HUP0001461A3 - N-oxides of heterocyclicesters, amides, thioesters, and ketones - Google Patents

N-oxides of heterocyclicesters, amides, thioesters, and ketones

Info

Publication number
HUP0001461A3
HUP0001461A3 HU0001461A HUP0001461A HUP0001461A3 HU P0001461 A3 HUP0001461 A3 HU P0001461A3 HU 0001461 A HU0001461 A HU 0001461A HU P0001461 A HUP0001461 A HU P0001461A HU P0001461 A3 HUP0001461 A3 HU P0001461A3
Authority
HU
Hungary
Prior art keywords
heterocyclicesters
thioesters
ketones
amides
oxides
Prior art date
Application number
HU0001461A
Other languages
English (en)
Original Assignee
Guilford Pharmaceuticals Inc B
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Guilford Pharmaceuticals Inc B filed Critical Guilford Pharmaceuticals Inc B
Publication of HUP0001461A2 publication Critical patent/HUP0001461A2/hu
Publication of HUP0001461A3 publication Critical patent/HUP0001461A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HU0001461A 1997-02-28 1998-02-26 N-oxides of heterocyclicesters, amides, thioesters, and ketones HUP0001461A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/807,406 US5846979A (en) 1997-02-28 1997-02-28 N-oxides of heterocyclic esters, amides, thioesters, and ketones
PCT/US1998/003484 WO1998037885A1 (en) 1997-02-28 1998-02-26 N-oxides of heterocyclic esters, amides, thioesters, and ketones

Publications (2)

Publication Number Publication Date
HUP0001461A2 HUP0001461A2 (hu) 2001-04-28
HUP0001461A3 true HUP0001461A3 (en) 2002-04-29

Family

ID=25196300

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0001461A HUP0001461A3 (en) 1997-02-28 1998-02-26 N-oxides of heterocyclicesters, amides, thioesters, and ketones

Country Status (16)

Country Link
US (4) US5846979A (hu)
EP (1) EP0993299A4 (hu)
JP (1) JPH10310581A (hu)
KR (1) KR20000075502A (hu)
CN (1) CN1249681A (hu)
AR (1) AR011882A1 (hu)
AU (1) AU723374B2 (hu)
CA (1) CA2229707A1 (hu)
GT (1) GT199800041A (hu)
HU (1) HUP0001461A3 (hu)
IL (1) IL131251A0 (hu)
PA (1) PA8448001A1 (hu)
PE (1) PE59599A1 (hu)
TW (1) TW458976B (hu)
WO (1) WO1998037885A1 (hu)
ZA (1) ZA981474B (hu)

