HRP20040573A2 - Substituted imidazolidines, method for the production thereof, use thereof as a drug or for diagnosis, and drug containing substituted imidazolidines - Google Patents
Substituted imidazolidines, method for the production thereof, use thereof as a drug or for diagnosis, and drug containing substituted imidazolidines Download PDFInfo
- Publication number
- HRP20040573A2 HRP20040573A2 HR20040573A HRP20040573A HRP20040573A2 HR P20040573 A2 HRP20040573 A2 HR P20040573A2 HR 20040573 A HR20040573 A HR 20040573A HR P20040573 A HRP20040573 A HR P20040573A HR P20040573 A2 HRP20040573 A2 HR P20040573A2
- Authority
- HR
- Croatia
- Prior art keywords
- ylidene
- substituted
- production
- compound
- dichlorophenyl
- Prior art date
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Transplantation (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Gastroenterology & Hepatology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10163239A DE10163239A1 (de) | 2001-12-21 | 2001-12-21 | Substituierte Imidazolidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie enthaltendes Medikament |
PCT/EP2002/013921 WO2003053434A1 (de) | 2001-12-21 | 2002-12-09 | Substituierte imidazolidine, verfahren zu ihrer herstellung, ihre verwendung als medikament oder diagnostikum sowie enthaltendes medikament |
Publications (1)
Publication Number | Publication Date |
---|---|
HRP20040573A2 true HRP20040573A2 (en) | 2004-10-31 |
Family
ID=7710363
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HR20040573A HRP20040573A2 (en) | 2001-12-21 | 2004-06-18 | Substituted imidazolidines, method for the production thereof, use thereof as a drug or for diagnosis, and drug containing substituted imidazolidines |
Country Status (27)
Country | Link |
---|---|
EP (1) | EP1461034B1 (no) |
JP (1) | JP4571803B2 (no) |
KR (1) | KR100959031B1 (no) |
CN (1) | CN100339079C (no) |
AR (1) | AR037932A1 (no) |
AT (1) | ATE345797T1 (no) |
AU (1) | AU2002361990B2 (no) |
BR (1) | BR0215154A (no) |
CA (1) | CA2470856A1 (no) |
CO (1) | CO5590925A2 (no) |
DE (2) | DE10163239A1 (no) |
DK (1) | DK1461034T3 (no) |
ES (1) | ES2275945T3 (no) |
HR (1) | HRP20040573A2 (no) |
HU (1) | HUP0600836A2 (no) |
IL (2) | IL162562A0 (no) |
MA (1) | MA27149A1 (no) |
MX (1) | MXPA04005388A (no) |
MY (1) | MY134344A (no) |
NO (1) | NO20043009L (no) |
PE (1) | PE20030741A1 (no) |
PL (1) | PL368940A1 (no) |
RS (1) | RS53204A (no) |
RU (1) | RU2004122415A (no) |
TW (1) | TW200305408A (no) |
WO (1) | WO2003053434A1 (no) |
ZA (1) | ZA200404149B (no) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10323701A1 (de) | 2003-05-22 | 2004-12-23 | Aventis Pharma Deutschland Gmbh | Verfahren zur Synthese heterocyclischer Verbindungen |
CA2531167C (en) | 2003-06-30 | 2012-05-22 | Sumitomo Chemical Company, Limited | Asymmetric urea compound and process for producing asymmetric compound by asymmetric conjugate addition reaction with the same as catalyst |
DE10341240A1 (de) * | 2003-09-08 | 2005-04-07 | Aventis Pharma Deutschland Gmbh | Substituierte Thienoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
