HUP0100619A3 - Thiazole-, isothiazole- and thiadiazole-derivatives having microbicidal and plant immunizing activities, intermediates and use thereof - Google Patents

Thiazole-, isothiazole- and thiadiazole-derivatives having microbicidal and plant immunizing activities, intermediates and use thereof

Info

Publication number
HUP0100619A3
HUP0100619A3 HU0100619A HUP0100619A HUP0100619A3 HU P0100619 A3 HUP0100619 A3 HU P0100619A3 HU 0100619 A HU0100619 A HU 0100619A HU P0100619 A HUP0100619 A HU P0100619A HU P0100619 A3 HUP0100619 A3 HU P0100619A3
Authority
HU
Hungary
Prior art keywords
microbicidal
isothiazole
thiadiazole
thiazole
intermediates
Prior art date
Application number
HU0100619A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of HUP0100619A2 publication Critical patent/HUP0100619A2/hu
Publication of HUP0100619A3 publication Critical patent/HUP0100619A3/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/781,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/30Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/061,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HU0100619A 1997-12-22 1998-12-18 Thiazole-, isothiazole- and thiadiazole-derivatives having microbicidal and plant immunizing activities, intermediates and use thereof HUP0100619A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9726989.8A GB9726989D0 (en) 1997-12-22 1997-12-22 Organic compounds
PCT/EP1998/008335 WO1999032464A1 (en) 1997-12-22 1998-12-18 Thiazole-, isothiazole- and thiadiazole-derivatives having microbicidal and plant immunizing activities

Publications (2)

Publication Number Publication Date
HUP0100619A2 HUP0100619A2 (hu) 2001-06-28
HUP0100619A3 true HUP0100619A3 (en) 2002-03-28

Family

ID=10823994

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0100619A HUP0100619A3 (en) 1997-12-22 1998-12-18 Thiazole-, isothiazole- and thiadiazole-derivatives having microbicidal and plant immunizing activities, intermediates and use thereof

Country Status (15)

Country Link
EP (1) EP1042306A1 (hu)
JP (1) JP2001526277A (hu)
CN (1) CN1282324A (hu)
AR (1) AR017438A1 (hu)
AU (1) AU2054699A (hu)
BR (1) BR9814394A (hu)
CA (1) CA2309973A1 (hu)
GB (1) GB9726989D0 (hu)
GT (1) GT199800193A (hu)
HU (1) HUP0100619A3 (hu)
IL (1) IL136589A0 (hu)
PL (1) PL341290A1 (hu)
TR (1) TR200001740T2 (hu)
WO (1) WO1999032464A1 (hu)
ZA (1) ZA9811706B (hu)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6310052B1 (en) 1996-06-04 2001-10-30 Queen's University At Kingston Nitrate esters and their use for neurological conditions
CA2408686A1 (en) * 2000-05-15 2002-11-12 Basf Aktiengesellschaft 3-arylisothiazoles and their use as herbicides
DE10029077A1 (de) * 2000-06-13 2001-12-20 Bayer Ag Thiazolylsubstituierte Heterocyclen
BR0208956A (pt) 2001-04-16 2004-07-13 Tanabe Seiyaku Co Abridor de canais de k ativados por cálcio de grande condutância
AU2002314744A1 (en) 2001-04-17 2002-10-28 Sepracor, Inc. Thiazole and other heterocyclic ligands and use thereof
GB0712653D0 (en) 2007-06-28 2007-08-08 Syngenta Ltd Novel herbicides
GB0717082D0 (en) 2007-09-03 2007-10-10 Syngenta Ltd Novel herbicides
MX2012006349A (es) * 2009-12-07 2012-10-03 Cardioxyl Pharmaceuticals Inc Derivados de n-aciloxisulfonamida y n-hidroxi-n-acilsulfonamida.
US9018411B2 (en) 2009-12-07 2015-04-28 Cardioxyl Pharmaceuticals, Inc. Bis-acylated hydroxylamine derivatives
BR112012030208A2 (pt) * 2010-05-27 2015-09-29 Bayer Intelectual Property Gmbh derivados de alcanol heterocíclicos como fungicidas
JP5872548B2 (ja) * 2010-05-27 2016-03-01 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 殺菌剤としてのヘテロ環式アルカノール誘導体
EP2576528A1 (de) * 2010-05-27 2013-04-10 Bayer CropScience AG Heterocyclische alkanolderivate als fungizide
EP2508511A1 (en) * 2011-04-07 2012-10-10 Laboratoire Biodim Inhibitors of viral replication, their process of preparation and their therapeutical uses
CN102417505B (zh) * 2011-08-29 2014-07-09 南开大学 含甲基-1,2,3-噻二唑的四氮唑类化合物及其制备方法和用途
CN108752287A (zh) * 2018-05-21 2018-11-06 南开大学 一类杂环叔醇衍生物的制备方法和用途
CN108912108B (zh) * 2018-06-27 2021-09-03 中国科学院上海有机化学研究所 三氟甲基化合物及其制备方法及其在农药中的应用
CN113214241A (zh) * 2021-04-29 2021-08-06 华东理工大学 一种用于检测十字花科蔬菜核盘菌的化合物及其应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1953861C2 (de) * 1969-10-25 1982-12-23 Fujisawa Pharmaceutical Co., Ltd., Osaka 7-Tetrazolylacetamido-3-thiomethyl-3-cephem-4- carbonsäuren
BE793037A (fr) * 1971-12-23 1973-06-20 Fujisawa Pharmaceutical Co Procede de preparation de derives d'acide 7-acylamino-3-substitue-3-cephem-4-carboxylique et nouveaux produits ainsi obtenus
EP0213079A3 (de) * 1985-08-23 1987-08-05 Ciba-Geigy Ag Thienylalkylester von alpha-Imidazolinon-nicotin- und -benzoesäuren
US5135927A (en) * 1987-01-30 1992-08-04 Ciba-Geigy Corporation Microbicidal composition
CA2014880A1 (en) * 1989-04-27 1990-10-27 Indu Sawhney Thiazole derivatives
JP3726306B2 (ja) * 1994-04-27 2005-12-14 日産化学工業株式会社 ピラゾールカルボン酸誘導体および植物病害防除剤
WO1996017840A1 (en) * 1994-12-06 1996-06-13 Agrevo Uk Limited Heterocyclyl substituted hydroxyacetamide derivatives as fongicides
MY113237A (en) * 1995-03-31 2001-12-31 Nihon Nohyaku Co Ltd An agricultural and horticultural disease controller and a method for controlling the diseases
DE19545638A1 (de) * 1995-12-07 1997-06-12 Bayer Ag Verwendung von 1,2,3-Thiadiazolcarbonsäure(thio)estern zur Bekämpfung von Schädlingen
CN1072657C (zh) * 1996-09-30 2001-10-10 日本农药株式会社 1,2,3-噻二唑衍生物和其盐以及农业园艺病毒防治剂及其使用方法

