HK1198741A1 - New (trimethoxyphenylamino)pyrimidinyl formulations () - Google Patents

New (trimethoxyphenylamino)pyrimidinyl formulations ()

Info

Publication number
HK1198741A1
HK1198741A1 HK14112235.4A HK14112235A HK1198741A1 HK 1198741 A1 HK1198741 A1 HK 1198741A1 HK 14112235 A HK14112235 A HK 14112235A HK 1198741 A1 HK1198741 A1 HK 1198741A1
Authority
HK
Hong Kong
Prior art keywords
trimethoxyphenylamino
pyrimidinyl
formulations
new
pyrimidinyl formulations
Prior art date
Application number
HK14112235.4A
Other languages
English (en)
Chinese (zh)
Inventor
Farhan Abdul Karim Alhusban
Ian Paul Gabbott
Bindhumadhavan Gururajan
Dawn Sievwright
David Bradley Brook Simpson
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46875902&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1198741(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of HK1198741A1 publication Critical patent/HK1198741A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53831,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Transplantation (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK14112235.4A 2011-07-28 2014-12-04 New (trimethoxyphenylamino)pyrimidinyl formulations () HK1198741A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161512621P 2011-07-28 2011-07-28
PCT/GB2012/051791 WO2013014454A1 (fr) 2011-07-28 2012-07-26 Nouvelles formulations de (triméthoxyphénylamino)pyrimidinyle

Publications (1)

Publication Number Publication Date
HK1198741A1 true HK1198741A1 (en) 2015-06-05

Family

ID=46875902

Family Applications (1)

Application Number Title Priority Date Filing Date
HK14112235.4A HK1198741A1 (en) 2011-07-28 2014-12-04 New (trimethoxyphenylamino)pyrimidinyl formulations ()

Country Status (26)

Country Link
US (2) US8771648B2 (fr)
EP (1) EP2736487B1 (fr)
JP (1) JP6019116B2 (fr)
KR (2) KR102090440B1 (fr)
CN (1) CN103826610B (fr)
AR (1) AR087371A1 (fr)
AU (1) AU2012288632B2 (fr)
BR (1) BR112014001999B1 (fr)
CA (1) CA2843138C (fr)
CY (1) CY1122596T1 (fr)
DK (1) DK2736487T3 (fr)
EA (1) EA028432B1 (fr)
ES (1) ES2710423T3 (fr)
HK (1) HK1198741A1 (fr)
HR (1) HRP20190186T1 (fr)
HU (1) HUE042611T2 (fr)
LT (1) LT2736487T (fr)
MX (1) MX339685B (fr)
PL (1) PL2736487T3 (fr)
PT (1) PT2736487T (fr)
RS (1) RS58433B1 (fr)
SI (1) SI2736487T1 (fr)
TR (1) TR201901792T4 (fr)
TW (1) TW201311251A (fr)
UY (1) UY34223A (fr)
WO (1) WO2013014454A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2380551T3 (es) * 2006-11-21 2012-05-16 Rigel Pharmaceuticals, Inc. Sales de profármaco de compuestos de 2,4-pirimidindiamina y sus usos
CA2843138C (fr) 2011-07-28 2020-06-02 Rigel Pharmaceuticals, Inc. Nouvelles formulations de (trimethoxyphenylamino)pyrimidinyle
JP6853786B2 (ja) 2015-04-02 2021-03-31 ストラ エンソ オーワイジェイ 活性化リグニン組成物、その製造方法及びその使用
WO2016172053A1 (fr) 2015-04-24 2016-10-27 Rigel Pharmaceuticals, Inc. Méthodes de traitement d'une maladie résistante à l'ibrutinib
EP4185126A1 (fr) * 2020-07-24 2023-05-31 DSM IP Assets B.V. Nouveaux comprimés à dissolution rapide

