HU231525B1 - Szelektív hisztamin H3 receptor antagonisták autizmus spektrum betegség kezelésére - Google Patents
Szelektív hisztamin H3 receptor antagonisták autizmus spektrum betegség kezelésére Download PDFInfo
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- HU231525B1 HU231525B1 HUP1900190A HUP1900190A HU231525B1 HU 231525 B1 HU231525 B1 HU 231525B1 HU P1900190 A HUP1900190 A HU P1900190A HU P1900190 A HUP1900190 A HU P1900190A HU 231525 B1 HU231525 B1 HU 231525B1
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- Prior art keywords
- treatment
- ásd
- symptoms
- compound
- pharmaceutically acceptable
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- A—HUMAN NECESSITIES
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- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J3/00—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms
- A61J3/07—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms into the form of capsules or similar small containers for oral use
- A61J3/071—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms into the form of capsules or similar small containers for oral use into the form of telescopically engaged two-piece capsules
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
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- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Priority Applications (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HUP1900190A HU231525B1 (hu) | 2019-05-31 | 2019-05-31 | Szelektív hisztamin H3 receptor antagonisták autizmus spektrum betegség kezelésére |
| EP20730490.8A EP3976035A1 (en) | 2019-05-31 | 2020-05-29 | Selective histamine h3 receptor antagonists for treating autism spectrum disorder |
| CN202080040238.0A CN113905736A (zh) | 2019-05-31 | 2020-05-29 | 用于治疗孤独症谱系障碍的选择性组胺h3受体拮抗剂 |
| PCT/IB2020/055104 WO2020240489A1 (en) | 2019-05-31 | 2020-05-29 | Selective histamine h3 receptor antagonists for treating autism spectrum disorder |
| CA3141694A CA3141694A1 (en) | 2019-05-31 | 2020-05-29 | Selective histamine h3 receptor antagonists for treating autism spectrum disorder |
| US17/614,412 US20220235034A1 (en) | 2019-05-31 | 2020-05-29 | Selective histamine h3 receptor antagonists for treating autism spectrum disorder |
| EA202193155A EA202193155A1 (ru) | 2019-05-31 | 2020-05-29 | Селективные антагонисты h3-гистаминовых рецепторов для лечения расстройства аутистического спектра |
| JP2021570821A JP2022534973A (ja) | 2019-05-31 | 2020-05-29 | 自閉症スペクトラム障害を治療するための選択的ヒスタミンｈ３受容体アンタゴニスト |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HUP1900190A HU231525B1 (hu) | 2019-05-31 | 2019-05-31 | Szelektív hisztamin H3 receptor antagonisták autizmus spektrum betegség kezelésére |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUP1900190A1 HUP1900190A1 (hu) | 2020-12-28 |
| HU231525B1 true HU231525B1 (hu) | 2024-08-28 |
Family
ID=89992916
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HUP1900190A HU231525B1 (hu) | 2019-05-31 | 2019-05-31 | Szelektív hisztamin H3 receptor antagonisták autizmus spektrum betegség kezelésére |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20220235034A1 (https=) |
| EP (1) | EP3976035A1 (https=) |
| JP (1) | JP2022534973A (https=) |
| CN (1) | CN113905736A (https=) |
| CA (1) | CA3141694A1 (https=) |
| EA (1) | EA202193155A1 (https=) |
| HU (1) | HU231525B1 (https=) |
| WO (1) | WO2020240489A1 (https=) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE354568T1 (de) * | 2000-08-08 | 2007-03-15 | Ortho Mcneil Pharm Inc | Nicht-imidazol aryloxypiperidine als h3 rezeptor liganden |
| HUP1300139A2 (en) * | 2013-03-06 | 2014-09-29 | Richter Gedeon Nyrt | Phenoxypiperidine h3 antagonists |
-
2019
- 2019-05-31 HU HUP1900190A patent/HU231525B1/hu unknown
-
2020
- 2020-05-29 WO PCT/IB2020/055104 patent/WO2020240489A1/en not_active Ceased
- 2020-05-29 CN CN202080040238.0A patent/CN113905736A/zh active Pending
- 2020-05-29 CA CA3141694A patent/CA3141694A1/en active Pending
- 2020-05-29 EP EP20730490.8A patent/EP3976035A1/en not_active Withdrawn
- 2020-05-29 EA EA202193155A patent/EA202193155A1/ru unknown
- 2020-05-29 JP JP2021570821A patent/JP2022534973A/ja active Pending
- 2020-05-29 US US17/614,412 patent/US20220235034A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20220235034A1 (en) | 2022-07-28 |
| EA202193155A1 (ru) | 2022-03-22 |
| CA3141694A1 (en) | 2020-12-03 |
| JP2022534973A (ja) | 2022-08-04 |
| WO2020240489A1 (en) | 2020-12-03 |
| CN113905736A (zh) | 2022-01-07 |
| EP3976035A1 (en) | 2022-04-06 |
| HUP1900190A1 (hu) | 2020-12-28 |
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