Also Published As

Publication number Publication date
GT199800193A (es) 2000-05-25
PL341290A1 (en) 2001-04-09
WO1999032464A1 (en) 1999-07-01
AR017438A1 (es) 2001-09-05
CN1282324A (zh) 2001-01-31
IL136589A0 (en) 2001-06-14
ZA9811706B (en) 1999-06-22
CA2309973A1 (en) 1999-07-01
HUP0100619A2 (hu) 2001-06-28
EP1042306A1 (en) 2000-10-11
TR200001740T2 (tr) 2000-11-21
BR9814394A (pt) 2000-10-10
GB9726989D0 (en) 1998-02-18
JP2001526277A (ja) 2001-12-18
AU2054699A (en) 1999-07-12

Similar Documents

Publication Publication Date Title
HUP0203624A3 (en) Pyrazolecarboxamide and pyrazolethioamide as fungicide, intermediates, preparation and use thereof
HUP0105098A3 (en) Fungicidal n2-phenylamidine derivatives, intermediates and use thereof
HUP0104171A3 (en) Pyrimidinylbenzimidazole and triatinylbenzimidazole derivatives, intermediates and use as agricultura/horticultural fungicides
IL129707A0 (en) Herbicide resistant plants
ZA9711121B (en) Reduction of hair growth.
HUP0004463A3 (en) Fluoropyrazole-biphenylamide fungicides, preparation and use thereof
PL334135A1 (en) Transgenous plants
HUP0100619A3 (en) Thiazole-, isothiazole- and thiadiazole-derivatives having microbicidal and plant immunizing activities, intermediates and use thereof
ZA976348B (en) Reduction of hair growth.
HUP0103859A3 (en) Fungicidal and insecticidal pyrimidin-4-enamines, intermediates, preparation and use thereof
ZA9711328B (en) Reduction of hair growth.
ZA978725B (en) Herbicidal and plant growth regulant compositions and the use thereof
HUP0102663A3 (en) Herbicidal 2,4-diamino-1,3,5-triazines, intermediates, preparation and use thereof
ZA95269B (en) Quinazoline-2,4-diones
GB2321852B (en) Hair growing agent
HUP0001009A3 (en) Herbicidal 3-carbamoyl/3-thiocarbamoyl-substituted 2-benzoyl-cyclohexan-1,3-diones, intermediates, preparation and use thereof
HUP0101041A3 (en) Fungicidal n-sulphonyl and n-sulphinyl phenylglycinamide, intermediates, preparation and use thereof
ZA969645B (en) Novel intermediates and their use to prepare N,N'-bridged bisindolylmaleimides.
ZA987533B (en) Irrigation sprinkler.
HUP0000491A3 (en) Herbicidal substituted 4-benzoyl-pyrazole derivatives, preparation and use thereof
ZA973549B (en) Substituted aminomethylphenylsulfonylureas, their preparation, and their use as herbicides and plant growth regulators.
NZ330551A (en) 2-aryloxy-6-aryl-3,5-difluoropyridines, their use as herbicides and their preparation thereof
GR3036217T3 (en) Arylheterocycles with herbicidal activity
HUP0002897A3 (en) Herbicidal substituted 2-benzoyl-cyclohexane-1,3-diones, preparation and use thereof
HUP0003622A3 (en) Fungicidal pyrimidin-2-oxy-4-one and pyrimidin-2-oxy-4-thione derivatives, their preparation, intermediates and use