HK1208859A1 - Catechol o-methyltransferase activity inhibiting compounds o- - Google Patents

Catechol o-methyltransferase activity inhibiting compounds o-

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Publication number
HK1208859A1
HK1208859A1 HK15109586.4A HK15109586A HK1208859A1 HK 1208859 A1 HK1208859 A1 HK 1208859A1 HK 15109586 A HK15109586 A HK 15109586A HK 1208859 A1 HK1208859 A1 HK 1208859A1
Authority
HK
Hong Kong
Prior art keywords
catechol
inhibiting compounds
methyltransferase activity
activity inhibiting
methyltransferase
Prior art date
Application number
HK15109586.4A
Other languages
English (en)
Chinese (zh)
Inventor
Marko Ahlmark
Belle David Din
Mika Kauppala
Anne Luiro
Taina Pajunen
Jarmo Pystynen
Eija Tiainen
Matti Vaismaa
Josef Messinger
Original Assignee
Orion Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Orion Corp filed Critical Orion Corp
Publication of HK1208859A1 publication Critical patent/HK1208859A1/xx

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    • A61K31/275—Nitriles; Isonitriles
    • A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid, pantothenic acid
    • A61K31/198—Alpha-aminoacids, e.g. alanine, edetic acids [EDTA]
    • A—HUMAN NECESSITIES
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    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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US20170165219A1 (en) 2017-06-15
TN2014000474A1 (en) 2016-03-30
MX357896B (es) 2018-07-27
JP2015522547A (ja) 2015-08-06
TW201408629A (zh) 2014-03-01
US20220047540A1 (en) 2022-02-17
CO7151502A2 (es) 2014-12-29
CN104334525B (zh) 2017-05-10
US9458128B2 (en) 2016-10-04
PL2855426T3 (pl) 2017-07-31
MD20140124A2 (ro) 2015-03-31

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