HK1212350A1 - Glycopyrrolate salts - Google Patents

Glycopyrrolate salts

Info

Publication number
HK1212350A1
HK1212350A1 HK16100407.9A HK16100407A HK1212350A1 HK 1212350 A1 HK1212350 A1 HK 1212350A1 HK 16100407 A HK16100407 A HK 16100407A HK 1212350 A1 HK1212350 A1 HK 1212350A1
Authority
HK
Hong Kong
Prior art keywords
glycopyrrolate salts
glycopyrrolate
salts
Prior art date
Application number
HK16100407.9A
Other languages
English (en)
Chinese (zh)
Inventor
John Allan Statler
Anthony Adrian Shaw
Delphine Caroline Imbert
Jennifer Leigh Nelson
Patricia Andres
Lisa Lynn Mcqueen
Stephan Xander Mattheus Boerrigter
Jon Gordon Selbo
Mark Christopher Andres
Original Assignee
Dermira Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51428856&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1212350(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US14/024,480 external-priority patent/US9006461B2/en
Application filed by Dermira Inc filed Critical Dermira Inc
Publication of HK1212350A1 publication Critical patent/HK1212350A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12Oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
HK16100407.9A 2013-02-28 2016-01-14 Glycopyrrolate salts HK1212350A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361770920P 2013-02-28 2013-02-28
US201361770925P 2013-02-28 2013-02-28
US14/024,480 US9006461B2 (en) 2013-02-28 2013-09-11 Crystalline glycopyrrolate tosylate
US14/024,484 US8859610B2 (en) 2013-02-28 2013-09-11 Crystalline glycopyrrolate tosylate
PCT/US2014/019552 WO2014134510A1 (en) 2013-02-28 2014-02-28 Glycopyrrolate salts

Publications (1)

Publication Number Publication Date
HK1212350A1 true HK1212350A1 (en) 2016-06-10

Family

ID=51428856

Family Applications (1)

Application Number Title Priority Date Filing Date
HK16100407.9A HK1212350A1 (en) 2013-02-28 2016-01-14 Glycopyrrolate salts

Country Status (14)

Country Link
US (4) US9610278B2 (de)
EP (3) EP2961734B1 (de)
JP (2) JP6114841B2 (de)
KR (4) KR102232806B1 (de)
CN (1) CN105026369A (de)
AU (2) AU2014223172B2 (de)
CA (1) CA2902795C (de)
ES (1) ES2699257T3 (de)
HK (1) HK1212350A1 (de)
IL (2) IL240684A (de)
MX (2) MX2015011228A (de)
NZ (1) NZ710740A (de)
SG (1) SG11201506789PA (de)
WO (1) WO2014134510A1 (de)

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JP6114841B2 (ja) 2013-02-28 2017-04-12 ダーミラ, インク.Dermira, Inc. グリコピロレート塩
US9006462B2 (en) 2013-02-28 2015-04-14 Dermira, Inc. Glycopyrrolate salts
US9926270B2 (en) * 2014-08-20 2018-03-27 Dermira, Inc. Process for production of glycopyrronium tosylate
JP2017528426A (ja) * 2014-08-27 2017-09-28 ダーミラ, インク.Dermira, Inc. 多汗症を治療する方法
US20220233500A1 (en) * 2014-08-29 2022-07-28 Journey Medical Corporation Glycopyrrolate salts
CN107915666A (zh) * 2016-10-09 2018-04-17 四川海思科制药有限公司 一种格隆溴铵化合物
EP3431072B1 (de) * 2017-07-17 2019-11-06 Dr. August Wolff GmbH & Co. KG Arzneimittel Öl-in-wasser-emulsion
KR20200091395A (ko) * 2017-09-27 2020-07-30 페도라 파마슈티칼스 인코포레이티드 디아자비시클로옥탄 유도체의 결정형 및 그의 제조 방법
US20210290536A1 (en) 2018-07-24 2021-09-23 Dr. August Wolff Gmbh & Co. Kg Arzneimittel Topical emulsion of an anticholinergic compound
US20220193382A1 (en) 2019-04-10 2022-06-23 Dr. August Wolff Gmbh & Co. Kg Arzneimittel System for Dermal Application of a Pharmaceutical and/or Cosmetic Composition
CN111349036B (zh) * 2020-03-13 2022-03-08 安徽恒星制药有限公司 一种格隆溴铵的替代物及其制备方法和医药用途
TW202245748A (zh) 2021-02-05 2022-12-01 日商三和化學研究所股份有限公司 包含吡咯醣・水楊酸鹽之藥品
EP4289424A1 (de) 2021-02-05 2023-12-13 Sanwa Kagaku Kenkyusho Co., Ltd. Pharmazeutische zusammensetzung enthaltend glykopyrroniumsalicylat
EP4260852A1 (de) 2022-04-14 2023-10-18 Dr. August Wolff GmbH & Co. KG Arzneimittel Topische formulierung einer anticholinergen verbindung zur behandlung von schwerer hyperhidrose und übermässigem schwitzen
WO2023198876A1 (en) 2022-04-14 2023-10-19 Dr. August Wolff Gmbh & Co. Kg Arzneimittel Topical formulation of an anticholinergic compound for treating severe hyperhidrosis and excessive sweating

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