HK1255452A1 - 改进的爱帕琳肽受体(apj)激动剂及其用途 - Google Patents
改进的爱帕琳肽受体(apj)激动剂及其用途 Download PDFInfo
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- HK1255452A1 HK1255452A1 HK18114625.4A HK18114625A HK1255452A1 HK 1255452 A1 HK1255452 A1 HK 1255452A1 HK 18114625 A HK18114625 A HK 18114625A HK 1255452 A1 HK1255452 A1 HK 1255452A1
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- agonists
- apj
- apelin receptor
- improved
- improved apelin
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| US62/265,177 | 2015-12-09 | ||
| PCT/US2016/065808 WO2017100558A1 (en) | 2015-12-09 | 2016-12-09 | Improved apelin receptor (apj) agonists and uses thereof |
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| CN108602806B (zh) | 2015-12-09 | 2022-07-12 | 研究三角协会 | 改进的爱帕琳肽受体(apj)激动剂及其用途 |
| WO2017192485A1 (en) | 2016-05-03 | 2017-11-09 | Amgen Inc. | Heterocyclic triazole compounds as agonists of the apj receptor |
| AU2017343638B2 (en) * | 2016-10-12 | 2021-12-09 | Research Triangle Institute | Heterocyclic apelin receptor (APJ) agonists and uses thereof |
| US10906890B2 (en) | 2016-11-16 | 2021-02-02 | Amgen Inc. | Triazole phenyl compounds as agonists of the APJ receptor |
| US10689367B2 (en) | 2016-11-16 | 2020-06-23 | Amgen Inc. | Triazole pyridyl compounds as agonists of the APJ receptor |
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| WO2018097945A1 (en) | 2016-11-16 | 2018-05-31 | Amgen Inc. | Heteroaryl-substituted triazoles as apj receptor agonists |
| EP3541792B1 (en) | 2016-11-16 | 2020-12-23 | Amgen Inc. | Triazole furan compounds as agonists of the apj receptor |
| MA46827A (fr) | 2016-11-16 | 2019-09-25 | Amgen Inc | Composés de triazole à substitution cycloalkyle en tant qu'agonistes du récepteur apj |
| US11247987B2 (en) | 2017-10-06 | 2022-02-15 | Forma Therapeutics, Inc. | Inhibiting ubiquitin specific peptidase 30 |
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| CN108602806A (zh) | 2018-09-28 |
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