HU198044B - Process for production of 2-oxo-1-/(substituated sulphonil)-/amin/-carbonil)-asetidines and medical preparatives containing these substances - Google Patents

Process for production of 2-oxo-1-/(substituated sulphonil)-/amin/-carbonil)-asetidines and medical preparatives containing these substances Download PDF

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Publication number
HU198044B
HU198044B HU864124A HU412486A HU198044B HU 198044 B HU198044 B HU 198044B HU 864124 A HU864124 A HU 864124A HU 412486 A HU412486 A HU 412486A HU 198044 B HU198044 B HU 198044B
Authority
HU
Hungary
Prior art keywords
oxo
amino
mmol
added
hydroxy
Prior art date
Application number
HU864124A
Other languages
English (en)
Hungarian (hu)
Other versions
HUT44535A (en
Inventor
Hermann Breuer
Uwe D Treuner
William H Koster
Robert Zahler
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of HUT44535A publication Critical patent/HUT44535A/hu
Publication of HU198044B publication Critical patent/HU198044B/hu

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
HU864124A 1985-09-26 1986-09-26 Process for production of 2-oxo-1-/(substituated sulphonil)-/amin/-carbonil)-asetidines and medical preparatives containing these substances HU198044B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US78047985A 1985-09-26 1985-09-26

Publications (2)

Publication Number Publication Date
HUT44535A HUT44535A (en) 1988-03-28
HU198044B true HU198044B (en) 1989-07-28

Family

ID=25119699

Family Applications (1)

Application Number Title Priority Date Filing Date
HU864124A HU198044B (en) 1985-09-26 1986-09-26 Process for production of 2-oxo-1-/(substituated sulphonil)-/amin/-carbonil)-asetidines and medical preparatives containing these substances

Country Status (31)

Country Link
JP (1) JPS6284082A (it)
KR (1) KR900001013B1 (it)
CN (1) CN86106980A (it)
AT (1) ATA257986A (it)
AU (1) AU600912B2 (it)
BE (1) BE905502A (it)
CA (1) CA1308719C (it)
CH (1) CH670828A5 (it)
DD (1) DD250121A5 (it)
DE (1) DE3632876A1 (it)
DK (1) DK460386A (it)
EG (1) EG18314A (it)
ES (1) ES2001995A6 (it)
FI (1) FI863890A (it)
FR (1) FR2587700B1 (it)
GB (1) GB2181130B (it)
GR (1) GR862449B (it)
HU (1) HU198044B (it)
IE (1) IE59686B1 (it)
IL (1) IL80160A (it)
IT (1) IT1214533B (it)
LU (1) LU86611A1 (it)
NL (1) NL8602446A (it)
NO (1) NO863837L (it)
NZ (1) NZ217704A (it)
PH (1) PH23315A (it)
PL (1) PL151546B1 (it)
PT (1) PT83440B (it)
SE (1) SE8604089L (it)
YU (1) YU46177B (it)
ZA (1) ZA867373B (it)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU7541487A (en) * 1986-05-23 1987-12-22 Upjohn Company, The N-1 substituted sulfonylaminocarbonyl, c-4 substituted monobactams
US5006650A (en) * 1987-02-11 1991-04-09 The Upjohn Company Novel N-1 substituted beta-lactams as antibiotics
WO1988006156A1 (en) * 1987-02-11 1988-08-25 The Upjohn Company NOVEL N-1 SUBSTITUTED beta-LACTAMS AS ANTIBIOTICS
WO1988006587A1 (en) * 1987-02-27 1988-09-07 The Upjohn Company ANTIBIOTIC beta-LACTAMS CONTAINING A PYRIDONE CARBOXYLIC ACID OR ACID DERIVATIVE
CA1317298C (en) * 1987-03-03 1993-05-04 Upjohn Company (The) Antibiotic sulfonylaminocarbonyl activated .beta.-lactams
US4762922A (en) * 1987-07-01 1988-08-09 Squibb Corporation 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4772693A (en) * 1987-07-01 1988-09-20 E. R. Squibb & Sons, Inc. 2-oxo-1-((Substituted sulfonyl)amino)-carbonyl)azetidines
EP0368908A1 (en) * 1987-07-22 1990-05-23 The Upjohn Company THERAPEUTICALLY USEFUL $g(b)-LACTAMS
US5015737A (en) * 1987-07-22 1991-05-14 The Upjohn Company Therapeutically useful beta-lactams
US4777252A (en) * 1987-08-13 1988-10-11 E. R. Squibb & Sons, Inc. 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4889930A (en) * 1987-12-21 1989-12-26 E. R. Squibb & Sons, Inc. Process for making 2-oxo-1-((substituted sulfonyl)amino)carbonzyl)azetidines and intermediates used therein
US4871841A (en) * 1987-12-23 1989-10-03 E. R. Squibb & Sons, Inc. 2-Oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
EP0336667A3 (en) * 1988-04-04 1991-04-10 E.R. Squibb & Sons, Inc. [3S(Z)]-3-[[(2-amino-4-thiazolyl)[[2-(hydroxyamino)-2-oxoethoxy]imino]acetyl]-amino]-2,2-dimethyl-4-oxo-1-azetidinyl sulfate
US4959470A (en) * 1988-08-17 1990-09-25 E. R. Squibb & Sons, Inc. 2-oxo-[[(substituted sulfonyl)-amino]carbonyl]-azetidines
EP0604365B1 (en) * 1992-12-23 1999-05-26 Novartis AG Imidazole derivatives and their use as agrochemical agents
DE69405535T2 (de) * 1994-03-11 1998-04-02 Agfa Gevaert Nv Photographisches Material, das einen neuen Typ eines Hydrazides enthält
US7511159B2 (en) * 2003-12-25 2009-03-31 Ono Pharmaceutical Co., Ltd. Azetidine ring compounds and drugs comprising the same
GB201111704D0 (en) 2011-07-07 2011-08-24 Takeda Pharmaceutical Novel compounds
GB201111705D0 (en) 2011-07-07 2011-08-24 Takeda Pharmaceutical Compounds and their use
JO3115B1 (ar) 2011-08-22 2017-09-20 Takeda Pharmaceuticals Co مركبات بيريدازينون واستخدامها كمثبطات daao
AP2014007637A0 (en) 2011-11-15 2014-05-31 Takeda Pharmaceutical Dihydroxy aromatic heterocyclic compound
GB201222711D0 (en) 2012-12-17 2013-01-30 Takeda Pharmaceutical Novel compounds
CN106986820B (zh) * 2017-02-24 2019-05-21 浙江工商大学 多功能的羟基吡啶酮衍生物及其水合物的制备法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ199981A (en) * 1981-04-09 1985-08-16 Squibb & Sons Inc 2-oxo-1-(((substituted sulphonyl)amino)carbonyl)azetidines
CA1272726C (en) * 1982-01-04 1990-08-14 2-oxo-1-(aminocarbonylaminosulfonyl- aminocarbonyl)azetidines
US4939253A (en) * 1982-08-04 1990-07-03 E. R. Squibb & Sons, Inc. 2-oxoazetidin-1-yloxy acetic acids and analogs
US4801705A (en) * 1986-06-23 1989-01-31 E. R. Squibb & Sons, Inc. 2-oxo-1-(((substituted sulfonyl)amino)-carbonyl)azetidines

