HK1053789A1 - Il-8受體拮抗劑 - Google Patents
Il-8受體拮抗劑Info
- Publication number
- HK1053789A1 HK1053789A1 HK03104498.6A HK03104498A HK1053789A1 HK 1053789 A1 HK1053789 A1 HK 1053789A1 HK 03104498 A HK03104498 A HK 03104498A HK 1053789 A1 HK1053789 A1 HK 1053789A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- receptor antagonists
- antagonists
- receptor
- Prior art date
Links
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- C07C311/50—Compounds containing any of the groups, X being a hetero atom, Y being any atom
- C07C311/52—Y being a hetero atom
- C07C311/64—X and Y being nitrogen atoms, e.g. N-sulfonylguanidine
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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- C—CHEMISTRY; METALLURGY
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- C07C311/47—Y being a hetero atom
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- C07D—HETEROCYCLIC COMPOUNDS
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- C07D207/14—Nitrogen atoms not forming part of a nitro radical
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- Diabetes (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US19213200P | 2000-03-24 | 2000-03-24 | |
PCT/US2001/009216 WO2001072960A2 (en) | 2000-03-24 | 2001-03-23 | Il-8 receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1053789A1 true HK1053789A1 (zh) | 2003-11-07 |
Family
ID=22708394
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK03104498.6A HK1053789A1 (zh) | 2000-03-24 | 2003-06-23 | Il-8受體拮抗劑 |
Country Status (31)
Country | Link |
---|---|
US (1) | US6680317B2 (zh) |
EP (1) | EP1272175B1 (zh) |
JP (1) | JP2004508287A (zh) |
KR (1) | KR20040014901A (zh) |
CN (1) | CN1452483A (zh) |
AP (1) | AP1548A (zh) |
AR (1) | AR031101A1 (zh) |
AT (1) | ATE464893T1 (zh) |
AU (1) | AU2001249354A1 (zh) |
BG (1) | BG107035A (zh) |
BR (1) | BR0108867A (zh) |
CA (1) | CA2403787A1 (zh) |
CZ (1) | CZ20023192A3 (zh) |
DE (1) | DE60141896D1 (zh) |
DZ (1) | DZ3333A1 (zh) |
EA (1) | EA200201019A1 (zh) |
ES (1) | ES2344587T3 (zh) |
HK (1) | HK1053789A1 (zh) |
HU (1) | HUP0302614A3 (zh) |
IL (1) | IL151210A0 (zh) |
MA (1) | MA25739A1 (zh) |
MX (1) | MXPA02009355A (zh) |
MY (1) | MY128154A (zh) |
NO (1) | NO20024554D0 (zh) |
OA (1) | OA12235A (zh) |
PE (1) | PE20020839A1 (zh) |
PL (1) | PL205103B1 (zh) |
SK (1) | SK13682002A3 (zh) |
UY (1) | UY26627A1 (zh) |
WO (1) | WO2001072960A2 (zh) |
ZA (1) | ZA200207576B (zh) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CO5170528A1 (es) * | 1999-05-28 | 2002-06-27 | Smithkline Beecham Corp | Antagonistas de los receptores de la il-8 nistas del recpetor de la il-8 |
MY143477A (en) * | 2002-10-29 | 2011-05-31 | Smithkline Beecham Corp | Il-8 receptor antagonists |
EP1745032B1 (en) | 2004-05-12 | 2013-07-31 | Merck Sharp & Dohme Corp. | CXCR1 and CXCR2 chemokine antagonists |
US20070249625A1 (en) * | 2004-10-20 | 2007-10-25 | Jakob Busch-Petersen | Il-8 Receptor Antagonists |
RU2008145871A (ru) * | 2006-04-21 | 2010-05-27 | Смитклайн Бичам Корпорейшн (US) | Антагонисты рецептора il-8 |
PL2009992T3 (pl) * | 2006-04-21 | 2012-11-30 | Glaxosmithkline Llc | Antagoniści receptora IL-8 |
TW200817006A (en) * | 2006-06-23 | 2008-04-16 | Smithkline Beecham Corp | IL-8 receptor antagonist |
US20090131329A1 (en) * | 2007-09-14 | 2009-05-21 | Edmund John Miller | Treatment for allograft rejection |
AU2011295727B2 (en) * | 2010-09-03 | 2015-04-02 | Forma Tm, Llc. | Guanidine compounds and compositions for the inhibition of NAMPT |
