HK1164057A1 - 含有剛性部分的吡啶並 吲哚類化合物 - Google Patents

含有剛性部分的吡啶並 吲哚類化合物

Info

Publication number
HK1164057A1
HK1164057A1 HK12104892.7A HK12104892A HK1164057A1 HK 1164057 A1 HK1164057 A1 HK 1164057A1 HK 12104892 A HK12104892 A HK 12104892A HK 1164057 A1 HK1164057 A1 HK 1164057A1
Authority
HK
Hong Kong
Prior art keywords
pyrido
containing rigid
rigid moieties
indoles containing
indoles
Prior art date
Application number
HK12104892.7A
Other languages
English (en)
Inventor
David T Hung
Andrew Asher Protter
Jain Rajendra Parasmal G
Sarvajit Chakravarty
Marco Giorgetti
Original Assignee
梅迪維新技術公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 梅迪維新技術公司 filed Critical 梅迪維新技術公司
Publication of HK1164057A1 publication Critical patent/HK1164057A1/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HK12104892.7A 2008-10-31 2012-05-18 含有剛性部分的吡啶並 吲哚類化合物 HK1164057A1 (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US11051908P 2008-10-31 2008-10-31
US17396009P 2009-04-29 2009-04-29
US24515009P 2009-09-23 2009-09-23
PCT/US2009/062869 WO2010051501A1 (en) 2008-10-31 2009-10-30 Pyrido (4,3-b) indoles containing rigid moieties

Publications (1)

Publication Number Publication Date
HK1164057A1 true HK1164057A1 (zh) 2012-09-21

Family

ID=42129313

Family Applications (1)

Application Number Title Priority Date Filing Date
HK12104892.7A HK1164057A1 (zh) 2008-10-31 2012-05-18 含有剛性部分的吡啶並 吲哚類化合物

Country Status (11)

Country Link
US (3) US8907097B2 (zh)
EP (1) EP2346332A4 (zh)
JP (2) JP5588991B2 (zh)
CN (1) CN102271508B (zh)
AR (1) AR073923A1 (zh)
AU (1) AU2009308706C1 (zh)
BR (1) BRPI0919948A2 (zh)
CA (1) CA2742320A1 (zh)
HK (1) HK1164057A1 (zh)
TW (1) TWI477503B (zh)
WO (1) WO2010051501A1 (zh)

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US9458155B2 (en) 2016-10-04
AU2009308706A1 (en) 2010-05-06
TW201022264A (en) 2010-06-16
BRPI0919948A2 (pt) 2015-08-25
US8906925B2 (en) 2014-12-09
US8907097B2 (en) 2014-12-09
JP2014133759A (ja) 2014-07-24
CA2742320A1 (en) 2010-05-06
CN102271508A (zh) 2011-12-07
US20100216814A1 (en) 2010-08-26
JP5588991B2 (ja) 2014-09-10
AU2009308706B2 (en) 2015-09-03
AU2009308706C1 (en) 2016-01-21
EP2346332A4 (en) 2012-08-08
US20150051218A1 (en) 2015-02-19
AR073923A1 (es) 2010-12-09
JP2012507566A (ja) 2012-03-29
US20130190322A1 (en) 2013-07-25
WO2010051501A1 (en) 2010-05-06
EP2346332A1 (en) 2011-07-27
CN102271508B (zh) 2015-04-29
TWI477503B (zh) 2015-03-21

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