Also Published As

Publication number Publication date
FI863890A (fi) 1987-03-27
FI863890A0 (fi) 1986-09-26
DE3632876A1 (de) 1987-04-02
KR900001013B1 (ko) 1990-02-24
CH670828A5 (it) 1989-07-14
AU6315686A (en) 1987-04-02
NL8602446A (nl) 1987-04-16
FR2587700B1 (fr) 1988-09-16
DK460386A (da) 1987-03-27
ATA257986A (de) 1994-07-15
IE59686B1 (en) 1994-03-23
NO863837L (no) 1987-03-27
JPS6284082A (ja) 1987-04-17
CA1308719C (en) 1992-10-13
IT1214533B (it) 1990-01-18
DK460386D0 (da) 1986-09-26
BE905502A (fr) 1987-01-16
SE8604089L (sv) 1987-03-27
HUT44535A (en) 1988-03-28
EG18314A (en) 1993-02-28
GB2181130B (en) 1989-09-20
LU86611A1 (fr) 1987-04-02
GR862449B (en) 1987-01-27
ZA867373B (en) 1987-05-27
ES2001995A6 (es) 1988-07-01
YU46177B (sh) 1993-05-28
YU165986A (en) 1988-06-30
PT83440B (pt) 1989-05-12
CN86106980A (zh) 1987-04-08
NO863837D0 (no) 1986-09-26
DD250121A5 (de) 1987-09-30
IT8621834A0 (it) 1986-09-26
GB8623151D0 (en) 1986-10-29
IL80160A0 (en) 1986-12-31
PH23315A (en) 1989-07-14
PT83440A (pt) 1986-10-01
PL261575A1 (en) 1988-07-21
NZ217704A (en) 1989-02-24
PL151546B1 (en) 1990-09-28
KR870003101A (ko) 1987-04-15
FR2587700A1 (fr) 1987-03-27
IE862547L (en) 1987-03-26
GB2181130A (en) 1987-04-15
IL80160A (en) 1991-04-15
AU600912B2 (en) 1990-08-30
SE8604089D0 (sv) 1986-09-26

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628
HMM4 Cancellation of final prot. due to non-payment of fee