HK1043369B - Compounds for the modulation of ppar-gamma activity - Google Patents
Compounds for the modulation of ppar-gamma activity Download PDFInfo
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- HK1043369B HK1043369B HK02105143.3A HK02105143A HK1043369B HK 1043369 B HK1043369 B HK 1043369B HK 02105143 A HK02105143 A HK 02105143A HK 1043369 B HK1043369 B HK 1043369B
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
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- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/08—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/09—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton the carbon skeleton being further substituted by at least two halogen atoms
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- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
- C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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- C07C311/22—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms
- C07C311/29—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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- C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C317/34—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
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- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/46—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having at least one of the nitrogen atoms, not being part of nitro or nitroso groups, further bound to other hetero atoms
- C07C323/49—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having at least one of the nitrogen atoms, not being part of nitro or nitroso groups, further bound to other hetero atoms to sulfur atoms
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
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- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
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- C07D277/62—Benzothiazoles
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- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
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- Chemical & Material Sciences (AREA)
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Quinoline Compounds (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US14167299P | 1999-06-30 | 1999-06-30 | |
| US60/141,672 | 1999-06-30 | ||
| PCT/US2000/018178 WO2001000579A1 (en) | 1999-06-30 | 2000-06-28 | COMPOUNDS FOR THE MODULATION OF PPARη ACTIVITY |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HK1043369A1 HK1043369A1 (en) | 2002-09-13 |
| HK1043369B true HK1043369B (en) | 2014-06-13 |
Family
ID=22496697
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK02105143.3A HK1043369B (en) | 1999-06-30 | 2000-06-28 | Compounds for the modulation of ppar-gamma activity |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP1192137B1 (enExample) |
| JP (1) | JP4295458B2 (enExample) |
| CN (1) | CN1171872C (enExample) |
| CA (1) | CA2377309C (enExample) |
| DK (1) | DK1192137T3 (enExample) |
| EA (1) | EA004887B1 (enExample) |
| ES (1) | ES2437103T3 (enExample) |
| HK (1) | HK1043369B (enExample) |
| IL (2) | IL147308A0 (enExample) |
| MX (2) | MXPA01013199A (enExample) |
| NZ (2) | NZ530833A (enExample) |
| SG (1) | SG148834A1 (enExample) |
| WO (1) | WO2001000579A1 (enExample) |
| ZA (1) | ZA200200057B (enExample) |
Families Citing this family (68)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6583157B2 (en) | 1998-01-29 | 2003-06-24 | Tularik Inc. | Quinolinyl and benzothiazolyl modulators |
| US7041691B1 (en) | 1999-06-30 | 2006-05-09 | Amgen Inc. | Compounds for the modulation of PPARγ activity |
| US6653332B2 (en) | 2000-05-03 | 2003-11-25 | Tularik Inc. | Combination therapeutic compositions and method of use |
| HUP0301482A3 (en) * | 2000-06-28 | 2005-12-28 | Japan Tobacco Inc | Quinolinnyl and benzothiazolyl ppar-gamma modulators pharmaceutical compositions containing them and their use |
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-
2000
- 2000-06-28 HK HK02105143.3A patent/HK1043369B/en unknown
- 2000-06-28 EP EP00946961.0A patent/EP1192137B1/en not_active Expired - Lifetime
- 2000-06-28 EA EA200200105A patent/EA004887B1/ru not_active IP Right Cessation
- 2000-06-28 NZ NZ530833A patent/NZ530833A/en not_active IP Right Cessation
- 2000-06-28 CN CNB008113076A patent/CN1171872C/zh not_active Expired - Lifetime
- 2000-06-28 IL IL14730800A patent/IL147308A0/xx unknown
- 2000-06-28 NZ NZ516455A patent/NZ516455A/xx not_active IP Right Cessation
- 2000-06-28 CA CA2377309A patent/CA2377309C/en not_active Expired - Lifetime
- 2000-06-28 SG SG200403480-7A patent/SG148834A1/en unknown
- 2000-06-28 WO PCT/US2000/018178 patent/WO2001000579A1/en not_active Ceased
- 2000-06-28 DK DK00946961.0T patent/DK1192137T3/da active
- 2000-06-28 ES ES00946961.0T patent/ES2437103T3/es not_active Expired - Lifetime
- 2000-06-28 JP JP2001506989A patent/JP4295458B2/ja not_active Expired - Lifetime
- 2000-06-28 MX MXPA01013199A patent/MXPA01013199A/es active IP Right Grant
-
2001
- 2001-12-18 MX MX2011005852A patent/MX339420B/es unknown
- 2001-12-25 IL IL147308A patent/IL147308A/en active IP Right Grant
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- 2002-01-03 ZA ZA200200057A patent/ZA200200057B/en unknown
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| Publication number | Publication date |
|---|---|
| IL147308A (en) | 2015-06-30 |
| IL147308A0 (en) | 2002-08-14 |
| JP2003503387A (ja) | 2003-01-28 |
| MXPA01013199A (es) | 2003-08-20 |
| CA2377309A1 (en) | 2001-01-04 |
| CN1171872C (zh) | 2004-10-20 |
| EA200200105A1 (ru) | 2002-06-27 |
| ZA200200057B (en) | 2003-03-19 |
| EP1192137B1 (en) | 2013-10-23 |
| WO2001000579A1 (en) | 2001-01-04 |
| SG148834A1 (en) | 2009-01-29 |
| HK1043369A1 (en) | 2002-09-13 |
| EP1192137A1 (en) | 2002-04-03 |
| EA004887B1 (ru) | 2004-08-26 |
| CN1368961A (zh) | 2002-09-11 |
| ES2437103T3 (es) | 2014-01-08 |
| DK1192137T3 (da) | 2013-11-11 |
| MX339420B (es) | 2016-05-25 |
| NZ516455A (en) | 2004-03-26 |
| CA2377309C (en) | 2010-11-23 |
| JP4295458B2 (ja) | 2009-07-15 |
| NZ530833A (en) | 2005-08-26 |
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