hu) |
PL (1) | PL347179A1 (hu) |
RU (1) | RU2226194C2 (hu) |
SK (1) | SK285386B6 (hu) |
TR (1) | TR200100953T2 (hu) |
TW (1) | TWI244485B (hu) |
UA (1) | UA70961C2 (hu) |
WO (1) | WO2000020423A1 (hu) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA69420C2 (uk) * | 1998-10-06 | 2004-09-15 | Янссен Фармацевтика Н.В. | ТРИЦИКЛІЧНІ <font face="Symbol">D3</font>-ПІПЕРИДИНИ ЯК <font face="Symbol">a<sub></font>2</sub>-АНТАГОНІСТИ |
EP1404679A2 (en) * | 2001-07-05 | 2004-04-07 | PHARMACIA & UPJOHN COMPANY | (hetero)aryl substituted benzofurans as 5-ht ligands |
WO2003082825A1 (en) * | 2002-04-03 | 2003-10-09 | Orion Corporation | Use of an alfa2-adrenoreceptor antagonist for cns-related diseases |
WO2005100355A1 (ja) | 2004-04-12 | 2005-10-27 | Taisho Pharmaceutical Co., Ltd. | 環状アミン化合物 |
CN101120002A (zh) | 2005-02-17 | 2008-02-06 | 惠氏公司 | 环烷基稠合的吲哚、苯并噻吩、苯并呋喃和茚衍生物 |
DE102005038947A1 (de) * | 2005-05-18 | 2006-11-30 | Grünenthal GmbH | Substituierte Benzo[d]isoxazol-3-yl-amin-Verbindungen und deren Verwendung in Arzneimitteln |
ES2897946T3 (es) | 2013-07-25 | 2022-03-03 | Dong A St Co Ltd | Método para preparar un derivado de benzamida, intermedio novedoso utilizado en la preparación de la benzamida y método para preparar un intermedio novedoso |
CN103755715B (zh) * | 2013-12-26 | 2015-12-09 | 武汉理工大学 | 苯并呋喃并[2,3-c]吡啶化合物及其合成方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3522959A1 (de) * | 1985-06-27 | 1987-01-08 | Merck Patent Gmbh | Indolderivate |
US4673680A (en) * | 1985-09-18 | 1987-06-16 | Pendleton Robert G | α2 -adrenergic receptor antagonists as modifiers of gastrointestinal motility |
US4985422A (en) * | 1988-04-27 | 1991-01-15 | Glaxo Group Limited | Lactam derivatives |
US5100891A (en) * | 1991-01-18 | 1992-03-31 | Hoechst-Roussel Pharmaceuticals Inc. | Substituted 1,2,3,4-tetrahydrocyclopent[b]indoles, 1,2,3,3a,4,8a-hexahydrocyclopent[B]indoles and related compounds |
AU735764B2 (en) * | 1996-12-06 | 2001-07-12 | Abbott Laboratories | Benzopyranopyrrole and benzopyranopyridine alpha-1 adrenergic compounds |
UA52681C2 (uk) * | 1997-04-08 | 2003-01-15 | Янссен Фармацевтика Н.В. | Похідні 1,2,3,4-тетрагідро-бензофуро[3,2,-c]піридину, спосіб їх одержання та фармацевтична композиція на їх основі |
UA69420C2 (uk) * | 1998-10-06 | 2004-09-15 | Янссен Фармацевтика Н.В. | ТРИЦИКЛІЧНІ <font face="Symbol">D3</font>-ПІПЕРИДИНИ ЯК <font face="Symbol">a<sub></font>2</sub>-АНТАГОНІСТИ |
-
1999
- 1999-10-01 DE DE69918148T patent/DE69918148T2/de not_active Expired - Lifetime
- 1999-10-01 AU AU63342/99A patent/AU759199B2/en not_active Ceased
- 1999-10-01 BR BR9913108-0A patent/BR9913108A/pt not_active Application Discontinuation
- 1999-10-01 CN CN998116688A patent/CN1131868C/zh not_active Expired - Fee Related
- 1999-10-01 AT AT99950628T patent/ATE269337T1/de not_active IP Right Cessation
- 1999-10-01 KR KR1020017000443A patent/KR20010071844A/ko active Search and Examination
- 1999-10-01 EE EEP200100210A patent/EE04680B1/xx not_active IP Right Cessation
- 1999-10-01 JP JP2000574535A patent/JP4590102B2/ja not_active Expired - Fee Related
- 1999-10-01 EP EP99950628A patent/EP1119570B1/en not_active Expired - Lifetime
- 1999-10-01 PL PL99347179A patent/PL347179A1/xx not_active Application Discontinuation
- 1999-10-01 ID IDW20010779A patent/ID28451A/id unknown
- 1999-10-01 SK SK433-2001A patent/SK285386B6/sk unknown
- 1999-10-01 TR TR2001/00953T patent/TR200100953T2/xx unknown
- 1999-10-01 IL IL14244499A patent/IL142444A0/xx active IP Right Grant
- 1999-10-01 UA UA2001032000A patent/UA70961C2/uk unknown
- 1999-10-01 HU HU0103749A patent/HUP0103749A3/hu unknown
- 1999-10-01 WO PCT/EP1999/007420 patent/WO2000020423A1/en not_active Application Discontinuation
- 1999-10-01 CZ CZ20011105A patent/CZ20011105A3/cs unknown
- 1999-10-01 NZ NZ510116A patent/NZ510116A/xx unknown
- 1999-10-01 CA CA2346082A patent/CA2346082C/en not_active Expired - Fee Related
- 1999-10-01 RU RU2001111811/04A patent/RU2226194C2/ru not_active IP Right Cessation
- 1999-10-01 ES ES99950628T patent/ES2222735T3/es not_active Expired - Lifetime
- 1999-10-01 US US09/806,587 patent/US6352999B1/en not_active Expired - Lifetime
- 1999-10-01 TW TW088116897A patent/TWI244485B/zh not_active IP Right Cessation
- 1999-10-05 AR ARP990105041A patent/AR023679A1/es active IP Right Grant
-
2001
- 2001-03-12 BG BG105334A patent/BG64871B1/bg unknown
- 2001-03-20 NO NO20011402A patent/NO20011402D0/no not_active Application Discontinuation
- 2001-04-04 IL IL142444A patent/IL142444A/en not_active IP Right Cessation
- 2001-12-10 HK HK01108630A patent/HK1038009A1/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD9A | Lapse of provisional protection due to non-payment of fees |