HRP20211810T1 - Liječenje i prevencija prehlade korištenjem povidon-joda - Google Patents

Liječenje i prevencija prehlade korištenjem povidon-joda Download PDF

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Publication number
HRP20211810T1
HRP20211810T1 HRP20211810TT HRP20211810T HRP20211810T1 HR P20211810 T1 HRP20211810 T1 HR P20211810T1 HR P20211810T T HRP20211810T T HR P20211810TT HR P20211810 T HRP20211810 T HR P20211810T HR P20211810 T1 HRP20211810 T1 HR P20211810T1
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HR
Croatia
Prior art keywords
use according
pharmaceutical composition
cold
pharmaceutical preparation
human subject
Prior art date
Application number
HRP20211810TT
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English (en)
Inventor
Stephen Goodall
Peter Molloy
Original Assignee
Firebrick Pharma Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AU2014206143A external-priority patent/AU2014206143C1/en
Application filed by Firebrick Pharma Limited filed Critical Firebrick Pharma Limited
Publication of HRP20211810T1 publication Critical patent/HRP20211810T1/hr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00Medicinal preparations containing inorganic active ingredients
    • A61K33/18Iodine; Compounds thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/74Synthetic polymeric materials
    • A61K31/785Polymers containing nitrogen
    • A61K31/787Polymers containing nitrogen containing heterocyclic rings having nitrogen as a ring hetero atom
    • A61K31/79Polymers of vinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/02Local antiseptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Inorganic Chemistry (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Claims (15)

1. Farmaceutski pripravak koji sadrži povidon-jod (PVP-I) u koncentraciji većoj od 0,10% m/v i manjoj od oko 2,5% m/v i u kojem najmanje 50% PVP-I nije povezano s liposomima ili drugim čestičnim nosačima za upotrebu u liječenju prehlade, smanjenju simptoma prehlade, smanjenju trajanja prehlade kod ljudskog subjekta ili izbjegavanju prehlade kod ljudskog subjekta koji je bio izložen trećima sa simptomima prehlade pri čemu se farmaceutski pripravak nanosi na nosne prolaze ljudskog subjekta na sobnoj temperaturi i pri čemu je uzročnik ili potencijalni uzročnik prehlade virus koji nije virus gripe.
2. Farmaceutski pripravak koji sadrži povidon-jod (PVP-I) u koncentraciji većoj od 0,10% m/v i manjoj od oko 2,5% m/v i u kojem najmanje 50% PVP-I nije povezano s liposomima ili drugim čestičnim nosačima za uporabu u liječenju za smanjenje aktivnosti, održivosti ili broja virusa koji nisu virusi gripe unutar nosnih prolaza ljudskog subjekta, pri čemu su virusi uzročnici ili potencijalni uzročnici prehlada i farmaceutski pripravak se nanosi na nosne prolaze ljudskog subjekta na sobnoj temperaturi.
3. Farmaceutski pripravak za uporabu prema patentnom zahtjevu 1, pri čemu liječenje smanjuje rizik, učestalost ili težinu sekundarne bolesti povezane s prehladom kod ljudskog subjekta, pri čemu se sekundarna bolest odabire iz skupine koju čine bronhitis, upala srednjeg uha i sinusitis i/ili smanjuje rizik, učestalost ili težinu bolesti donjeg dišnog sustava povezane s prehladom u ljudi koji pate od KOPB, astme, emfizema ili cistične fibroze, ili osobe s narušenim imunitetom.
4. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 3, pri čemu je koncentracija PVP-I u farmaceutskom pripravku koji se primjenjuje na nosne prolaze oko 0,1% do oko 1,0% m/v, poželjno oko 0,2% do oko 0,5% m/v, poželjno oko 0,2% do oko 0,45% m/v.
5. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 4, pri čemu najmanje 70%, 80% ili 90% PVP-I nije povezano s liposomima ili drugim čestičnim nosačima.
6. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 5, pri čemu farmaceutski pripravak ne sadrži liposome.
7. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 6, pri čemu se farmaceutski pripravak primjenjuje u nosnice ljudskog subjekta, između 1 i 12 puta dnevno.
8. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 7, pri čemu je između oko 0,05 mL i oko 1,0 mL farmaceutskog pripravka primijenjeno u svaku nosnicu ljudskog subjekta pri svakoj primjeni pripravka.
9. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 8, pri čemu je uzročnik ili potencijalni uzročnik prehlade odabran iz skupine koju čine rinovirusi, humani koronavirusi, humani virusi parainfluence, humani respiratorni sincicijski virusi, adenovirusi, enterovirusi osim rinovirusa, metapneumovirusi i sve njihove kombinacije.
10. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 9, pri čemu je uzročnik ili potencijalni uzročnik prehlade humani rinovirus.
11. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1, 3 do 10, pri čemu je simptom prehlade odabran iz skupine koju čine zimica, glavobolje, bolovi i tegobe, umor, curenje iz nosa, kihanje, kašalj, začepljenost nosa, grlobolja i njihove kombinacije.
12. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 11, pri čemu je farmaceutski pripravak u obliku doziranja odabranom iz skupine koju čine intranazalne otopine, kapi, sprejevi, gelovi, aerosoli i inhalanti.
13. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 12, pri čemu farmaceutski pripravak nadalje sadrži najmanje jedno sredstvo odabrano iz skupine koju čine dekongestiv, antihistaminik, analgetik, antipiretik, protuupalno sredstvo, steroid, sredstvo za suzbijanje kašlja i ekspektorans.
14. Farmaceutski pripravak za uporabu prema bilo kojem od patentnih zahtjeva 1 do 13, pri čemu farmaceutski pripravak nadalje sadrži najmanje jedan farmaceutski prihvatljiv razrjeđivač, ekscipijent ili nosač.
15. Farmaceutski pripravak za uporabu prema patentnom zahtjevu 14, pri čemu je razrjeđivač, ekscipijent ili nosač aroma, zaslađivač, bojilo, otapalo, pufer, alkohol, polimer, surfaktant ili drugi razrjeđivač ili ekscipijent dizajniran za optimiziranje nazalne dostave, intranazalne distribucije, stabilnosti, učinkovitosti, prihvatljivosti, podnošljivosti pripravka.
HRP20211810TT 2014-07-23 2015-07-06 Liječenje i prevencija prehlade korištenjem povidon-joda HRP20211810T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AU2014206143A AU2014206143C1 (en) 2014-07-23 Treatment and prevention of the common cold using povidone-iodine
EP18152155.0A EP3326635B1 (en) 2014-07-23 2015-07-06 Treatment and prevention of the common cold using povidone-iodine