US8648070B2 (en) | 2010-12-17 | 2014-02-11 | Boehringer Ingelheim International Gmbh | Bicyclic ring system substituted sulfonamide functionalised phenols as medicaments |
IN2014DN09251A (zh) * | 2012-05-08 | 2015-07-10 | Ishihara Sangyo Kaisha | |
US20230046077A1 (en) | 2019-02-07 | 2023-02-16 | Bayer Aktiengesellschaft | 3-amino-2-[2-(acylamino)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one as csnk1 inhibitors |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH11503110A (ja) | 1995-02-17 | 1999-03-23 | スミスクライン・ビーチャム・コーポレイション | Il−8受容体拮抗剤 |
AR008290A1 (es) * | 1996-08-15 | 1999-12-29 | Smithkline Beecham Corp | Nuevos compuestos que contienen guanidina utiles como antagonistas de los receptores de il-8, composiciones farmaceuticas que los contienenprocedimiento para la preparacion de dichos compuestos y procedimiento para la preparacion de intermediarios. |
US6214880B1 (en) * | 1998-09-23 | 2001-04-10 | Tularik Inc. | Arylsulfonanilide ureas |
UY25842A1 (es) * | 1998-12-16 | 2001-04-30 | Smithkline Beecham Corp | Antagonistas de receptores de il-8 |
-
2001
- 2001-03-21 UY UY26627A patent/UY26627A1/es not_active Application Discontinuation
- 2001-03-22 AR ARP010101346A patent/AR031101A1/es not_active Application Discontinuation
- 2001-03-22 MY MYPI20011375A patent/MY128154A/en unknown
- 2001-03-23 CA CA002403787A patent/CA2403787A1/en not_active Abandoned
- 2001-03-23 KR KR1020027012514A patent/KR20040014901A/ko active IP Right Grant
- 2001-03-23 AT AT01922568T patent/ATE464893T1/de not_active IP Right Cessation
- 2001-03-23 MX MXPA02009355A patent/MXPA02009355A/es active IP Right Grant
- 2001-03-23 PE PE2001000277A patent/PE20020839A1/es not_active Application Discontinuation
- 2001-03-23 EA EA200201019A patent/EA200201019A1/ru unknown
- 2001-03-23 EP EP01922568A patent/EP1272175B1/en not_active Expired - Lifetime
- 2001-03-23 HU HU0302614A patent/HUP0302614A3/hu unknown
- 2001-03-23 ES ES01922568T patent/ES2344587T3/es not_active Expired - Lifetime
- 2001-03-23 IL IL15121001A patent/IL151210A0/xx unknown
- 2001-03-23 BR BR0108867-0A patent/BR0108867A/pt not_active IP Right Cessation
- 2001-03-23 DZ DZ013333A patent/DZ3333A1/fr active
- 2001-03-23 AP APAP/P/2002/002599A patent/AP1548A/en active
- 2001-03-23 WO PCT/US2001/009216 patent/WO2001072960A2/en active Application Filing
- 2001-03-23 AU AU2001249354A patent/AU2001249354A1/en not_active Abandoned
- 2001-03-23 OA OA1200200297A patent/OA12235A/en unknown
- 2001-03-23 CN CN01806920A patent/CN1452483A/zh active Pending
- 2001-03-23 SK SK1368-2002A patent/SK13682002A3/sk not_active Application Discontinuation
- 2001-03-23 JP JP2001571875A patent/JP2004508287A/ja not_active Withdrawn
- 2001-03-23 CZ CZ20023192A patent/CZ20023192A3/cs unknown
- 2001-03-23 US US10/221,908 patent/US6680317B2/en not_active Expired - Fee Related
- 2001-03-23 PL PL366315A patent/PL205103B1/pl not_active IP Right Cessation
- 2001-03-23 DE DE60141896T patent/DE60141896D1/de not_active Expired - Lifetime
-
2002
- 2002-08-26 BG BG107035A patent/BG107035A/bg unknown
- 2002-09-20 MA MA26831A patent/MA25739A1/fr unknown
- 2002-09-20 ZA ZA200207576A patent/ZA200207576B/en unknown
- 2002-09-23 NO NO20024554A patent/NO20024554D0/no not_active Application Discontinuation
-
2003
- 2003-06-23 HK HK03104498.6A patent/HK1053789A1/zh unknown
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