HK1180326A1 - 吡啶酮和氮雜吡啶酮化合物及使用方法 - Google Patents

吡啶酮和氮雜吡啶酮化合物及使用方法

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Publication number
HK1180326A1
HK1180326A1 HK13107639.7A HK13107639A HK1180326A1 HK 1180326 A1 HK1180326 A1 HK 1180326A1 HK 13107639 A HK13107639 A HK 13107639A HK 1180326 A1 HK1180326 A1 HK 1180326A1
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HK
Hong Kong
Prior art keywords
pyridone
aza
methods
compounds
pyridone compounds
Prior art date
Application number
HK13107639.7A
Other languages
English (en)
Inventor
Antonio J M Barbosa
Peter A Blomgren
Kevin S Currie
Ravi Krishnamoorthy
Jeffrey E Kropf
Seung H Lee
Scott A Mitchell
Daniel ORTWINE
Aaron C Schmitt
Xiaojing Wang
Jianjun Xu
Wendy Young
Honglu Zhang
Zhongdong Zhao
Pavel E Zhichkin
Original Assignee
Gilead Connecticut Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US33235310P priority Critical
Priority to US201161443952P priority
Priority to PCT/US2011/035596 priority patent/WO2011140488A1/en
Application filed by Gilead Connecticut Inc filed Critical Gilead Connecticut Inc
Publication of HK1180326A1 publication Critical patent/HK1180326A1/zh

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    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
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HK13107639.7A 2010-05-07 2013-06-28 吡啶酮和氮雜吡啶酮化合物及使用方法 HK1180326A1 (zh)

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US33235310P true 2010-05-07 2010-05-07
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PCT/US2011/035596 WO2011140488A1 (en) 2010-05-07 2011-05-06 Pyridone and aza-pyridone compounds and methods of use

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EP2566869B1 (en) * 2010-05-07 2016-03-02 Gilead Connecticut, Inc. Pyridone and aza-pyridone compounds and methods of use
US20130116231A1 (en) * 2010-07-12 2013-05-09 Merck Sharp & Dohme Corp. Tyrosine kinase inhibitors
CN106220614B (zh) * 2010-09-01 2019-07-16 吉利德康涅狄格有限公司 吡啶酮/吡嗪酮、其制备方法及使用方法
BR112013007499A2 (pt) * 2010-09-01 2016-07-12 Genentech Inc piridazinonas - métodos de criação e usos
US8722676B2 (en) 2011-11-03 2014-05-13 Genentech, Inc. Bicyclic piperazine compounds
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