Publications (1)

Publication Number Publication Date
HRP20211810T1 true HRP20211810T1 (hr) 2022-03-04

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Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20211810TT HRP20211810T1 (hr) 2014-07-23 2015-07-06 Liječenje i prevencija prehlade korištenjem povidon-joda

Country Status (18)

Country Link
US (2) US11000542B2 (hr)
EP (2) EP3171881A4 (hr)
JP (2) JP2017522330A (hr)
CN (1) CN106794198A (hr)
AU (2) AU2015292256B2 (hr)
CA (1) CA2955982C (hr)
DK (1) DK3326635T3 (hr)
ES (1) ES2895429T3 (hr)
HK (1) HK1249851A1 (hr)
HR (1) HRP20211810T1 (hr)
HU (1) HUE056533T2 (hr)
MY (1) MY189342A (hr)
NZ (1) NZ728284A (hr)
PH (1) PH12017500135A1 (hr)
PL (1) PL3326635T3 (hr)
PT (1) PT3326635T (hr)
SG (2) SG11201700286XA (hr)
WO (1) WO2016011496A1 (hr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016011496A1 (en) 2014-07-23 2016-01-28 Firebrick Pharma Pty Ltd Treatment and prevention of the common cold using povidone-iodine
SG11202112735QA (en) * 2019-06-10 2021-12-30 Firebrick Pharma Ltd Prevention of infection by highly pathogenic viruses using topical application of povidone-iodine on mucous membranes
CN114269354A (zh) * 2019-08-30 2022-04-01 3M创新有限公司 应用消毒剂组合物进行病毒的传播预防
CN113244262A (zh) * 2020-02-07 2021-08-13 北京天衡军威医药技术开发有限公司 一种用于预防及治疗呼吸道感染性疾病的吸入粉雾制剂
CN113244263A (zh) * 2020-02-07 2021-08-13 北京天衡军威医药技术开发有限公司 一种用于预防及治疗呼吸道感染性疾病的雾化吸入制剂
EP4240340A1 (en) * 2020-11-09 2023-09-13 Rucker Capital Advisors Oral rinse, nasal spray and methods for prevention of covid-19 by lowering viral load of covid-19

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Also Published As

Publication number Publication date
CA2955982A1 (en) 2016-01-28
AU2014206143B1 (en) 2014-10-23
US20170165296A1 (en) 2017-06-15
EP3326635A1 (en) 2018-05-30
HUE056533T2 (hu) 2022-02-28
AU2015292256A1 (en) 2017-06-15
WO2016011496A1 (en) 2016-01-28
AU2019100465B4 (en) 2020-06-18
NZ728284A (en) 2020-07-31
JP2017522330A (ja) 2017-08-10
HK1249851A1 (zh) 2018-11-16
PT3326635T (pt) 2021-11-04
ES2895429T3 (es) 2022-02-21
AU2015292256B2 (en) 2020-09-17
MY189342A (en) 2022-02-04
US20200316109A1 (en) 2020-10-08
PL3326635T3 (pl) 2022-02-07
PH12017500135B1 (en) 2017-05-29
CA2955982C (en) 2023-09-05
EP3171881A4 (en) 2018-01-10
JP2021059553A (ja) 2021-04-15
US11000542B2 (en) 2021-05-11
SG11201700286XA (en) 2017-02-27
CN106794198A (zh) 2017-05-31
AU2019100465A4 (en) 2019-06-06
SG10201900559VA (en) 2019-02-27
PH12017500135A1 (en) 2017-05-29
EP3326635B1 (en) 2021-09-01
EP3171881A1 (en) 2017-05-31
DK3326635T3 (da) 2021-11-15

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