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US20010049381A1 (en) * 1997-06-04 2001-12-06 Gpl Nil Holdings, Inc., Pyrrolidine derivative hair growth compositions and uses
US6331537B1 (en) 1998-06-03 2001-12-18 Gpi Nil Holdings, Inc. Carboxylic acids and carboxylic acid isosteres of N-heterocyclic compounds
KR20010052503A (ko) 1998-06-03 2001-06-25 다니엘 피. 맥컬럼 Ｎ-헤테로사이클릭 카복실산 또는 카복실산 등입체의ｎ-결합된 설폰아미드
PL194262B1 (pl) * 1998-06-03 2007-05-31 Amgen Inc Kwasy karboksylowe i izostery kwasów karboksylowych związków N-heterocyklicznych
US6429215B1 (en) 1998-06-03 2002-08-06 Gpi Nil Holdings, Inc. N-oxide of heterocyclic ester, amide, thioester, or ketone hair growth compositions and uses
BR9912423A (pt) 1998-07-17 2001-06-05 Agouron Pharmaceticals Inc Compostos e/ou derivados farmaceuticamente aceitáveis, composições farmacêuticas, métodos de tratamento das disordens neurológicas em pacientes e processos de preparação dos compostos ou derivados farmaceuticamente aceitáveis
US7338976B1 (en) * 1998-08-14 2008-03-04 Gpi Nil Holdings, Inc. Heterocyclic esters or amides for vision and memory disorders
US6399648B1 (en) * 1998-08-14 2002-06-04 Gpi Nil Holdings, Inc. N-oxides of heterocyclic ester, amide, thioester, or ketone for vision and memory disorders
US6218423B1 (en) * 1998-08-14 2001-04-17 Gpi Nil Holdings, Inc. Pyrrolidine derivatives for vision and memory disorders
US6337340B1 (en) * 1998-08-14 2002-01-08 Gpi Nil Holdings, Inc. Carboxylic acids and isosteres of heterocyclic ring compounds having multiple heteroatoms for vision and memory disorders
WO2000009108A2 (en) * 1998-08-14 2000-02-24 Gpi Nil Holdings, Inc. Compositions and uses for vision and memory disorders
JP4708567B2 (ja) * 1998-12-03 2011-06-22 ジーピーアイ ニル ホールディングス インコーポレイテッド Ｎ−複素環化合物のカルボン酸およびカルボン酸アイソスター
CA2379149A1 (en) 1999-07-09 2001-01-18 Ortho-Mcneil Pharmaceutical, Inc. Neurotrophic pyrrolidines and piperidines, and related compositions and methods
WO2001004091A1 (en) 1999-07-09 2001-01-18 Ortho-Mcneil Pharmaceutical, Inc. Neurotrophic 2-azetidinecarboxylic acid derivatives, and related compositions and methods
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US7253169B2 (en) 1999-11-12 2007-08-07 Gliamed, Inc. Aza compounds, pharmaceutical compositions and methods of use
EP1227859B1 (en) * 1999-11-12 2006-08-09 Alcon, Inc Neurophilin ligands for treating ocular conditions
GT200000203A (es) 1999-12-01 2002-05-24 Compuestos, composiciones y metodos para estimular el crecimiento y elongacion de neuronas.
JP2003518122A (ja) 1999-12-21 2003-06-03 ジーピーアイ エヌアイエル ホールディングズ インコーポレーテッド ヒダントイン誘導体化合物、医薬合成品およびこれらの使用方法
EP1333096A1 (en) * 2000-09-01 2003-08-06 Yale University Method to identify gene function using phage display screening
JP2004532187A (ja) 2001-01-25 2004-10-21 ギルフォード ファーマシュウティカルズ インコーポレイテッド 三置換カルボサイクリックサイクロフィリン結合化合物とその用途
US6593362B2 (en) 2001-05-21 2003-07-15 Guilford Pharmaceuticals Inc. Non-peptidic cyclophilin binding compounds and their use
CA2449019A1 (en) * 2001-05-29 2002-12-05 Guilford Pharmaceuticals Inc. Method for treating nerve injury caused by surgery
DE10347573B4 (de) * 2003-10-14 2007-03-08 Koenig & Bauer Ag Druckwerk und ein Verfahren zum Bewegen eines Gestellteils
EP2309858A4 (en) 2008-07-31 2011-09-14 Dekel Pharmaceuticals Ltd COMPOSITIONS AND METHOD FOR THE TREATMENT OF INFLAMMATORY DISEASES
EP3773571A1 (en) 2018-03-28 2021-02-17 Georg-August-Universitaet Goettingen Stiftung Oeffentlichen Rechts, Universitaetsmedizin Prevention or treatment of chronic organ injury

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US6218424B1 (en) * 1996-09-25 2001-04-17 Gpi Nil Holdings, Inc. Heterocyclic ketone and thioester compounds and uses
US5786378A (en) * 1996-09-25 1998-07-28 Gpi Nil Holdings, Inc. Heterocyclic thioesters
US5721256A (en) * 1997-02-12 1998-02-24 Gpi Nil Holdings, Inc. Method of using neurotrophic sulfonamide compounds
US5846979A (en) * 1997-02-28 1998-12-08 Gpi Nil Holdings, Inc. N-oxides of heterocyclic esters, amides, thioesters, and ketones
US5945441A (en) * 1997-06-04 1999-08-31 Gpi Nil Holdings, Inc. Pyrrolidine carboxylate hair revitalizing agents

Also Published As

Publication number Publication date
EP0993299A4 (en) 2001-03-07
CA2229707A1 (en) 1998-08-28
HUP0001461A2 (hu) 2001-04-28
PA8448001A1 (es) 2000-05-24
TW458976B (en) 2001-10-11
JPH10310581A (ja) 1998-11-24
ZA981474B (en) 1998-06-08
US6054452A (en) 2000-04-25
US6251892B1 (en) 2001-06-26
EP0993299A1 (en) 2000-04-19
CN1249681A (zh) 2000-04-05
US6486151B2 (en) 2002-11-26
US5846979A (en) 1998-12-08
IL131251A0 (en) 2001-01-28
KR20000075502A (ko) 2000-12-15
US20010036942A1 (en) 2001-11-01
GT199800041A (es) 1999-08-14
AU723374B2 (en) 2000-08-24
WO1998037885A1 (en) 1998-09-03
PE59599A1 (es) 1999-06-17
AU6181598A (en) 1998-09-18
AR011882A1 (es) 2000-09-13

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