HK1200456A1 - Aryl or n-heteroaryl substituted methanesulfonamide derivatives as vanilloid receptor ligands n- - Google Patents

Aryl or n-heteroaryl substituted methanesulfonamide derivatives as vanilloid receptor ligands n-

Info

Publication number
HK1200456A1
HK1200456A1 HK15101022.3A HK15101022A HK1200456A1 HK 1200456 A1 HK1200456 A1 HK 1200456A1 HK 15101022 A HK15101022 A HK 15101022A HK 1200456 A1 HK1200456 A1 HK 1200456A1
Authority
HK
Hong Kong
Prior art keywords
aryl
receptor ligands
heteroaryl substituted
vanilloid receptor
methanesulfonamide derivatives
Prior art date
Application number
HK15101022.3A
Other languages
English (en)
Chinese (zh)
Inventor
Robert Frank-Foltyn
Gregor Bahrenberg
Thomas Christoph
Bernhard Lesch
Jeewoo Lee
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of HK1200456A1 publication Critical patent/HK1200456A1/xx

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom
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    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Virology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
HK15101022.3A 2011-09-26 2015-01-29 Aryl or n-heteroaryl substituted methanesulfonamide derivatives as vanilloid receptor ligands n- HK1200456A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP11007807 2011-09-26
PCT/EP2012/068877 WO2013045447A1 (en) 2011-09-26 2012-09-25 Aryl or n-heteroaryl substituted methanesulfonamide derivatives as vanilloid receptor ligands

Publications (1)

Publication Number Publication Date
HK1200456A1 true HK1200456A1 (en) 2015-08-07

Family

ID=46888474

Family Applications (1)

Application Number Title Priority Date Filing Date
HK15101022.3A HK1200456A1 (en) 2011-09-26 2015-01-29 Aryl or n-heteroaryl substituted methanesulfonamide derivatives as vanilloid receptor ligands n-

Country Status (13)

Country Link
US (1) US8937092B2 (xx)
EP (1) EP2760835A1 (xx)
JP (1) JP2014531451A (xx)
KR (1) KR20140074363A (xx)
CN (1) CN103958472A (xx)
AR (1) AR088002A1 (xx)
AU (1) AU2012314587A1 (xx)
BR (1) BR112014006788A2 (xx)
CA (1) CA2849960A1 (xx)
HK (1) HK1200456A1 (xx)
MX (1) MX2014003455A (xx)
TW (1) TW201317214A (xx)
WO (1) WO2013045447A1 (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015004035A1 (en) * 2013-07-09 2015-01-15 Lonza Ltd Method for preparation of 4-alkoxy-1,1,1-trifluorobut-3-en-2-ones from trifluoroacetylacetic acid
TW201625511A (zh) 2014-06-26 2016-07-16 隆沙有限公司 由１，１，１－三氟丙酮製備４－烷氧基－１，１，１－三氟丁－３－烯－２－酮之方法
BR112017010402B1 (pt) 2014-11-24 2023-12-12 Medifron Dbt Inc Carboxamida substituída à base de tiazol e oxazol e derivados de ureia como ligantes de receptor vanilóide ii
EP3130589A1 (en) * 2015-08-13 2017-02-15 Grünenthal GmbH Heterocyclic aza compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7135575B2 (en) 2003-03-03 2006-11-14 Array Biopharma, Inc. P38 inhibitors and methods of use thereof
JP2005314407A (ja) * 2004-03-31 2005-11-10 Nippon Nohyaku Co Ltd 新規なハロアルキルスルホンアニリド誘導体、除草剤及びその使用方法並びにその中間体
BRPI0618417A2 (pt) 2005-10-19 2012-07-31 Gruenenthal Chemie novos ligandos de receptores de vanilàide e seu uso para produzir medicamentos
CN102869261A (zh) * 2010-03-01 2013-01-09 瑞科西有限公司 化合物及其治疗应用

Also Published As

Publication number Publication date
BR112014006788A2 (pt) 2017-06-13
CA2849960A1 (en) 2013-04-04
AU2012314587A1 (en) 2014-03-06
AR088002A1 (es) 2014-04-30
JP2014531451A (ja) 2014-11-27
CN103958472A (zh) 2014-07-30
KR20140074363A (ko) 2014-06-17
US8937092B2 (en) 2015-01-20
MX2014003455A (es) 2014-06-04
EP2760835A1 (en) 2014-08-06
US20130079377A1 (en) 2013-03-28
TW201317214A (zh) 2013-05-01
WO2013045447A1 (en) 2013-04-04

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