BR112017000691B1 (pt) | 2014-07-25 | 2023-02-14 | Taisho Pharmaceutical Co., Ltd | Feniltetra-hidroisoquinolina substituído com heteroari-la, seu uso, medicamento, inibidores de nhe3, de absorção de sódio e de absorção de fósforo, promotor de secre-ção de água intestinal e fármaco profilático ou terapêu-tico para constipação |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3202660A (en) * | 1961-10-09 | 1965-08-24 | Boehringer Sohn Ingelheim | Process for the preparation of 3-arylamino-1, 3-diazacycloalkenes |
US3236857A (en) * | 1961-10-09 | 1966-02-22 | Boehringer Sohn Ingelheim | 2-(phenyl-amino)-1, 3-diazacyclopentene-(2) substitution products |
EP0070084A3 (en) * | 1981-04-24 | 1983-02-16 | Beecham Group Plc | Imidazoline derivatives |
DE3712385A1 (de) * | 1987-04-11 | 1988-10-27 | Boehringer Ingelheim Kg | 2-(phenylimino)imidazolidine |
GB9313330D0 (en) * | 1993-06-28 | 1993-08-11 | Fujisawa Pharmaceutical Co | New compound and its preparation |
EP0639573A1 (de) * | 1993-08-03 | 1995-02-22 | Hoechst Aktiengesellschaft | Benzokondensierte 5-Ringheterocyclen, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament, ihre Verwendung als Diagnostikum, sowie sie enthaltendes Medikament |
DE4328869A1 (de) * | 1993-08-27 | 1995-03-02 | Hoechst Ag | Ortho-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
KR100257129B1 (ko) * | 1993-09-11 | 2000-05-15 | 성재갑 | 신규 세팔로스포린계 항생제 및 이의 제조방법 |
US5552415A (en) * | 1993-12-21 | 1996-09-03 | Eli Lilly And Company | Method of inhibiting Alzheimer's Disease |
DE19548812A1 (de) * | 1995-12-27 | 1997-07-03 | Hoechst Ag | Verwendung von Inhibitoren des zellulären Na·+·/H·+·-Exchangers (NHE) zur Herstellung eines Medikaments zur Atemstimulation |
DE19633966A1 (de) * | 1996-08-22 | 1998-02-26 | Hoechst Ag | Phenylsubstituierte Alkenylcarbonsäure-guanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
DK0966465T3 (da) * | 1997-03-14 | 2003-10-20 | Vertex Pharma | Inhibitorer af IMPDH-enzymer |
DE19945302A1 (de) * | 1999-09-22 | 2001-03-29 | Merck Patent Gmbh | Biphenylderivate als NHE-3-Inhibitoren |
DE19950898A1 (de) * | 1999-10-22 | 2001-04-26 | Aventis Pharma Gmbh | Heterocyclisch substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
DE19960204A1 (de) * | 1999-12-14 | 2001-06-28 | Aventis Pharma Gmbh | Substituierte Norlbornylamino-Derivate, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
DE10015248A1 (de) * | 2000-03-28 | 2001-10-04 | Merck Patent Gmbh | Bisamidino-Verbindungen als NHE-3 Inhibitoren |
DE10019062A1 (de) * | 2000-04-18 | 2001-10-25 | Merck Patent Gmbh | 2-Guanidino-4-aryl-chinazoline als NHE-3 Inhibitoren |
DE10060292A1 (de) * | 2000-12-05 | 2002-06-20 | Aventis Pharma Gmbh | Verwendung substituierter Benzimidazole zur Herstellung eines Medikaments zur Behandlung von Krankheiten, welche durch Inhibierung des Na+/H+-Austauschers beeinflusst werden können und sie enthaltendes Medikament |
-
2001
- 2001-12-21 DE DE10163239A patent/DE10163239A1/de not_active Withdrawn
-
2002
- 2002-12-09 BR BR0215154-5A patent/BR0215154A/pt not_active IP Right Cessation
- 2002-12-09 DK DK02796586T patent/DK1461034T3/da active
