GR861762B - Method for the preparation of stable peroral medicine containing 9-deoxo-11-deoxy-9,11-(imino (2-(2-methoxy ethoxy) ethyliden)-oxy)-(9s) erythromycin - Google Patents

Method for the preparation of stable peroral medicine containing 9-deoxo-11-deoxy-9,11-(imino (2-(2-methoxy ethoxy) ethyliden)-oxy)-(9s) erythromycin

Info

Publication number
GR861762B
GR861762B GR861762A GR860101762A GR861762B GR 861762 B GR861762 B GR 861762B GR 861762 A GR861762 A GR 861762A GR 860101762 A GR860101762 A GR 860101762A GR 861762 B GR861762 B GR 861762B
Authority
GR
Greece
Prior art keywords
deoxo
erythromycin
deoxy
imino
oxy
Prior art date
Application number
GR861762A
Other languages
English (en)
Inventor
Etienne Alain
Gruber Dr Peter
Busch Dr Ulrich
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of GR861762B publication Critical patent/GR861762B/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1611Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
GR861762A 1985-07-10 1986-07-07 Method for the preparation of stable peroral medicine containing 9-deoxo-11-deoxy-9,11-(imino (2-(2-methoxy ethoxy) ethyliden)-oxy)-(9s) erythromycin GR861762B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19853524572 DE3524572A1 (de) 1985-07-10 1985-07-10 Feste arzneimittelformen zur peroralen anwendung enthaltend 9-deoxo-11-deoxy-9,11-(imino(2-(2-methoxyethoxy)ethyliden)-oxy)-(9s)-erythromycin und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
GR861762B true GR861762B (en) 1986-11-10

Family

ID=6275375

Family Applications (1)

Application Number Title Priority Date Filing Date
GR861762A GR861762B (en) 1985-07-10 1986-07-07 Method for the preparation of stable peroral medicine containing 9-deoxo-11-deoxy-9,11-(imino (2-(2-methoxy ethoxy) ethyliden)-oxy)-(9s) erythromycin

Country Status (25)

Country Link
US (1) US4755385A (el)
EP (1) EP0208971B1 (el)
JP (1) JPH0688905B2 (el)
KR (1) KR930010586B1 (el)
AT (1) ATE63819T1 (el)
AU (1) AU586262B2 (el)
CA (1) CA1271138A (el)
DD (1) DD248057A5 (el)
DE (2) DE3524572A1 (el)
DK (1) DK165670C (el)
ES (1) ES2000269A6 (el)
FI (1) FI85649C (el)
GR (1) GR861762B (el)
HK (1) HK79791A (el)
HU (1) HU195730B (el)
IE (1) IE58951B1 (el)
IL (1) IL79375A (el)
MX (1) MX9202785A (el)
NL (1) NL970004I2 (el)
NO (1) NO175351C (el)
NZ (1) NZ216794A (el)
PH (1) PH26147A (el)
PT (1) PT82949B (el)
SG (1) SG72191G (el)
ZA (1) ZA865105B (el)

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HU217629B (hu) * 1991-12-12 2000-03-28 Novartis Ag. Eljárás fluvasztatint tartalmazó stabilizált gyógyszerkészítmények előállítására
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JP4040084B2 (ja) * 1994-02-16 2008-01-30 アボツト・ラボラトリーズ 微粒子医薬調合物の調製プロセス
MX9605419A (es) * 1994-05-06 1997-12-31 Pfizer Formas de dosificacion de liberacion controlada de azitromicina.
US5853787A (en) * 1995-12-22 1998-12-29 Tamer International Method for reducing coffee acidity
US6045843A (en) * 1995-12-22 2000-04-04 Tamer International, Inc. Acid-reduced, whole bean coffee process
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US6066342A (en) * 1995-12-22 2000-05-23 Tamer International, Ltd. Antacid composition
BE1011045A3 (fr) * 1997-03-14 1999-04-06 Ucb Sa Compositions pharmaceutiques pour la liberation controlee de substances actives.
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PT1187601E (pt) * 1999-06-07 2005-11-30 Altana Pharma Ag Nova forma de preparacao e a administracao compreendendo um inibidor da bomba de protoes instavel em meio acido
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EP1118321A1 (fr) * 2000-01-14 2001-07-25 Ucb, S.A. Compositions pharmaceutiques solides pour la libération contrôlée de substances actives
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US6565882B2 (en) 2000-02-24 2003-05-20 Advancis Pharmaceutical Corp Antibiotic composition with inhibitor
US6242003B1 (en) 2000-04-13 2001-06-05 Novartis Ag Organic compounds
MXPA03000082A (es) * 2000-06-28 2004-07-08 Procter & Gamble Estructuras y composiciones que aumentan la estabilidad de los ingredientes activos de peroxido.
US20020068078A1 (en) 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
US6541014B2 (en) 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US20060127474A1 (en) * 2001-04-11 2006-06-15 Oskar Kalb Pharmaceutical compositions comprising fluvastatin
US6949240B2 (en) * 2002-05-23 2005-09-27 The Procter & Gamble Company Tooth whitening products
US8524200B2 (en) 2002-09-11 2013-09-03 The Procter & Gamble Company Tooth whitening products
AU2004258953B2 (en) 2003-07-21 2011-02-10 Shionogi, Inc. Antibiotic product, use and formulation thereof
AU2004258949B2 (en) 2003-07-21 2011-02-10 Shionogi, Inc. Antibiotic product, use and formulation thereof
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JP2009515993A (ja) * 2005-11-17 2009-04-16 ノバルティス アクチエンゲゼルシャフト 医薬組成物
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Also Published As

Publication number Publication date
MX9202785A (es) 1992-06-30
DE3524572A1 (de) 1987-01-15
KR870000920A (ko) 1987-03-10
NL970004I1 (nl) 1997-04-01
IL79375A (en) 1990-01-18
PT82949A (de) 1986-08-01
NO175351B (no) 1994-06-27
AU5987686A (en) 1987-01-15
AU586262B2 (en) 1989-07-06
DK165670C (da) 1993-06-07
DK324786A (da) 1987-01-11
EP0208971A3 (en) 1988-01-27
JPS6212717A (ja) 1987-01-21
IE58951B1 (en) 1993-12-01
HU195730B (en) 1988-07-28
HUT42945A (en) 1987-09-28
PT82949B (pt) 1989-01-30
CA1271138A (en) 1990-07-03
DD248057A5 (de) 1987-07-29
FI862898A (fi) 1987-01-11
FI862898A0 (fi) 1986-07-10
EP0208971A2 (de) 1987-01-21
DK165670B (da) 1993-01-04
DK324786D0 (da) 1986-07-08
ZA865105B (en) 1988-03-30
EP0208971B1 (de) 1991-05-29
IE861842L (en) 1987-01-10
JPH0688905B2 (ja) 1994-11-09
NZ216794A (en) 1988-11-29
NL970004I2 (nl) 1997-06-02
NO862772D0 (no) 1986-07-09
ES2000269A6 (es) 1988-02-01
US4755385A (en) 1988-07-05
FI85649C (fi) 1992-05-25
SG72191G (en) 1991-11-22
PH26147A (en) 1992-03-18
NO862772L (no) 1987-01-12
FI85649B (fi) 1992-02-14
ATE63819T1 (de) 1991-06-15
DE3679463D1 (de) 1991-07-04
IL79375A0 (en) 1986-10-31
KR930010586B1 (ko) 1993-10-30
NO175351C (no) 1994-10-05
HK79791A (en) 1991-10-18

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