HK1211293A1 - Brutons tyrosine kinase inhibitors - Google Patents

Brutons tyrosine kinase inhibitors

Info

Publication number
HK1211293A1
HK1211293A1 HK15112141.6A HK15112141A HK1211293A1 HK 1211293 A1 HK1211293 A1 HK 1211293A1 HK 15112141 A HK15112141 A HK 15112141A HK 1211293 A1 HK1211293 A1 HK 1211293A1
Authority
HK
Hong Kong
Prior art keywords
tyrosine kinase
kinase inhibitors
brutons tyrosine
brutons
inhibitors
Prior art date
Application number
HK15112141.6A
Other languages
English (en)
Chinese (zh)
Inventor
‧施普林格
‧戴瓦達斯
‧加蘭
‧格拉佩豪斯
‧韓
‧霍克曼
‧休斯
‧薩亞
‧施努特
‧賽爾內斯
‧沃克
‧萬
‧邢
‧查普夫
‧施密特
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49596360&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1211293(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of HK1211293A1 publication Critical patent/HK1211293A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK15112141.6A 2012-11-02 2015-12-09 Brutons tyrosine kinase inhibitors HK1211293A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261721920P 2012-11-02 2012-11-02
US201361772028P 2013-03-04 2013-03-04
PCT/IB2013/059846 WO2014068527A1 (en) 2012-11-02 2013-11-01 Bruton's tyrosine kinase inhibitors

Publications (1)

Publication Number Publication Date
HK1211293A1 true HK1211293A1 (en) 2016-05-20

Family

ID=49596360

Family Applications (1)

Application Number Title Priority Date Filing Date
HK15112141.6A HK1211293A1 (en) 2012-11-02 2015-12-09 Brutons tyrosine kinase inhibitors

Country Status (27)

Country Link
US (4) US20150291554A1 (ko)
EP (1) EP2914586B1 (ko)
JP (1) JP6178861B2 (ko)
KR (1) KR101668574B1 (ko)
CN (1) CN105008344B (ko)
AP (1) AP2015008381A0 (ko)
AU (1) AU2013340345B2 (ko)
BR (1) BR112015009624A2 (ko)
CA (1) CA2888960C (ko)
CL (1) CL2015001168A1 (ko)
CO (1) CO7350624A2 (ko)
CR (1) CR20150228A (ko)
DO (1) DOP2015000100A (ko)
EA (1) EA201500393A1 (ko)
ES (1) ES2625944T3 (ko)
GE (1) GEP201606597B (ko)
HK (1) HK1211293A1 (ko)
IL (1) IL238571A0 (ko)
MD (1) MD20150035A2 (ko)
MX (1) MX2015005422A (ko)
NI (1) NI201500059A (ko)
PE (1) PE20151070A1 (ko)
PH (1) PH12015500940A1 (ko)
SG (1) SG11201502893WA (ko)
TN (1) TN2015000168A1 (ko)
TW (1) TWI518080B (ko)
WO (1) WO2014068527A1 (ko)

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AU2013312296B2 (en) 2012-09-10 2017-06-22 Principia Biopharma Inc. Pyrazolopyrimidine compounds as kinase inhibitors
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KR102311329B1 (ko) * 2013-03-15 2021-10-14 얀센 파마슈티카 엔.브이. 약제를 제조하기 위한 방법 및 중간체
WO2014152114A1 (en) 2013-03-15 2014-09-25 Boehringer Ingelheim International Gmbh Heteroaromatic compounds as btk inhibitors
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KR102272792B1 (ko) * 2013-09-30 2021-07-05 광저우 이노케어 파마 테크 씨오., 엘티디. Btk의 치환된 니코틴이미드 저해제 및 그의 제조 방법 및 암, 염증 및 자가면역 질환에의 용도
JP6486954B2 (ja) * 2014-01-29 2019-03-20 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Btk阻害剤としてのピラゾール化合物
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EP3390390B1 (en) 2015-12-16 2021-09-01 Boehringer Ingelheim International Gmbh Bipyrazolyl derivatives useful for the treatment of autoimmune diseases
EP3402789B1 (en) 2016-01-13 2020-03-18 Boehringer Ingelheim International Gmbh Isoquinolones as btk inhibitors
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WO2019091438A1 (zh) * 2017-11-10 2019-05-16 苏州信诺维医药科技有限公司 作为btk抑制剂的5-氨基吡唑甲酰胺化合物的无定型固体分散体
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Also Published As

Publication number Publication date
PE20151070A1 (es) 2015-08-01
EP2914586B1 (en) 2017-04-05
AU2013340345A1 (en) 2015-04-30
MD20150035A2 (ro) 2015-10-31
DOP2015000100A (es) 2015-12-31
CA2888960A1 (en) 2014-05-08
US20190202798A1 (en) 2019-07-04
KR20150075114A (ko) 2015-07-02
US10815213B2 (en) 2020-10-27
KR101668574B1 (ko) 2016-10-24
EP2914586A1 (en) 2015-09-09
TW201431851A (zh) 2014-08-16
MX2015005422A (es) 2015-08-05
AP2015008381A0 (en) 2015-04-30
TWI518080B (zh) 2016-01-21
CL2015001168A1 (es) 2015-07-10
CN105008344B (zh) 2017-07-25
GEP201606597B (en) 2017-01-10
TN2015000168A1 (fr) 2016-10-03
JP6178861B2 (ja) 2017-08-09
CR20150228A (es) 2015-09-14
NI201500059A (es) 2015-06-05
US20170283393A1 (en) 2017-10-05
US20210002251A1 (en) 2021-01-07
CA2888960C (en) 2017-08-15
AU2013340345B2 (en) 2016-10-27
CN105008344A (zh) 2015-10-28
JP2015535277A (ja) 2015-12-10
IL238571A0 (en) 2015-06-30
WO2014068527A1 (en) 2014-05-08
US20150291554A1 (en) 2015-10-15
EA201500393A1 (ru) 2016-05-31
CO7350624A2 (es) 2015-08-10
SG11201502893WA (en) 2015-05-28
ES2625944T3 (es) 2017-07-21
PH12015500940A1 (en) 2015-06-29
BR112015009624A2 (pt) 2017-11-14
US10266513B2 (en) 2019-04-23

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