- 2002-12-09 WO PCT/EP2002/013921 patent/WO2003053434A1/de active IP Right Grant
- 2002-12-09 ES ES02796586T patent/ES2275945T3/es not_active Expired - Lifetime
- 2002-12-09 EP EP02796586A patent/EP1461034B1/de not_active Expired - Lifetime
- 2002-12-09 DE DE50208809T patent/DE50208809D1/de not_active Expired - Lifetime
- 2002-12-09 PL PL02368940A patent/PL368940A1/xx not_active Application Discontinuation
- 2002-12-09 IL IL16256202A patent/IL162562A0/xx unknown
- 2002-12-09 HU HU0600836A patent/HUP0600836A2/hu unknown
- 2002-12-09 AU AU2002361990A patent/AU2002361990B2/en not_active Ceased
- 2002-12-09 RU RU2004122415/04A patent/RU2004122415A/ru not_active Application Discontinuation
- 2002-12-09 CN CNB028258177A patent/CN100339079C/zh not_active Expired - Fee Related
- 2002-12-09 KR KR1020047009820A patent/KR100959031B1/ko not_active IP Right Cessation
- 2002-12-09 AT AT02796586T patent/ATE345797T1/de not_active IP Right Cessation
- 2002-12-09 JP JP2003554191A patent/JP4571803B2/ja not_active Expired - Fee Related
- 2002-12-09 CA CA002470856A patent/CA2470856A1/en not_active Abandoned
- 2002-12-09 MX MXPA04005388A patent/MXPA04005388A/es active IP Right Grant
- 2002-12-09 RS YU53204A patent/RS53204A/sr unknown
- 2002-12-11 PE PE2002001194A patent/PE20030741A1/es not_active Application Discontinuation
- 2002-12-19 AR ARP020105018A patent/AR037932A1/es unknown
- 2002-12-19 TW TW091136596A patent/TW200305408A/zh unknown
- 2002-12-20 MY MYPI20024821A patent/MY134344A/en unknown
-
2004
- 2004-05-27 ZA ZA200404149A patent/ZA200404149B/en unknown
- 2004-06-01 MA MA27709A patent/MA27149A1/fr unknown
- 2004-06-16 IL IL162562A patent/IL162562A/en not_active IP Right Cessation
- 2004-06-17 CO CO04056920A patent/CO5590925A2/es not_active Application Discontinuation
- 2004-06-18 HR HR20040573A patent/HRP20040573A2/hr not_active Application Discontinuation
- 2004-07-15 NO NO20043009A patent/NO20043009L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2003053434A1 (de) | 2003-07-03 |
BR0215154A (pt) | 2004-10-19 |
ZA200404149B (en) | 2006-05-31 |
MY134344A (en) | 2007-12-31 |
CA2470856A1 (en) | 2003-07-03 |
IL162562A0 (en) | 2005-11-20 |
RS53204A (en) | 2006-10-27 |
AU2002361990B2 (en) | 2008-10-09 |
ES2275945T3 (es) | 2007-06-16 |
HUP0600836A2 (en) | 2008-04-28 |
EP1461034A1 (de) | 2004-09-29 |
EP1461034B1 (de) | 2006-11-22 |
RU2004122415A (ru) | 2005-03-27 |
AU2002361990A1 (en) | 2003-07-09 |
KR100959031B1 (ko) | 2010-05-20 |
DK1461034T3 (da) | 2007-03-26 |
JP2005516947A (ja) | 2005-06-09 |
KR20040068322A (ko) | 2004-07-30 |
DE10163239A1 (de) | 2003-07-10 |
CN100339079C (zh) | 2007-09-26 |
MA27149A1 (fr) | 2005-01-03 |
TW200305408A (en) | 2003-11-01 |
AR037932A1 (es) | 2004-12-22 |
ATE345797T1 (de) | 2006-12-15 |
NO20043009L (no) | 2004-07-15 |
JP4571803B2 (ja) | 2010-10-27 |
DE50208809D1 (de) | 2007-01-04 |
PE20030741A1 (es) | 2003-09-29 |
CN1606440A (zh) | 2005-04-13 |
CO5590925A2 (es) | 2005-12-30 |
MXPA04005388A (es) | 2004-10-11 |
IL162562A (en) | 2009-12-24 |
PL368940A1 (en) | 2005-04-04 |
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