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
CN103169708B (zh) 2002-07-29 2018-02-02 里格尔药品股份有限公司 用2,4‑嘧啶二胺化合物治疗或者预防自体免疫性疾病的方法
RS53109B (en) 2003-07-30 2014-06-30 Rigel Pharmaceuticals Inc. 2,4 PIRIMIDINDIAMINE COMPOUNDS FOR USE IN TREATMENT OR PREVENTION OF AUTOIMMUNE DISEASES
DK1663242T3 (da) 2003-08-07 2011-08-01 Rigel Pharmaceuticals Inc 2,4-Pyrimidindiamin-forbindelser og anvendelse som antiproliferative midler
US20060051406A1 (en) * 2004-07-23 2006-03-09 Manjeet Parmar Formulation of insoluble small molecule therapeutics in lipid-based carriers
EP1794135A1 (fr) * 2004-09-27 2007-06-13 Amgen Inc. Composes heterocycliques substitues et procedes d'utilisation
ES2337496T3 (es) * 2005-01-19 2010-04-26 Rigel Pharmaceuticals, Inc. Profarmacos de compuestos de 2,4-pirimidindiamina y sus usos.
US8227455B2 (en) 2005-04-18 2012-07-24 Rigel Pharmaceuticals, Inc. Methods of treating cell proliferative disorders
JP2009518443A (ja) * 2005-12-06 2009-05-07 リゲル ファーマシューティカルズ インコーポレーティッド 脂質を主材料とする担体に内封された、不溶性小分子治療剤の製剤
CA2642211C (fr) * 2006-02-17 2012-01-24 Rigel Pharmaceuticals, Inc. Composes de 2,4-pyrimidinediamine pour le traitement ou la prevention de maladies autoimmunes
US20090048214A1 (en) * 2006-11-15 2009-02-19 Rigel Pharmaceuticals, Inc Methods for Treating Renal Tumors Using 2, 4-Pyrimidinediamine Drug and Prodrug Compounds
ES2380551T3 (es) * 2006-11-21 2012-05-16 Rigel Pharmaceuticals, Inc. Sales de profármaco de compuestos de 2,4-pirimidindiamina y sus usos
US20090012045A1 (en) * 2007-06-26 2009-01-08 Rigel Pharmaceuticals, Inc. Methods of Treating Cell Proliferative Disorders
WO2009029682A1 (fr) * 2007-08-28 2009-03-05 Rigel Pharmaceuticals, Inc. Thérapie de combinaison avec un inhibiteur de la kinase syk
EA020210B1 (ru) * 2007-11-07 2014-09-30 Райджел Фармасьютикалз, Инк. Влажное гранулирование с использованием вещества, связывающего воду
DK2252300T3 (en) 2008-02-22 2017-02-06 Rigel Pharmaceuticals Inc USE OF 2,4-PYRIMIDINE DIAMINES TO TREAT Atherosclerosis
UA108077C2 (xx) 2009-07-02 2015-03-25 Синтез динатрієвої солі n4-(2,2-диметил-4-$(дигідрофосфонокси)метил]-3-оксо-5-піридо$1,4]оксазин-6-іл)-5-фтор-n2-(3,4,5-триметоксифеніл)-2,4-піримідиндіаміну
WO2011009075A2 (fr) 2009-07-17 2011-01-20 Rigel Pharmaceuticals, Inc. Composés 2,4-pyrimidine diamine deutérés et leurs promédicaments et leurs utilisations
WO2011063241A1 (fr) 2009-11-20 2011-05-26 Rigel Pharmaceuticals, Inc. Composés 2,4-pyrimidinediamines et promédicaments de ceux-ci et leurs utilisations
JP6067550B2 (ja) 2010-04-13 2017-01-25 ライジェル ファーマシューティカルズ, インコーポレイテッド 2,4−ピリミジンジアミン化合物およびそのプロドラッグならびにそれらの使用
CA2843138C (fr) 2011-07-28 2020-06-02 Rigel Pharmaceuticals, Inc. Nouvelles formulations de (trimethoxyphenylamino)pyrimidinyle

Also Published As

Publication number Publication date
EP2736487A1 (fr) 2014-06-04
SI2736487T1 (sl) 2019-04-30
TW201311251A (zh) 2013-03-16
BR112014001999B1 (pt) 2023-11-28
CN103826610B (zh) 2017-08-04
PT2736487T (pt) 2019-02-13
CA2843138A1 (fr) 2013-01-31
JP6019116B2 (ja) 2016-11-02
EA028432B1 (ru) 2017-11-30
CY1122596T1 (el) 2021-01-27
LT2736487T (lt) 2019-02-25
HUE042611T2 (hu) 2019-07-29
CA2843138C (fr) 2020-06-02
AU2012288632B2 (en) 2017-08-17
KR102024120B1 (ko) 2019-09-23
US8951504B2 (en) 2015-02-10
ES2710423T3 (es) 2019-04-25
EP2736487B1 (fr) 2018-11-07
TR201901792T4 (tr) 2019-03-21
JP2014521630A (ja) 2014-08-28
US20130058876A1 (en) 2013-03-07
US20140271493A1 (en) 2014-09-18
UY34223A (es) 2013-02-28
RS58433B1 (sr) 2019-04-30
CN103826610A (zh) 2014-05-28
EA201490363A1 (ru) 2014-06-30
HRP20190186T1 (hr) 2019-03-22
US8771648B2 (en) 2014-07-08
BR112014001999A2 (pt) 2017-02-21
MX339685B (es) 2016-06-06
WO2013014454A1 (fr) 2013-01-31
KR102090440B1 (ko) 2020-03-17
AR087371A1 (es) 2014-03-19
PL2736487T3 (pl) 2019-06-28
KR20190109576A (ko) 2019-09-25
KR20140058576A (ko) 2014-05-14
AU2012288632A1 (en) 2014-02-20
DK2736487T3 (en) 2019-03-04
MX2014001065A (es) 2014-08-01

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